| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
Alpneumines A–H, new anti-melanogenic indole alkaloids from Alstonia pneumatophora
|
Koyama, Koichiro
|
|
2010
|
18 |
12 |
p. 4415-4421
7 p.
|
artikel
|
| 2 |
A new class of potential anti-tuberculosis agents: Synthesis and preliminary evaluation of novel acrylic acid ethyl ester derivatives
|
Kabir, M. Shahjahan
|
|
2010
|
18 |
12 |
p. 4178-4186
9 p.
|
artikel
|
| 3 |
A novel and one-pot synthesis of new 1-tosyl pyrrol-2-one derivatives and analysis of carbonic anhydrase inhibitory potencies
|
Alp, Cemalettin
|
|
2010
|
18 |
12 |
p. 4468-4474
7 p.
|
artikel
|
| 4 |
Anti-AIDS agents 82: Synthesis of seco-(3′R,4′R)-3′,4′-di-O-(S)-camphanoyl-(+)-cis-khellactone (DCK) derivatives as novel anti-HIV agents
|
Tang, Jian
|
|
2010
|
18 |
12 |
p. 4363-4373
11 p.
|
artikel
|
| 5 |
Aromatic β-amino-ketone derivatives as novel selective non-steroidal progesterone receptor antagonists
|
Du, Yongli
|
|
2010
|
18 |
12 |
p. 4255-4268
14 p.
|
artikel
|
| 6 |
A statistical analysis of in vitro human microsomal metabolic stability of small phenyl group substituents, leading to improved design sets for parallel SAR exploration of a chemical series
|
Dossetter, Alexander G.
|
|
2010
|
18 |
12 |
p. 4405-4414
10 p.
|
artikel
|
| 7 |
Bacterial transferase MraY inhibitors: Synthesis and biological evaluation
|
Lecerclé, Delphine
|
|
2010
|
18 |
12 |
p. 4560-4569
10 p.
|
artikel
|
| 8 |
Controlled release of PEG chain from gold nanorods: Targeted delivery to tumor
|
Niidome, Takuro
|
|
2010
|
18 |
12 |
p. 4453-4458
6 p.
|
artikel
|
| 9 |
Corrigendum to “Identification and characterisation of 2-aminopyridine inhibitors of checkpoint kinase 2” [Bioorg. Med. Chem. 18 (2010) 707]
|
Hilton, Stephen
|
|
2010
|
18 |
12 |
p. 4591-
1 p.
|
artikel
|
| 10 |
Design and synthesis of spirotryprostatin-inspired diketopiperazine systems from prolyl spirooxoindolethiazolidine derivatives
|
Bertamino, Alessia
|
|
2010
|
18 |
12 |
p. 4328-4337
10 p.
|
artikel
|
| 11 |
Design, synthesis and antibacterial activity of novel andrographolide derivatives
|
Wang, Zhongli
|
|
2010
|
18 |
12 |
p. 4269-4274
6 p.
|
artikel
|
| 12 |
Design, synthesis, and biological evaluation of novel coxsackievirus B3 inhibitors
|
Šála, Michal
|
|
2010
|
18 |
12 |
p. 4374-4384
11 p.
|
artikel
|
| 13 |
Design, synthesis and biological evaluation of trans 2-(thiophen-2-yl)vinyl heteroaromatic iodides
|
Fortuna, Cosimo G.
|
|
2010
|
18 |
12 |
p. 4516-4523
8 p.
|
artikel
|
| 14 |
Design, synthesis, and docking of highly hypolipidemic agents: Schizosaccharomyces pombe as a new model for evaluating α-asarone-based HMG-CoA reductase inhibitors
|
Argüelles, Nancy
|
|
2010
|
18 |
12 |
p. 4238-4248
11 p.
|
artikel
|
| 15 |
Development of antiproliferative phenylmaleimides that activate the unfolded protein response
|
Muus, Ulrike
|
|
2010
|
18 |
12 |
p. 4535-4541
7 p.
|
artikel
|
| 16 |
Discovery of tetrahydro-β-carbolines as inhibitors of the mitotic kinesin KSP
|
Liu, Fei
|
|
2010
|
18 |
12 |
p. 4167-4177
11 p.
|
artikel
|
| 17 |
Editorial board
|
|
|
2010
|
18 |
12 |
p. IFC-
1 p.
|
artikel
|
| 18 |
(E)-2-Styrylchromones as potential anti-norovirus agents
|
Rocha-Pereira, Joana
|
|
2010
|
18 |
12 |
p. 4195-4201
7 p.
|
artikel
|
| 19 |
Graphical contents list
|
|
|
2010
|
18 |
12 |
p. 4155-4166
12 p.
|
artikel
|
| 20 |
Identification of csypyrone B1 as the novel product of Aspergillus oryzae type III polyketide synthase CsyB
|
Seshime, Yasuyo
|
|
2010
|
18 |
12 |
p. 4542-4546
5 p.
|
artikel
|
| 21 |
Identification of novel quinazolin-4(3H)-ones as inhibitors of thermolysin, the prototype of the M4 family of proteinases
|
Khan, Mahmud Tareq Hassan
|
|
2010
|
18 |
12 |
p. 4317-4327
11 p.
|
artikel
|
| 22 |
Identification of the three-dimensional pharmacophore of κ-opioid receptor agonists
|
Yamaotsu, Noriyuki
|
|
2010
|
18 |
12 |
p. 4446-4452
7 p.
|
artikel
|
| 23 |
New aryldithiolethione derivatives as potent histone deacetylase inhibitors
|
Tazzari, Valerio
|
|
2010
|
18 |
12 |
p. 4187-4194
8 p.
|
artikel
|
| 24 |
Novel analogues of Istaroxime, a potent inhibitor of Na+,K+-ATPase: Synthesis, structure–activity relationship and 3D-quantitative structure–activity relationship of derivatives at position 6 on the androstane scaffold
|
Gobbini, Mauro
|
|
2010
|
18 |
12 |
p. 4275-4299
25 p.
|
artikel
|
| 25 |
Novel pyrazole derivatives: Synthesis and evaluation of anti-angiogenic activity
|
Christodoulou, Michael S.
|
|
2010
|
18 |
12 |
p. 4338-4350
13 p.
|
artikel
|
| 26 |
Novel tricyclic Δ2-isoxazoline and 3-oxo-2-methyl-isoxazolidine derivatives: Synthesis and binding affinity at neuronal nicotinic acetylcholine receptor subtypes
|
Dallanoce, Clelia
|
|
2010
|
18 |
12 |
p. 4498-4508
11 p.
|
artikel
|
| 27 |
ortho-Substituted C-aryl glucosides as highly potent and selective renal sodium-dependent glucose co-transporter 2 (SGLT2) inhibitors
|
Xu, Baihua
|
|
2010
|
18 |
12 |
p. 4422-4432
11 p.
|
artikel
|
| 28 |
Peptide fragmentation as an approach in modeling of an active peptide and designing a competitive inhibitory peptide for HMG-CoA reductase
|
Pak, Valeriy V.
|
|
2010
|
18 |
12 |
p. 4300-4309
10 p.
|
artikel
|
| 29 |
Pharmacophore and structure–activity relationships of integrase inhibition within a dual inhibitor scaffold of HIV reverse transcriptase and integrase
|
Wang, Zhengqiang
|
|
2010
|
18 |
12 |
p. 4202-4211
10 p.
|
artikel
|
| 30 |
ppGpp analogues inhibit synthetase activity of Rel proteins from Gram-negative and Gram-positive bacteria
|
Wexselblatt, Ezequiel
|
|
2010
|
18 |
12 |
p. 4485-4497
13 p.
|
artikel
|
| 31 |
Selective angiotensin II AT2 receptor agonists with reduced CYP 450 inhibition
|
Mahalingam, A.K.
|
|
2010
|
18 |
12 |
p. 4570-4590
21 p.
|
artikel
|
| 32 |
Semi-synthetic analogues of thiostrepton delimit the critical nature of tail region modifications in the control of protein biosynthesis and antibacterial activity
|
Myers, Cullen L.
|
|
2010
|
18 |
12 |
p. 4231-4237
7 p.
|
artikel
|
| 33 |
Study of benzo[a]phenazine 7,12-dioxide as selective hypoxic cytotoxin-scaffold. Identification of aerobic-antitumoral activity through DNA fragmentation
|
Lavaggi, María Laura
|
|
2010
|
18 |
12 |
p. 4433-4440
8 p.
|
artikel
|
| 34 |
Synthesis and antitumor activity of 2,5-bis(3′-indolyl)-furans and 3,5-bis(3′-indolyl)-isoxazoles, nortopsentin analogues
|
Diana, Patrizia
|
|
2010
|
18 |
12 |
p. 4524-4529
6 p.
|
artikel
|
| 35 |
Synthesis and biological evaluation of a new series of berberine derivatives as dual inhibitors of acetylcholinesterase and butyrylcholinesterase
|
Huang, Ling
|
|
2010
|
18 |
12 |
p. 4475-4484
10 p.
|
artikel
|
| 36 |
Synthesis and biological evaluation of 4(5)-(6-methylpyridin-2-yl)imidazoles and -pyrazoles as transforming growth factor-β type 1 receptor kinase inhibitors
|
Kim, Dae-Kee
|
|
2010
|
18 |
12 |
p. 4459-4467
9 p.
|
artikel
|
| 37 |
Synthesis and biological evaluation of novel (4 or 5-aryl)pyrazolyl-indoles as inhibitors of interleukin-2 inducible T-cell kinase (ITK)
|
Velankar, Avdhoot D.
|
|
2010
|
18 |
12 |
p. 4547-4559
13 p.
|
artikel
|
| 38 |
Synthesis and characterization of N,N-dialkyl and N-alkyl-N-aralkyl fenpropimorph-derived compounds as high affinity ligands for sigma receptors
|
Hajipour, Abdol R.
|
|
2010
|
18 |
12 |
p. 4397-4404
8 p.
|
artikel
|
| 39 |
Synthesis and cytotoxicity of novel indirubin-5-carboxamides
|
Cheng, Xinlai
|
|
2010
|
18 |
12 |
p. 4509-4515
7 p.
|
artikel
|
| 40 |
Synthesis and evaluation of in vitro anticancer activity of some novel isopentenyladenosine derivatives
|
Ottria, Roberta
|
|
2010
|
18 |
12 |
p. 4249-4254
6 p.
|
artikel
|
| 41 |
Synthesis and in vitro antiprotozoal evaluation of substituted phenalenone analogues
|
Rosquete, Laura I.
|
|
2010
|
18 |
12 |
p. 4530-4534
5 p.
|
artikel
|
| 42 |
Synthesis and in vitro evaluation of novel 1,2,4-triazine derivatives as neuroprotective agents
|
Irannejad, Hamid
|
|
2010
|
18 |
12 |
p. 4224-4230
7 p.
|
artikel
|
| 43 |
Synthesis and structure–activity relationships of 1,2,3,4-tetrahydropyrido[2,3-b]pyrazines as potent and selective inhibitors of the anaplastic lymphoma kinase
|
Milkiewicz, Karen L.
|
|
2010
|
18 |
12 |
p. 4351-4362
12 p.
|
artikel
|
| 44 |
Synthesis and structure–activity relationship study of novel cytotoxic carbamate and N-acylheterocyclic bearing derivatives of betulin and betulinic acid
|
Santos, Rita C.
|
|
2010
|
18 |
12 |
p. 4385-4396
12 p.
|
artikel
|
| 45 |
Synthesis, molecular modeling and biological evaluation of dithiocarbamates as novel antitubulin agents
|
Qian, Yong
|
|
2010
|
18 |
12 |
p. 4310-4316
7 p.
|
artikel
|
| 46 |
Targeting efflux pumps—In vitro investigations with acridone derivatives and identification of a lead molecule for MDR modulation
|
Singh, Palwinder
|
|
2010
|
18 |
12 |
p. 4212-4223
12 p.
|
artikel
|
| 47 |
The scope of thallium nitrate oxidative cyclization of chalcones; synthesis and evaluation of isoflavone and aurone analogs for their inhibitory activity against interleukin-5
|
Thanigaimalai, P.
|
|
2010
|
18 |
12 |
p. 4441-4445
5 p.
|
artikel
|
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