| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
2-Acylamino-4,6-diphenylpyridine derivatives as novel GPR54 antagonists with good brain exposure and in vivo efficacy for plasma LH level in male rats
|
Kobayashi, Toshitake
|
|
2010
|
18 |
14 |
p. 5157-5171
15 p.
|
artikel
|
| 2 |
An integrative in silico methodology for the identification of modulators of macrophage migration inhibitory factor (MIF) tautomerase activity
|
El Turk, Farah
|
|
2010
|
18 |
14 |
p. 5425-5440
16 p.
|
artikel
|
| 3 |
A novel achiral seco-cyclopropylpyrido[e]indolone (CPyI) analog of CC-1065 and the duocarmycins: Synthesis, DNA interactions, in vivo anticancer and anti-parasitic evaluation
|
Chavda, Sameer
|
|
2010
|
18 |
14 |
p. 5016-5024
9 p.
|
artikel
|
| 4 |
Anti-influenza activity of phenethylphenylphthalimide analogs derived from thalidomide
|
Iwai, Yuma
|
|
2010
|
18 |
14 |
p. 5379-5390
12 p.
|
artikel
|
| 5 |
Antineoplastic agents 582. Part 1: Isolation and structure of a cyclobutane-type sesquiterpene cancer cell growth inhibitor from Coprinus cinereus (Coprinaceae)
|
Pettit, George R.
|
|
2010
|
18 |
14 |
p. 4879-4883
5 p.
|
artikel
|
| 6 |
Callyaerins A–F and H, new cytotoxic cyclic peptides from the Indonesian marine sponge Callyspongia aerizusa
|
Ibrahim, Sabrin R.M.
|
|
2010
|
18 |
14 |
p. 4947-4956
10 p.
|
artikel
|
| 7 |
Cell-penetration by Co(III)cyclen-based peptide-cleaving catalysts selective for pathogenic proteins of amyloidoses
|
Chei, Woo Suk
|
|
2010
|
18 |
14 |
p. 5248-5253
6 p.
|
artikel
|
| 8 |
Characterization of multivalent lactose quantum dots and its application in carbohydrate–protein interactions study and cell imaging
|
Yang, Yang
|
|
2010
|
18 |
14 |
p. 5234-5240
7 p.
|
artikel
|
| 9 |
Constrained peptidomimetics as antiplasmodial falcipain-2 inhibitors
|
Bova, Floriana
|
|
2010
|
18 |
14 |
p. 4928-4938
11 p.
|
artikel
|
| 10 |
Coumarinyl-substituted sulfonamides strongly inhibit several human carbonic anhydrase isoforms: solution and crystallographic investigations
|
Wagner, Jason
|
|
2010
|
18 |
14 |
p. 4873-4878
6 p.
|
artikel
|
| 11 |
Design and synthesis of novel benzimidazole derivatives as inhibitors of hepatitis B virus
|
Luo, Yu
|
|
2010
|
18 |
14 |
p. 5048-5055
8 p.
|
artikel
|
| 12 |
Design, synthesis, and biological evaluation of resveratrol analogues as aromatase and quinone reductase 2 inhibitors for chemoprevention of cancer
|
Sun, Bin
|
|
2010
|
18 |
14 |
p. 5352-5366
15 p.
|
artikel
|
| 13 |
Design, synthesis and evaluation of 2-amino-4-m-bromoanilino-6-arylmethyl-7H-pyrrolo[2,3-d]pyrimidines as tyrosine kinase inhibitors and antiangiogenic agents 1
|
Gangjee, Aleem
|
|
2010
|
18 |
14 |
p. 5261-5273
13 p.
|
artikel
|
| 14 |
Development and evaluation of a 68Ga labeled pamoic acid derivative for in vivo visualization of necrosis using positron emission tomography
|
Prinsen, Kristof
|
|
2010
|
18 |
14 |
p. 5274-5281
8 p.
|
artikel
|
| 15 |
Development of a new radioligand for cholecystokinin receptor subtype 2 scintigraphy: From molecular modeling to in vivo evaluation
|
Brillouet, Séverine
|
|
2010
|
18 |
14 |
p. 5400-5412
13 p.
|
artikel
|
| 16 |
Development of chemical probes: Toward the mode of action of a methylene-linked di(aryl acetate) E1
|
Smith, Mark E.B.
|
|
2010
|
18 |
14 |
p. 4917-4927
11 p.
|
artikel
|
| 17 |
Development of tryptase inhibitors derived from thalidomide
|
Tetsuhashi, Masashi
|
|
2010
|
18 |
14 |
p. 5323-5338
16 p.
|
artikel
|
| 18 |
Discovery of orally available spirodiketopiperazine-based CCR5 antagonists
|
Nishizawa, Rena
|
|
2010
|
18 |
14 |
p. 5208-5223
16 p.
|
artikel
|
| 19 |
Discovery of potent and orally active tricyclic-based FBPase inhibitors
|
Tsukada, Tomoharu
|
|
2010
|
18 |
14 |
p. 5346-5351
6 p.
|
artikel
|
| 20 |
Editorial board
|
|
|
2010
|
18 |
14 |
p. IFC-
1 p.
|
artikel
|
| 21 |
Evaluation of N-substitution in 6,7-benzomorphan compounds
|
Pasquinucci, Lorella
|
|
2010
|
18 |
14 |
p. 4975-4982
8 p.
|
artikel
|
| 22 |
Graphical contents list
|
|
|
2010
|
18 |
14 |
p. 4855-4871
17 p.
|
artikel
|
| 23 |
1H-1,2,3-Triazol-1-yl thiodigalactoside derivatives as high affinity galectin-3 inhibitors
|
Salameh, Bader A.
|
|
2010
|
18 |
14 |
p. 5367-5378
12 p.
|
artikel
|
| 24 |
Hybrid diarylbenzopyrimidine non-nucleoside reverse transcriptase inhibitors as promising new leads for improved anti-HIV-1 chemotherapy
|
Zeng, Zhao-Sen
|
|
2010
|
18 |
14 |
p. 5039-5047
9 p.
|
artikel
|
| 25 |
Hypoxic selectivity and solubility—investigating the properties of A-ring substituted nitro seco-1,2,9,9a-tetrahydrocyclopropa[c]benz[e]indol-4-ones (nitroCBIs) as hypoxia-activated prodrugs for antitumor therapy
|
Tercel, Moana
|
|
2010
|
18 |
14 |
p. 4997-5006
10 p.
|
artikel
|
| 26 |
Identification and evaluation of apoptotic compounds from Garcinia paucinervis
|
Gao, Xue-Mei
|
|
2010
|
18 |
14 |
p. 4957-4964
8 p.
|
artikel
|
| 27 |
Identification of chalcones as in vivo liver monofunctional phase II enzymes inducers
|
Cabrera, Mauricio
|
|
2010
|
18 |
14 |
p. 5391-5399
9 p.
|
artikel
|
| 28 |
Identification of novel bacterial histidine biosynthesis inhibitors using docking, ensemble rescoring, and whole-cell assays
|
Henriksen, S.T.
|
|
2010
|
18 |
14 |
p. 5148-5156
9 p.
|
artikel
|
| 29 |
Identification of novel inhibitors for a low molecular weight protein tyrosine phosphatase via virtual screening
|
Homan, Kristoff T.
|
|
2010
|
18 |
14 |
p. 5449-5456
8 p.
|
artikel
|
| 30 |
Improved P2 phenylglycine-based hepatitis C virus NS3 protease inhibitors with alkenylic prime-side substituents
|
Lampa, Anna
|
|
2010
|
18 |
14 |
p. 5413-5424
12 p.
|
artikel
|
| 31 |
Morphinans and isoquinolines: Acetylcholinesterase inhibition, pharmacophore modeling, and interaction with opioid receptors
|
Schuster, Daniela
|
|
2010
|
18 |
14 |
p. 5071-5080
10 p.
|
artikel
|
| 32 |
New antimalarials with a triterpenic scaffold from Momordica balsamina
|
Ramalhete, Cátia
|
|
2010
|
18 |
14 |
p. 5254-5260
7 p.
|
artikel
|
| 33 |
New 2-arylnaphthalenediols and triol inhibitors of HIV-1 integrase—Discovery of a new polyhydroxylated antiviral agent
|
Maurin, Cédric
|
|
2010
|
18 |
14 |
p. 5194-5201
8 p.
|
artikel
|
| 34 |
(−)-N-Formylanonaine from Michelia alba as a human tyrosinase inhibitor and antioxidant
|
Wang, Hui-Min
|
|
2010
|
18 |
14 |
p. 5241-5247
7 p.
|
artikel
|
| 35 |
Novel antimicrobial peptides that exhibit activity against select agents and other drug resistant bacteria
|
Venugopal, Divakaramenon
|
|
2010
|
18 |
14 |
p. 5137-5147
11 p.
|
artikel
|
| 36 |
Novel anti-viability ceramide analogs: Design, synthesis, and structure–activity relationship studies of substituted (S)-2-(benzylideneamino)-3-hydroxy-N-tetradecylpropanamides
|
Liu, Jiawang
|
|
2010
|
18 |
14 |
p. 5316-5322
7 p.
|
artikel
|
| 37 |
Novel structure–activity relationships and selectivity profiling of cage dimeric 1,4-dihydropyridines as multidrug resistance (MDR) modulators
|
Coburger, Claudius
|
|
2010
|
18 |
14 |
p. 4983-4990
8 p.
|
artikel
|
| 38 |
2-Phenyl-1-[4-(2-piperidine-1-yl-ethoxy)benzyl]-1H-benzimidazoles as ligands for the estrogen receptor: Synthesis and pharmacological evaluation
|
Dettmann, Sandra
|
|
2010
|
18 |
14 |
p. 4905-4916
12 p.
|
artikel
|
| 39 |
Pteridine–sulfonamide conjugates as dual inhibitors of carbonic anhydrases and dihydrofolate reductase with potential antitumor activity
|
Marques, Sérgio M.
|
|
2010
|
18 |
14 |
p. 5081-5089
9 p.
|
artikel
|
| 40 |
Publisher’s Note
|
|
|
2010
|
18 |
14 |
p. 4872-
1 p.
|
artikel
|
| 41 |
Spectroscopic characterization of the inclusion complexes of luteolin with native and derivatized β-cyclodextrin
|
Jullian, Carolina
|
|
2010
|
18 |
14 |
p. 5025-5031
7 p.
|
artikel
|
| 42 |
STD-NMR studies of two acceptor substrates of GlfT2, a galactofuranosyltransferase from Mycobacterium tuberculosis: Epitope mapping studies
|
Szczepina, Monica G.
|
|
2010
|
18 |
14 |
p. 5123-5128
6 p.
|
artikel
|
| 43 |
Structural characteristics of green tea catechins for formation of protein carbonyl in human serum albumin
|
Ishii, Takeshi
|
|
2010
|
18 |
14 |
p. 4892-4896
5 p.
|
artikel
|
| 44 |
Structure–activity relationship of brominated 3-alkyl-5-methylene-2(5H)-furanones and alkylmaleic anhydrides as inhibitors of Salmonella biofilm formation and quorum sensing regulated bioluminescence in Vibrio harveyi
|
Steenackers, Hans P.
|
|
2010
|
18 |
14 |
p. 5224-5233
10 p.
|
artikel
|
| 45 |
Studies on the anti-hepatitis C virus activity of newly synthesized tropolone derivatives: Identification of NS3 helicase inhibitors that specifically inhibit subgenomic HCV replication
|
Najda-Bernatowicz, Andżelika
|
|
2010
|
18 |
14 |
p. 5129-5136
8 p.
|
artikel
|
| 46 |
Substituted 2-(3′,4′,5′-trimethoxybenzoyl)-benzo[b]thiophene derivatives as potent tubulin polymerization inhibitors
|
Romagnoli, Romeo
|
|
2010
|
18 |
14 |
p. 5114-5122
9 p.
|
artikel
|
| 47 |
Syntheses and herbicidal activity of new triazolopyrimidine-2-sulfonamides as acetohydroxyacid synthase inhibitor
|
Chen, Chao-Nan
|
|
2010
|
18 |
14 |
p. 4897-4904
8 p.
|
artikel
|
| 48 |
Synthesis and antiproliferative evaluation of certain iminonaphtho[2,3-b]furan derivatives
|
Tseng, Chih-Hua
|
|
2010
|
18 |
14 |
p. 5172-5182
11 p.
|
artikel
|
| 49 |
Synthesis and biodistribution of [11C]A-836339, a new potential radioligand for PET imaging of cannabinoid type 2 receptors (CB2)
|
Horti, Andrew G.
|
|
2010
|
18 |
14 |
p. 5202-5207
6 p.
|
artikel
|
| 50 |
Synthesis and biological evaluation of cytotoxic activity of novel anthracene l-rhamnopyranosides
|
Song, Gaopeng
|
|
2010
|
18 |
14 |
p. 5183-5193
11 p.
|
artikel
|
| 51 |
Synthesis and biological study of 3-(phenylsulfonyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidines as potent and selective serotonin 5-HT6 receptor antagonists
|
Ivachtchenko, Alexandre V.
|
|
2010
|
18 |
14 |
p. 5282-5290
9 p.
|
artikel
|
| 52 |
Synthesis and characterization of selective dopamine D2 receptor antagonists. 2. Azaindole, benzofuran, and benzothiophene analogs of L-741,626
|
Vangveravong, Suwanna
|
|
2010
|
18 |
14 |
p. 5291-5300
10 p.
|
artikel
|
| 53 |
Synthesis and CYP24A1 inhibitory activity of N-(2-(1H-imidazol-1-yl)-2-phenylethyl)arylamides
|
Aboraia, Ahmed S.
|
|
2010
|
18 |
14 |
p. 4939-4946
8 p.
|
artikel
|
| 54 |
Synthesis and cytotoxic activity of a new potential DNA bisintercalator: 1,4-Bis{3-[N-(4-chlorobenzo[g]phthalazin-1-yl)aminopropyl]}piperazine
|
Galisteo, Juan
|
|
2010
|
18 |
14 |
p. 5301-5309
9 p.
|
artikel
|
| 55 |
Synthesis and pharmacological evaluation of pyrazine N-acylhydrazone derivatives designed as novel analgesic and anti-inflammatory drug candidates
|
Silva, Yolanda Karla Cupertino da
|
|
2010
|
18 |
14 |
p. 5007-5015
9 p.
|
artikel
|
| 56 |
Synthesis and structure–activity relationships of N-aryl-piperidine derivatives as potent (partial) agonists for human histamine H3 receptor
|
Ishikawa, Makoto
|
|
2010
|
18 |
14 |
p. 5441-5448
8 p.
|
artikel
|
| 57 |
Synthesis, molecular modeling, and biological evaluation of cinnamic acid metronidazole ester derivatives as novel anticancer agents
|
Qian, Yong
|
|
2010
|
18 |
14 |
p. 4991-4996
6 p.
|
artikel
|
| 58 |
Synthesis of 5-arylidene-2-amino-4-azolones and evaluation of their anticancer activity
|
Subtel’na, Ivanna
|
|
2010
|
18 |
14 |
p. 5090-5102
13 p.
|
artikel
|
| 59 |
Synthesis of a series of caffeic acid phenethyl amide (CAPA) fluorinated derivatives: Comparison of cytoprotective effects to caffeic acid phenethyl ester (CAPE)
|
Yang, John
|
|
2010
|
18 |
14 |
p. 5032-5038
7 p.
|
artikel
|
| 60 |
Synthesis of 5-deoxy-β-d-galactofuranosides as tools for the characterization of β-d-galactofuranosidases
|
Bordoni, Andrea
|
|
2010
|
18 |
14 |
p. 5339-5345
7 p.
|
artikel
|
| 61 |
Synthesis of novel pyrazolic analogues of chalcones and their 3-aryl-4-(3-aryl-4,5-dihydro-1H-pyrazol-5-yl)-1-phenyl-1H-pyrazole derivatives as potential antitumor agents
|
Insuasty, Braulio
|
|
2010
|
18 |
14 |
p. 4965-4974
10 p.
|
artikel
|
| 62 |
Synthesis, semipreparative HPLC separation, biological evaluation, and 3D-QSAR of hydrazothiazole derivatives as human monoamine oxidase B inhibitors
|
Chimenti, Franco
|
|
2010
|
18 |
14 |
p. 5063-5070
8 p.
|
artikel
|
| 63 |
Target-specific control of lymphoid-specific protein tyrosine phosphatase (Lyp) activity
|
Walton, Zandra E.
|
|
2010
|
18 |
14 |
p. 4884-4891
8 p.
|
artikel
|
| 64 |
Terpioside B, a difucosyl GSL from the marine sponge Terpios sp. is a potent inhibitor of NO release
|
Costantino, Valeria
|
|
2010
|
18 |
14 |
p. 5310-5315
6 p.
|
artikel
|
| 65 |
Tryptamine-derived alkaloids from Annonaceae exerting neurotrophin-like properties on primary dopaminergic neurons
|
Schmidt, Fanny
|
|
2010
|
18 |
14 |
p. 5103-5113
11 p.
|
artikel
|
| 66 |
Virtual fragment screening for novel inhibitors of 6-phosphogluconate dehydrogenase
|
Ruda, Gian Filippo
|
|
2010
|
18 |
14 |
p. 5056-5062
7 p.
|
artikel
|
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