| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
Acyclic nucleoside phosphonates with 5-azacytosine base moiety substituted in C-6 position
|
Krečmerová, Marcela
|
|
2010
|
18 |
1 |
p. 387-395
9 p.
|
artikel
|
| 2 |
3-(2-Aminocarbonylphenyl)propanoic acid analogs as potent and selective EP3 receptor antagonists. Part 1: Discovery and exploration of the carboxyamide side chain
|
Asada, Masaki
|
|
2010
|
18 |
1 |
p. 80-90
11 p.
|
artikel
|
| 3 |
Aminopyridinecarboxamide-based inhibitors: Structure–activity relationship
|
Bonafoux, Dominique F.
|
|
2010
|
18 |
1 |
p. 403-414
12 p.
|
artikel
|
| 4 |
Anti-inflammatory diterpenes from the seeds of Vitex negundo
|
Zheng, Cheng-Jian
|
|
2010
|
18 |
1 |
p. 175-181
7 p.
|
artikel
|
| 5 |
Antimalarial and antileishmanial activities of histone deacetylase inhibitors with triazole-linked cap group
|
Patil, Vishal
|
|
2010
|
18 |
1 |
p. 415-425
11 p.
|
artikel
|
| 6 |
Application of a novel [3+2] cycloaddition reaction to prepare substituted imidazoles and their use in the design of potent DFG-out allosteric B-Raf inhibitors
|
Dietrich, Justin
|
|
2010
|
18 |
1 |
p. 292-304
13 p.
|
artikel
|
| 7 |
Biotransformation of isoimperatorin and imperatorin by Glomerella cingulata and β-secretase inhibitory activity
|
Marumoto, Shinsuke
|
|
2010
|
18 |
1 |
p. 455-459
5 p.
|
artikel
|
| 8 |
Carbonic anhydrase inhibitors. Identification of selective inhibitors of the human mitochondrial isozymes VA and VB over the cytosolic isozymes I and II from a natural product-based phenolic library
|
Davis, Rohan A.
|
|
2010
|
18 |
1 |
p. 14-18
5 p.
|
artikel
|
| 9 |
Carboxymethylated-κ-casein: A convenient tool for the identification of polyphenolic inhibitors of amyloid fibril formation
|
Carver, John A.
|
|
2010
|
18 |
1 |
p. 222-228
7 p.
|
artikel
|
| 10 |
Corrigendum to “Design and synthesis of 4-methoxyphenylacetic acid esters as 15-lipoxygenase inhibitors and SAR comparative studies of them” [Bioorg. Med. Chem. 17 (2009) 2327]
|
Sadeghian, Hamid
|
|
2010
|
18 |
1 |
p. 462-
1 p.
|
artikel
|
| 11 |
Corrigendum to “Design, parallel synthesis, and crystal structures of biphenyl antithrombotics as selective inhibitors of tissue factor FVIIa complex. Part 1: Exploration of S2 pocket pharmacophores” [Bioorg. Med. Chem. 17 (2009) 3934]
|
Kotian, Pravin L.
|
|
2010
|
18 |
1 |
p. 460-
1 p.
|
artikel
|
| 12 |
Corrigendum to “Sildenafil is a strong activator of mammalian carbonic anhydrase isoforms I–XIV” [Bioorg. Med. Chem. 17 (2009) 5791]
|
Coban, T. Abdülkadir
|
|
2010
|
18 |
1 |
p. 461-
1 p.
|
artikel
|
| 13 |
Design, synthesis and biological evaluation of thiazolidinone derivatives as potential EGFR and HER-2 kinase inhibitors
|
Lv, Peng-Cheng
|
|
2010
|
18 |
1 |
p. 314-319
6 p.
|
artikel
|
| 14 |
Detection of multiple network-based allosteric interactions between peptides and arrays of DNA binding sites
|
Kao, Karen K.L.
|
|
2010
|
18 |
1 |
p. 366-376
11 p.
|
artikel
|
| 15 |
Editorial board
|
|
|
2010
|
18 |
1 |
p. IFC-
1 p.
|
artikel
|
| 16 |
α-Glucosidase inhibitory antihyperglycemic activity of substituted chromenone derivatives
|
Raju, B. China
|
|
2010
|
18 |
1 |
p. 358-365
8 p.
|
artikel
|
| 17 |
Graphical contents list
|
|
|
2010
|
18 |
1 |
p. 1-13
13 p.
|
artikel
|
| 18 |
Identification of a novel ligand binding motif in the transthyretin channel
|
Lima, Luis Mauricio T.R.
|
|
2010
|
18 |
1 |
p. 100-110
11 p.
|
artikel
|
| 19 |
Inhibition of IkB kinase and NF-κB by a novel synthetic compound SK 2009
|
Anchoori, Ravi Kumar
|
|
2010
|
18 |
1 |
p. 229-235
7 p.
|
artikel
|
| 20 |
Inhibitors of human tyrosyl-DNA phospodiesterase (hTdp1) developed by virtual screening using ligand-based pharmacophores
|
Weidlich, Iwona E.
|
|
2010
|
18 |
1 |
p. 182-189
8 p.
|
artikel
|
| 21 |
Inhibitory activity of Brazilian green propolis components and their derivatives on the release of cys-leukotrienes
|
Tani, Hiroko
|
|
2010
|
18 |
1 |
p. 151-157
7 p.
|
artikel
|
| 22 |
In silico prediction of human carboxylesterase-1 (hCES1) metabolism combining docking analyses and MD simulations
|
Vistoli, Giulio
|
|
2010
|
18 |
1 |
p. 320-329
10 p.
|
artikel
|
| 23 |
Isoxazole analogues bind the System x c - transporter: Structure–activity relationship and pharmacophore model
|
Patel, Sarjubhai A.
|
|
2010
|
18 |
1 |
p. 202-213
12 p.
|
artikel
|
| 24 |
Microwave assisted synthesis and antimicrobial activity of 2-quinoxalinone-3-hydrazone derivatives
|
Ajani, Olayinka O.
|
|
2010
|
18 |
1 |
p. 214-221
8 p.
|
artikel
|
| 25 |
Modulation of Wnt signaling through inhibition of secreted frizzled-related protein I (sFRP-1) with N-substituted piperidinyl diphenylsulfonyl sulfonamides: Part II
|
Moore, William J.
|
|
2010
|
18 |
1 |
p. 190-201
12 p.
|
artikel
|
| 26 |
99mTc-tricarbonyl labeled agents for cell labeling: Development, biodistribution in normal mice and preliminary in vitro evaluation
|
Fonge, Humphrey
|
|
2010
|
18 |
1 |
p. 396-402
7 p.
|
artikel
|
| 27 |
Multivalent catanionic GalCer analogs derived from first generation dendrimeric phosphonic acids
|
Pérez-Anes, Alexandra
|
|
2010
|
18 |
1 |
p. 242-248
7 p.
|
artikel
|
| 28 |
Nanomolar affinity, iminosugar-based chemical probes for specific labeling of lysosomal glucocerebrosidase
|
Scherpenzeel, Monique van
|
|
2010
|
18 |
1 |
p. 267-273
7 p.
|
artikel
|
| 29 |
New oligo-β-(1,3)-glucan derivatives as immunostimulating agents
|
Descroix, Karine
|
|
2010
|
18 |
1 |
p. 348-357
10 p.
|
artikel
|
| 30 |
New oxapolycyclic cage amines with NMDA receptor antagonist and trypanocidal activities
|
Duque, María D.
|
|
2010
|
18 |
1 |
p. 46-57
12 p.
|
artikel
|
| 31 |
New small-size peptides possessing antifungal activity
|
Garibotto, Francisco M.
|
|
2010
|
18 |
1 |
p. 158-167
10 p.
|
artikel
|
| 32 |
Novel 4-thiazolidinone derivatives as potential antifungal and antibacterial drugs
|
Omar, Kouatli
|
|
2010
|
18 |
1 |
p. 426-432
7 p.
|
artikel
|
| 33 |
Novel tumor-targeted RGD peptide–camptothecin conjugates: Synthesis and biological evaluation
|
Dal Pozzo, Alma
|
|
2010
|
18 |
1 |
p. 64-72
9 p.
|
artikel
|
| 34 |
Potent activity against K562 cells by polyamide–seco-CBI conjugates targeting histone H4 genes
|
Minoshima, Masafumi
|
|
2010
|
18 |
1 |
p. 168-174
7 p.
|
artikel
|
| 35 |
Probes for narcotic receptor mediated phenomena. 40. N-Substituted cis-4a-ethyl-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-8-ols
|
Iyer, Malliga R.
|
|
2010
|
18 |
1 |
p. 91-99
9 p.
|
artikel
|
| 36 |
Probing the carbohydrate recognition domain of E-selectin: The importance of the acid orientation in sLex mimetics
|
Titz, Alexander
|
|
2010
|
18 |
1 |
p. 19-27
9 p.
|
artikel
|
| 37 |
Reliability of bond dissociation enthalpy calculated by the PM6 method and experimental TEAC values in antiradical QSAR of flavonoids
|
Amić, Dragan
|
|
2010
|
18 |
1 |
p. 28-35
8 p.
|
artikel
|
| 38 |
Silicon switch approach in TRPV1 antagonist MK-056 and its analogues
|
Chang, Minsun
|
|
2010
|
18 |
1 |
p. 111-116
6 p.
|
artikel
|
| 39 |
Solid phase synthesis of novel asymmetric hydrophilic head cholesterol-based cationic lipids with potential DNA delivery
|
Radchatawedchakoon, Widchaya
|
|
2010
|
18 |
1 |
p. 330-342
13 p.
|
artikel
|
| 40 |
Substituted aryl malonamates as new serine β-lactamase substrates: Structure–activity studies
|
Adediran, S.A.
|
|
2010
|
18 |
1 |
p. 282-291
10 p.
|
artikel
|
| 41 |
Synthesis and anti-HIV evaluation of water-soluble calixarene-based bithiazolyl podands
|
Mourer, Maxime
|
|
2010
|
18 |
1 |
p. 36-45
10 p.
|
artikel
|
| 42 |
Synthesis and antiproliferative evaluations of certain 2-phenylvinylquinoline (2-styrylquinoline) and 2-furanylvinylquinoline derivatives
|
Chang, Feng-Shuo
|
|
2010
|
18 |
1 |
p. 124-133
10 p.
|
artikel
|
| 43 |
Synthesis and biological evaluation of trifluralin analogues as antileishmanial agents
|
Esteves, M.A.
|
|
2010
|
18 |
1 |
p. 274-281
8 p.
|
artikel
|
| 44 |
Synthesis and in vitro evaluation of fluorinated diphenyloxide derivatives and sulfur analogs as serotonin transporter ligands
|
Mavel, Sylvie
|
|
2010
|
18 |
1 |
p. 236-241
6 p.
|
artikel
|
| 45 |
Synthesis and structure–activity relationships of N-benzyl-N-(X-2-hydroxybenzyl)-N′-phenylureas and thioureas as antitumor agents
|
Li, Huan-Qiu
|
|
2010
|
18 |
1 |
p. 305-313
9 p.
|
artikel
|
| 46 |
Synthesis, nanosizing and in vitro drug release of a novel anti-HIV polymeric prodrug: Chitosan-O-isopropyl-5′-O-d4T monophosphate conjugate
|
Yang, Lin
|
|
2010
|
18 |
1 |
p. 117-123
7 p.
|
artikel
|
| 47 |
Synthesis of a new cytotoxic cephalostatin/ritterazine analogue from hecogenin and 22-epi-hippuristanol
|
Poza, Javier Jesús
|
|
2010
|
18 |
1 |
p. 58-63
6 p.
|
artikel
|
| 48 |
Synthesis of glycyrrhetinic acid derivatives for the treatment of metabolic diseases
|
Beseda, Igor
|
|
2010
|
18 |
1 |
p. 433-454
22 p.
|
artikel
|
| 49 |
Synthesis of 3-[(N-carboalkoxy)ethylamino]-indazole-dione derivatives and their biological activities on human liver carbonyl reductase
|
Berhe, Solomon
|
|
2010
|
18 |
1 |
p. 134-141
8 p.
|
artikel
|
| 50 |
Synthesis, physico-chemical properties and penetration activity of alkyl-6-(2,5-dioxopyrrolidin-1-yl)-2-(2-oxopyrrolidin-1-yl)hexanoates as potential transdermal penetration enhancers
|
Brychtova, Katerina
|
|
2010
|
18 |
1 |
p. 73-79
7 p.
|
artikel
|
| 51 |
Synthesis, stereoelectronic characterization and antiparasitic activity of new 1-benzenesulfonyl-2-methyl-1,2,3,4-tetrahydroquinolines
|
Pagliero, Romina J.
|
|
2010
|
18 |
1 |
p. 142-150
9 p.
|
artikel
|
| 52 |
The synthesis and evaluation of flavone and isoflavone chimeras of novobiocin and derrubone
|
Mays, Jared R.
|
|
2010
|
18 |
1 |
p. 249-266
18 p.
|
artikel
|
| 53 |
2-Thienyl-4-furyl-6-aryl pyridine derivatives: Synthesis, topoisomerase I and II inhibitory activity, cytotoxicity, and structure–activity relationship study
|
Thapa, Pritam
|
|
2010
|
18 |
1 |
p. 377-386
10 p.
|
artikel
|
| 54 |
Total synthesis and cytotoxicity evaluation of all ochratoxin A stereoisomers
|
Cramer, Benedikt
|
|
2010
|
18 |
1 |
p. 343-347
5 p.
|
artikel
|
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