| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
A new metabotropic glutamate receptor agonist with in vivo anti-allodynic activity
|
Stanley, Nathan J.
|
|
2010
|
18 |
16 |
p. 6089-6098
10 p.
|
artikel
|
| 2 |
Anhydrotetracycline–peptide conjugates as representatives for ligand-based transactivating systems
|
Lochner, Susanne
|
|
2010
|
18 |
16 |
p. 6127-6133
7 p.
|
artikel
|
| 3 |
Anti-HIV and antiplasmodial activity of original flavonoid derivatives
|
Casano, Gilles
|
|
2010
|
18 |
16 |
p. 6012-6023
12 p.
|
artikel
|
| 4 |
Anti-Plasmodium activity of imidazolium and triazolium salts
|
Vlahakis, Jason Z.
|
|
2010
|
18 |
16 |
p. 6184-6196
13 p.
|
artikel
|
| 5 |
A simple procedure for the derivation of electron density based surfaces of drug-receptor complexes from a combination of X-ray data and theoretical calculations
|
Mebs, Stefan
|
|
2010
|
18 |
16 |
p. 5965-5974
10 p.
|
artikel
|
| 6 |
Bioorganic & Medicinal Chemistry Reviews and Perspectives
|
|
|
2010
|
18 |
16 |
p. I-III
nvt p.
|
artikel
|
| 7 |
Characterization of new PPARγ agonists: Benzimidazole derivatives—importance of positions 5 and 6, and computational studies on the binding mode
|
Goebel, Matthias
|
|
2010
|
18 |
16 |
p. 5885-5895
11 p.
|
artikel
|
| 8 |
CLEFMA—An anti-proliferative curcuminoid from structure–activity relationship studies on 3,5-bis(benzylidene)-4-piperidones
|
Lagisetty, Pallavi
|
|
2010
|
18 |
16 |
p. 6109-6120
12 p.
|
artikel
|
| 9 |
Comparison of MRI properties between derivatized DTPA and DOTA gadolinium–dendrimer conjugates
|
Nwe, K.
|
|
2010
|
18 |
16 |
p. 5925-5931
7 p.
|
artikel
|
| 10 |
Concise synthesis of 5,6-dihydrovaltrate leading to enhanced Rev-export inhibitory congener
|
Tamura, Satoru
|
|
2010
|
18 |
16 |
p. 5975-5980
6 p.
|
artikel
|
| 11 |
Design, synthesis, and anticonvulsant activity of new N-Mannich bases derived from spirosuccinimides and spirohydantoins
|
Obniska, Jolanta
|
|
2010
|
18 |
16 |
p. 6134-6142
9 p.
|
artikel
|
| 12 |
Design, synthesis, and biological evaluation of ketoprofen analogs as potent cyclooxygenase-2 inhibitors
|
Zarghi, Afshin
|
|
2010
|
18 |
16 |
p. 5855-5860
6 p.
|
artikel
|
| 13 |
Design, synthesis, and biological evaluation of prenylated chalcones as 5-LOX inhibitors
|
Reddy, Nimmanapalli P.
|
|
2010
|
18 |
16 |
p. 5807-5815
9 p.
|
artikel
|
| 14 |
Dimethylaminopyridine derivatives of lupane triterpenoids are potent disruptors of mitochondrial structure and function
|
Holy, Jon
|
|
2010
|
18 |
16 |
p. 6080-6088
9 p.
|
artikel
|
| 15 |
8,8-Dimethyldihydroberberine with improved bioavailability and oral efficacy on obese and diabetic mouse models
|
Cheng, Zhe
|
|
2010
|
18 |
16 |
p. 5915-5924
10 p.
|
artikel
|
| 16 |
Dual inhibitors of inosine monophosphate dehydrogenase and histone deacetylase based on a cinnamic hydroxamic acid core structure
|
Chen, Liqiang
|
|
2010
|
18 |
16 |
p. 5950-5964
15 p.
|
artikel
|
| 17 |
Editorial board
|
|
|
2010
|
18 |
16 |
p. IFC-
1 p.
|
artikel
|
| 18 |
Efficient synthesis and biological evaluation of demethyl geranylgeranoic acid derivatives
|
Wada, Akimori
|
|
2010
|
18 |
16 |
p. 5795-5806
12 p.
|
artikel
|
| 19 |
Functional profiling of p53-binding sites in Hdm2 and Hdmx using a genetic selection system
|
Datta, Shreya
|
|
2010
|
18 |
16 |
p. 6099-6108
10 p.
|
artikel
|
| 20 |
Further optimization of novel pyrrole 3-carboxamides for targeting serotonin 5-HT2A, 5-HT2C, and the serotonin transporter as a potential antidepressant
|
Kang, Suk Youn
|
|
2010
|
18 |
16 |
p. 6156-6169
14 p.
|
artikel
|
| 21 |
Graphical contents list
|
|
|
2010
|
18 |
16 |
p. 5763-5774
12 p.
|
artikel
|
| 22 |
Improved inhibition of the histone acetyltransferase PCAF by an anacardic acid derivative
|
Ghizzoni, Massimo
|
|
2010
|
18 |
16 |
p. 5826-5834
9 p.
|
artikel
|
| 23 |
Inactivation of protein tyrosine phosphatases by oltipraz and other cancer chemopreventive 1,2-dithiole-3-thiones
|
Bhattacharyya, Sanjib
|
|
2010
|
18 |
16 |
p. 5945-5949
5 p.
|
artikel
|
| 24 |
Intramolecular acyl migration and enzymatic hydrolysis of a novel monoacylated ascorbic acid derivative, 6-O-dodecanoyl-2-O-α-d-glucopyranosyl-l-ascorbic acid
|
Tai, Akihiro
|
|
2010
|
18 |
16 |
p. 6179-6183
5 p.
|
artikel
|
| 25 |
In vitro ADMET and physicochemical investigations of poly-N-methylated peptides designed to inhibit Aβ aggregation
|
Bose, Partha Pratim
|
|
2010
|
18 |
16 |
p. 5896-5902
7 p.
|
artikel
|
| 26 |
Large flanking sequence effects in single nucleotide mismatch detection using fluorescent nucleoside Çf
|
Gardarsson, Haraldur
|
|
2010
|
18 |
16 |
p. 6121-6126
6 p.
|
artikel
|
| 27 |
Lipophilic phenolic antioxidants: Correlation between antioxidant profile, partition coefficients and redox properties
|
Roleira, Fernanda M.F.
|
|
2010
|
18 |
16 |
p. 5816-5825
10 p.
|
artikel
|
| 28 |
Multipotent drugs with cholinergic and neuroprotective properties for the treatment of Alzheimer and neuronal vascular diseases. I. Synthesis, biological assessment, and molecular modeling of simple and readily available 2-aminopyridine-, and 2-chloropyridine-3,5-dicarbonitriles
|
Samadi, Abdelouahid
|
|
2010
|
18 |
16 |
p. 5861-5872
12 p.
|
artikel
|
| 29 |
Natural and semisynthetic azaphilones as a new scaffold for Hsp90 inhibitors
|
Musso, Loana
|
|
2010
|
18 |
16 |
p. 6031-6043
13 p.
|
artikel
|
| 30 |
New bioactive halenaquinone derivatives from South Pacific marine sponges of the genus Xestospongia
|
Longeon, Arlette
|
|
2010
|
18 |
16 |
p. 6006-6011
6 p.
|
artikel
|
| 31 |
New N-(phenoxydecyl)phthalimide derivatives displaying potent inhibition activity towards α-glucosidase
|
Pascale, Rossana
|
|
2010
|
18 |
16 |
p. 5903-5914
12 p.
|
artikel
|
| 32 |
New porphyrin amino acid conjugates: Synthesis and photodynamic effect in human epithelial cells
|
Serra, V. Vaz
|
|
2010
|
18 |
16 |
p. 6170-6178
9 p.
|
artikel
|
| 33 |
NMR spectroscopy and computational analysis of interaction between Serratia marcescens chitinase B and a dipeptide derived from natural-product cyclopentapeptide chitinase inhibitor argifin
|
Gouda, Hiroaki
|
|
2010
|
18 |
16 |
p. 5835-5844
10 p.
|
artikel
|
| 34 |
Novel aminopeptidase N (APN/CD13) inhibitors derived from 3-phenylalanyl-N′-substituted-2,6-piperidinedione
|
Zhang, Xiaopan
|
|
2010
|
18 |
16 |
p. 5981-5987
7 p.
|
artikel
|
| 35 |
Novel antifungal agents: Triazolopyridines as inhibitors of β-1,6-glucan synthesis
|
Kuroyanagi, Jun-ichi
|
|
2010
|
18 |
16 |
p. 5845-5854
10 p.
|
artikel
|
| 36 |
Phenolic constituents isolated from Fragaria ananassa Duch. inhibit antigen-stimulated degranulation through direct inhibition of spleen tyrosine kinase activation
|
Ninomiya, Masayuki
|
|
2010
|
18 |
16 |
p. 5932-5937
6 p.
|
artikel
|
| 37 |
Process R&D under the magnifying glass: Organization, business model, challenges, and scientific context
|
Federsel, Hans-Jürgen
|
|
2010
|
18 |
16 |
p. 5775-5794
20 p.
|
artikel
|
| 38 |
Role of 2′,6′-dimethyl-l-tyrosine (Dmt) in some opioid lead compounds
|
Balboni, Gianfranco
|
|
2010
|
18 |
16 |
p. 6024-6030
7 p.
|
artikel
|
| 39 |
Synergistic experimental/computational studies on arylazoenamine derivatives that target the bovine viral diarrhea virus RNA-dependent RNA polymerase
|
Giliberti, Gabriele
|
|
2010
|
18 |
16 |
p. 6055-6068
14 p.
|
artikel
|
| 40 |
Syntheses and pharmacological characterization of novel thiazole derivatives as potential mGluR5 PET ligands
|
Baumann, Cindy A.
|
|
2010
|
18 |
16 |
p. 6044-6054
11 p.
|
artikel
|
| 41 |
Synthesis and anti-hepatitis C virus activity of novel ethyl 1H-indole-3-carboxylates in vitro
|
Sellitto, Grazia
|
|
2010
|
18 |
16 |
p. 6143-6148
6 p.
|
artikel
|
| 42 |
Synthesis, and biological evaluation of 2-(4-aminophenyl)benzothiazole derivatives as photosensitizing agents
|
Hu, Wan-Ping
|
|
2010
|
18 |
16 |
p. 6197-6207
11 p.
|
artikel
|
| 43 |
Synthesis and biological evaluation of tetracyclic fluoroquinolones as antibacterial and anticancer agents
|
Al-Trawneh, Salah A.
|
|
2010
|
18 |
16 |
p. 5873-5884
12 p.
|
artikel
|
| 44 |
Synthesis and T-type calcium channel blocking activity of novel diphenylpiperazine compounds, and evaluation of in vivo analgesic activity
|
Kam, Yoo Lim
|
|
2010
|
18 |
16 |
p. 5938-5944
7 p.
|
artikel
|
| 45 |
Synthesis of aryl-heteroaryl ureas (AHUs) based on 4-aminoquinoline and their evaluation against the insulin-like growth factor receptor (IGF-1R)
|
Engen, William
|
|
2010
|
18 |
16 |
p. 5995-6005
11 p.
|
artikel
|
| 46 |
Synthesis of novel 3,5-diaryl pyrazole derivatives using combinatorial chemistry as inhibitors of tyrosinase as well as potent anticancer, anti-inflammatory agents
|
Bandgar, Babasaheb P.
|
|
2010
|
18 |
16 |
p. 6149-6155
7 p.
|
artikel
|
| 47 |
Synthesis of pyridazine and thiazole analogs as SGLT2 inhibitors
|
Kang, Suk Youn
|
|
2010
|
18 |
16 |
p. 6069-6079
11 p.
|
artikel
|
| 48 |
The marine sponge metabolite mycothiazole: A novel prototype mitochondrial complex I inhibitor
|
Morgan, J. Brian
|
|
2010
|
18 |
16 |
p. 5988-5994
7 p.
|
artikel
|
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