| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
A novel and potent VLA-4 antagonist based on trans-4-substituted cyclohexanecarboxylic acid
|
Muro, Fumihito
|
|
2009
|
17 |
3 |
p. 1232-1243
12 p.
|
artikel
|
| 2 |
A road less traveled by: Exploring a decade of Ellman chemistry
|
Shelat, Anang A.
|
|
2009
|
17 |
3 |
p. 1088-1093
6 p.
|
artikel
|
| 3 |
A small molecule inhibitor of α4 integrin-dependent cell migration
|
Lee, Jongkook
|
|
2009
|
17 |
3 |
p. 977-980
4 p.
|
artikel
|
| 4 |
ATP competitive inhibitors of d-alanine–d-alanine ligase based on protein kinase inhibitor scaffolds
|
Triola, Gemma
|
|
2009
|
17 |
3 |
p. 1079-1087
9 p.
|
artikel
|
| 5 |
Benzopyridooxathiazepine derivatives as novel potent antimitotic agents
|
Gallet, Sebastien
|
|
2009
|
17 |
3 |
p. 1132-1138
7 p.
|
artikel
|
| 6 |
Biographical Sketch: Professor Jonathan Ellman
|
|
|
2009
|
17 |
3 |
p. 951-
1 p.
|
artikel
|
| 7 |
Bisubstrate Inhibitors of the MYST HATs Esa1 and Tip60
|
Wu, Jiang
|
|
2009
|
17 |
3 |
p. 1381-1386
6 p.
|
artikel
|
| 8 |
Carbonic anhydrase inhibitors. Comparison of chlorthalidone, indapamide, trichloromethiazide, and furosemide X-ray crystal structures in adducts with isozyme II, when several water molecules make the difference
|
Temperini, Claudia
|
|
2009
|
17 |
3 |
p. 1214-1221
8 p.
|
artikel
|
| 9 |
Carbonic anhydrase inhibitors: Inhibition of the β-class enzyme from the yeast Saccharomyces cerevisiae with sulfonamides and sulfamates
|
Isik, Semra
|
|
2009
|
17 |
3 |
p. 1158-1163
6 p.
|
artikel
|
| 10 |
Conformational analysis of trimeric maleimide substituted 1,5,9-triazacyclododecane HIV fusion scaffolds
|
Remmert, Sarah
|
|
2009
|
17 |
3 |
p. 1251-1258
8 p.
|
artikel
|
| 11 |
Cooperative alkylation of double-strand human telomere repeat sequences by PI polyamides with 11-base-pair recognition based on a heterotrimeric design
|
Kashiwazaki, Gengo
|
|
2009
|
17 |
3 |
p. 1393-1397
5 p.
|
artikel
|
| 12 |
Correlation of binding constants and molecular modelling of inhibitors in the active sites of aldose reductase and aldehyde reductase
|
Carbone, Vincenzo
|
|
2009
|
17 |
3 |
p. 1244-1250
7 p.
|
artikel
|
| 13 |
Coulombic effects on the traceless Staudinger ligation in water
|
Tam, Annie
|
|
2009
|
17 |
3 |
p. 1055-1063
9 p.
|
artikel
|
| 14 |
Death receptor 5 targeting activity-guided isolation of isoflavones from Millettia brandisiana and Ardisia colorata and evaluation of ability to induce TRAIL-mediated apoptosis
|
Kikuchi, Hiroyuki
|
|
2009
|
17 |
3 |
p. 1181-1186
6 p.
|
artikel
|
| 15 |
Determination of 1-aryl-4-propylpiperazine pK a values: The substituent on aryl modulates basicity
|
Lacivita, Enza
|
|
2009
|
17 |
3 |
p. 1339-1344
6 p.
|
artikel
|
| 16 |
Discovery of N-[(1R,2S,5S)-2-{[(5-chloroindol-2-yl)carbonyl]amino}-5-(dimethylcarbamoyl)cyclohexyl]-5-methyl-4,5,6,7-tetrahydrothiazolo[5,4-c]pyridine-2-carboxamide hydrochloride: A novel, potent and orally active direct inhibitor of factor Xa
|
Nagata, Tsutomu
|
|
2009
|
17 |
3 |
p. 1193-1206
14 p.
|
artikel
|
| 17 |
Editorial board
|
|
|
2009
|
17 |
3 |
p. IFC-
1 p.
|
artikel
|
| 18 |
Evaluation of α,β-unsaturated ketone-based probes for papain-family cysteine proteases
|
Yang, Zhimou
|
|
2009
|
17 |
3 |
p. 1071-1078
8 p.
|
artikel
|
| 19 |
Expanding the repertoire of small molecule transcriptional activation domains
|
Casey, Ryan J.
|
|
2009
|
17 |
3 |
p. 1034-1043
10 p.
|
artikel
|
| 20 |
Function-oriented synthesis applied to the anti-botulinum natural product toosendanin
|
Nakai, Yuya
|
|
2009
|
17 |
3 |
p. 1152-1157
6 p.
|
artikel
|
| 21 |
Graphical contents list
|
|
|
2009
|
17 |
3 |
p. 935-949
15 p.
|
artikel
|
| 22 |
High throughput screening of potentially selective MMP-13 exosite inhibitors utilizing a triple-helical FRET substrate
|
Lauer-Fields, Janelle L.
|
|
2009
|
17 |
3 |
p. 990-1005
16 p.
|
artikel
|
| 23 |
Instructions to contributors
|
|
|
2009
|
17 |
3 |
p. I-
1 p.
|
artikel
|
| 24 |
In vitro solubility, stability and permeability of novel quercetin–amino acid conjugates
|
Kim, Mi Kyoung
|
|
2009
|
17 |
3 |
p. 1164-1171
8 p.
|
artikel
|
| 25 |
Isolation, structure and biological activity of phomafungin, a cyclic lipodepsipeptide from a widespread tropical Phoma sp.
|
Herath, Kithsiri
|
|
2009
|
17 |
3 |
p. 1361-1369
9 p.
|
artikel
|
| 26 |
Isolation, structure elucidation and cytotoxic evaluation of endiandrin B from the Australian rainforest plant Endiandra anthropophagorum
|
Davis, Rohan A.
|
|
2009
|
17 |
3 |
p. 1387-1392
6 p.
|
artikel
|
| 27 |
Modification of the furan ring of salvinorin A: Identification of a selective partial agonist at the kappa opioid receptor
|
Béguin, Cécile
|
|
2009
|
17 |
3 |
p. 1370-1380
11 p.
|
artikel
|
| 28 |
New N-substituted 9-azabicyclo[3.3.1]nonan-3α-yl phenylcarbamate analogs as σ 2 receptor ligands: Synthesis, in vitro characterization, and evaluation as PET imaging and chemosensitization agents
|
Chu, Wenhua
|
|
2009
|
17 |
3 |
p. 1222-1231
10 p.
|
artikel
|
| 29 |
Novel boronated chlorin e6-based photosensitizers: Synthesis, binding to albumin and antitumour efficacy
|
Ol’shevskaya, Valentina A.
|
|
2009
|
17 |
3 |
p. 1297-1306
10 p.
|
artikel
|
| 30 |
Novel DNA-directed alkylating agents: Design, synthesis and potent antitumor effect of phenyl N-mustard-9-anilinoacridine conjugates via a carbamate or carbonate linker
|
Kapuriya, Naval
|
|
2009
|
17 |
3 |
p. 1264-1275
12 p.
|
artikel
|
| 31 |
Novel 6-methanesulfonamide-3,4-methylenedioxyphenyl-N-acylhydrazones: Orally effective anti-inflammatory drug candidates
|
Tributino, Jorge L.M.
|
|
2009
|
17 |
3 |
p. 1125-1131
7 p.
|
artikel
|
| 32 |
5′-O-Aliphatic and amino acid ester prodrugs of (−)-β-d-(2R,4R)-dioxolane-thymine (DOT): Synthesis, anti-HIV activity, cytotoxicity and stability studies
|
Liang, Yuzeng
|
|
2009
|
17 |
3 |
p. 1404-1409
6 p.
|
artikel
|
| 33 |
On-bead cyclization in a combinatorial library of 15,625 octapeptides
|
Fluxa, Viviana S.
|
|
2009
|
17 |
3 |
p. 1018-1025
8 p.
|
artikel
|
| 34 |
Preliminary evaluation of pharmacological properties of some xanthone derivatives
|
Marona, Henryk
|
|
2009
|
17 |
3 |
p. 1345-1352
8 p.
|
artikel
|
| 35 |
Ranking the selectivity of PubChem screening hits by activity-based protein profiling: MMP13 as a case study
|
Nakai, Ryuichiro
|
|
2009
|
17 |
3 |
p. 1101-1108
8 p.
|
artikel
|
| 36 |
Sidechain-linked inhibitors of HIV-1 protease dimerization
|
Bowman, Michael J.
|
|
2009
|
17 |
3 |
p. 967-976
10 p.
|
artikel
|
| 37 |
Site-specific covalent labeling of proteins inside live cells using small molecule probes
|
Chattopadhaya, Souvik
|
|
2009
|
17 |
3 |
p. 981-989
9 p.
|
artikel
|
| 38 |
Solid-phase parallel synthesis and SAR of 4-amidofuran-3-one inhibitors of cathepsin S: Effect of sulfonamides P3 substituents on potency and selectivity
|
Ayesa, Susana
|
|
2009
|
17 |
3 |
p. 1307-1324
18 p.
|
artikel
|
| 39 |
Solution- and solid-phase synthesis and anti-HIV activity of maslinic acid derivatives containing amino acids and peptides
|
Parra, Andres
|
|
2009
|
17 |
3 |
p. 1139-1145
7 p.
|
artikel
|
| 40 |
Structure–activity relationship study on polyglutamine binding peptide QBP1
|
Tomita, Kenji
|
|
2009
|
17 |
3 |
p. 1259-1263
5 p.
|
artikel
|
| 41 |
Structure-based virtual screening for novel inhibitors of the sarco/endoplasmic reticulum calcium ATPase and their experimental evaluation
|
Deye, Joel
|
|
2009
|
17 |
3 |
p. 1353-1360
8 p.
|
artikel
|
| 42 |
Substrate optimization for monitoring cathepsin C activity in live cells
|
Li, Jun
|
|
2009
|
17 |
3 |
p. 1064-1070
7 p.
|
artikel
|
| 43 |
Synthesis and antitumor activity of novel enediyne-linked pyrrolo[2,1-c][1,4]benzodiazepine hybrids
|
Hu, Wan-Ping
|
|
2009
|
17 |
3 |
p. 1172-1180
9 p.
|
artikel
|
| 44 |
Synthesis and biological evaluation of a library of resveratrol analogues as inhibitors of COX-1, COX-2 and NF-κB
|
Kang, Soo Sung
|
|
2009
|
17 |
3 |
p. 1044-1054
11 p.
|
artikel
|
| 45 |
Synthesis and biological evaluation of curcuminoid pyrazoles as new therapeutic agents in inflammatory bowel disease: Effect on matrix metalloproteinases
|
Claramunt, R.M.
|
|
2009
|
17 |
3 |
p. 1290-1296
7 p.
|
artikel
|
| 46 |
Synthesis and biological evaluation of extraordinarily potent C-10 carba artemisinin dimers against P. falciparum malaria parasites and HL-60 cancer cells
|
Chadwick, James
|
|
2009
|
17 |
3 |
p. 1325-1338
14 p.
|
artikel
|
| 47 |
Synthesis and biological evaluation of p-carborane bisphenols and their derivatives: Structure–activity relationship for estrogenic activity
|
Ogawa, Takumi
|
|
2009
|
17 |
3 |
p. 1109-1117
9 p.
|
artikel
|
| 48 |
Synthesis and cyclooxygenase inhibition of various (aryl-1,2,3-triazole-1-yl)-methanesulfonylphenyl derivatives
|
Wuest, Frank
|
|
2009
|
17 |
3 |
p. 1146-1151
6 p.
|
artikel
|
| 49 |
Synthesis and in vitro anti-proliferative activity of β-elemene monosubstituted derivatives in HeLa cells mediated through arrest of cell cycle at the G1 phase
|
Sun, Yanhong
|
|
2009
|
17 |
3 |
p. 1118-1124
7 p.
|
artikel
|
| 50 |
Synthesis and preliminary antibacterial evaluation of simplified thiomarinol analogs
|
Marion, Olivier
|
|
2009
|
17 |
3 |
p. 1006-1017
12 p.
|
artikel
|
| 51 |
Synthesis and screening of a cyclic peptide library: Discovery of small-molecule ligands against human prolactin receptor
|
Liu, Tao
|
|
2009
|
17 |
3 |
p. 1026-1033
8 p.
|
artikel
|
| 52 |
Synthesis of buprestins D, E, F, G and H; structural confirmation and biological testing of acyl glucoses from jewel beetles (Coleoptera: Buprestidae)
|
Ryczek, Sebastian
|
|
2009
|
17 |
3 |
p. 1187-1192
6 p.
|
artikel
|
| 53 |
Synthesis of oligodeoxynucleotides incorporating 2-N-carbamoylguanine and evaluation of the hybridization properties
|
Sasami, Takeshi
|
|
2009
|
17 |
3 |
p. 1398-1403
6 p.
|
artikel
|
| 54 |
Synthesis, penetrability and intracellular targeting of fluorescein-tagged peptoids and peptide–peptoid hybrids
|
Unciti-Broceta, Asier
|
|
2009
|
17 |
3 |
p. 959-966
8 p.
|
artikel
|
| 55 |
Synthesis, structure and antibacterial activity of new 2-(1-(2-(substituted-phenyl)-5-methyloxazol-4-yl)-3-(2-substitued-phenyl)-4,5-dihydro-1H-pyrazol-5-yl)-7-substitued-1,2,3,4-tetrahydroisoquinoline derivatives
|
Liu, Xin-Hua
|
|
2009
|
17 |
3 |
p. 1207-1213
7 p.
|
artikel
|
| 56 |
Tetrahedron Young Investigator Award for Bioorganic and Medicinal Chemistry
|
Wong, Chi-Huey
|
|
2009
|
17 |
3 |
p. 950-
1 p.
|
artikel
|
| 57 |
Towards Gram-negative antivirulence drugs: New inhibitors of HldE kinase
|
Desroy, Nicolas
|
|
2009
|
17 |
3 |
p. 1276-1289
14 p.
|
artikel
|
| 58 |
β-Turn secondary structure and melanocortin ligands
|
Haslach, Erica M.
|
|
2009
|
17 |
3 |
p. 952-958
7 p.
|
artikel
|
| 59 |
Using specificity to strategically target proteases
|
Lim, Mark D.
|
|
2009
|
17 |
3 |
p. 1094-1100
7 p.
|
artikel
|
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