| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
3- and 6-Substituted 2-amino-4,5,6,7-tetrahydrothieno[2,3-c]pyridines as A1 adenosine receptor allosteric modulators and antagonists
|
Aurelio, Luigi
|
|
2009
|
17 |
20 |
p. 7353-7361
9 p.
|
artikel
|
| 2 |
Antibacterial activity of aminoderivatized chitosans against methicillin-resistant Staphylococcus aureus (MRSA)
|
Lee, Dae-Sung
|
|
2009
|
17 |
20 |
p. 7108-7112
5 p.
|
artikel
|
| 3 |
A single circularly permuted GFP sensor for inositol-1,3,4,5-tetrakisphosphate based on a split PH domain
|
Sakaguchi, Reiko
|
|
2009
|
17 |
20 |
p. 7381-7386
6 p.
|
artikel
|
| 4 |
Benzamide derivatives as dual-action hypoglycemic agents that inhibit glycogen phosphorylase and activate glucokinase
|
Zhang, Lei
|
|
2009
|
17 |
20 |
p. 7301-7312
12 p.
|
artikel
|
| 5 |
2-Benzoylpyridine-N(4)-tolyl thiosemicarbazones and their palladium(II) complexes: Cytotoxicity against leukemia cells
|
Ferraz, Karina S.O.
|
|
2009
|
17 |
20 |
p. 7138-7144
7 p.
|
artikel
|
| 6 |
Carbonic anhydrase inhibitors. Diazenylbenzenesulfonamides are potent and selective inhibitors of the tumor-associated isozymes IX and XII over the cytosolic isoforms I and II
|
Carta, Fabrizio
|
|
2009
|
17 |
20 |
p. 7093-7099
7 p.
|
artikel
|
| 7 |
Cytosporones, coumarins, and an alkaloid from the endophytic fungus Pestalotiopsis sp. isolated from the Chinese mangrove plant Rhizophora mucronata
|
Xu, Jing
|
|
2009
|
17 |
20 |
p. 7362-7367
6 p.
|
artikel
|
| 8 |
Design, synthesis and evaluation of monovalent ligands for the asialoglycoprotein receptor (ASGP-R)
|
Stokmaier, Daniela
|
|
2009
|
17 |
20 |
p. 7254-7264
11 p.
|
artikel
|
| 9 |
Design, synthesis, and preliminary studies of the activity of novel derivatives of N-cinnamoyl-l-aspartic acid as inhibitors of aminopeptidase N/CD13
|
Liu, Yingzi
|
|
2009
|
17 |
20 |
p. 7398-7404
7 p.
|
artikel
|
| 10 |
Design, synthesis, and X-ray crystal structures of 2,4-diaminofuro[2,3-d]pyrimidines as multireceptor tyrosine kinase and dihydrofolate reductase inhibitors
|
Gangjee, Aleem
|
|
2009
|
17 |
20 |
p. 7324-7336
13 p.
|
artikel
|
| 11 |
2,4-Diaminopyrimidines as histamine H4 receptor ligands—Scaffold optimization and pharmacological characterization
|
Sander, Kerstin
|
|
2009
|
17 |
20 |
p. 7186-7196
11 p.
|
artikel
|
| 12 |
Discovery and structure–activity relationship analysis of Staphylococcus aureus sortase A inhibitors
|
Suree, Nuttee
|
|
2009
|
17 |
20 |
p. 7174-7185
12 p.
|
artikel
|
| 13 |
Editorial board
|
|
|
2009
|
17 |
20 |
p. IFC-
1 p.
|
artikel
|
| 14 |
Glucose-based spiro-isoxazolines: A new family of potent glycogen phosphorylase inhibitors
|
Benltifa, Mahmoud
|
|
2009
|
17 |
20 |
p. 7368-7380
13 p.
|
artikel
|
| 15 |
Graphical contents list
|
|
|
2009
|
17 |
20 |
p. 7075-7084
10 p.
|
artikel
|
| 16 |
Hepatoprotective amide constituents from the fruit of Piper chaba: Structural requirements, mode of action, and new amides
|
Matsuda, Hisashi
|
|
2009
|
17 |
20 |
p. 7313-7323
11 p.
|
artikel
|
| 17 |
Indene-based frameworks targeting the 5-HT6 serotonin receptor: Ring constraint in indenylsulfonamides using cyclic amines and structurally abbreviated counterparts
|
Alcalde, Ermitas
|
|
2009
|
17 |
20 |
p. 7387-7397
11 p.
|
artikel
|
| 18 |
Instructions to contributors
|
|
|
2009
|
17 |
20 |
p. I-
1 p.
|
artikel
|
| 19 |
Natural product leads for drug discovery: Isolation, synthesis and biological evaluation of 6-cyano-5-methoxyindolo[2,3-a]carbazole based ligands as antibacterial agents
|
Guo, Songpo
|
|
2009
|
17 |
20 |
p. 7126-7130
5 p.
|
artikel
|
| 20 |
PET-compatible endothelin receptor radioligands: Synthesis and first in vitro and in vivo studies
|
Höltke, Carsten
|
|
2009
|
17 |
20 |
p. 7197-7208
12 p.
|
artikel
|
| 21 |
Pochonicine, a polyhydroxylated pyrrolizidine alkaloid from fungus Pochonia suchlasporia var. suchlasporia TAMA 87 as a potent β-N-acetylglucosaminidase inhibitor
|
Usuki, Hirokazu
|
|
2009
|
17 |
20 |
p. 7248-7253
6 p.
|
artikel
|
| 22 |
Pyranonaphthoquinone derivatives of eleutherin, ventiloquinone L, thysanone and nanaomycin A possessing a diverse topoisomerase II inhibition and cytotoxicity spectrum
|
Sperry, Jonathan
|
|
2009
|
17 |
20 |
p. 7131-7137
7 p.
|
artikel
|
| 23 |
Structure–activity relationship of antiparasitic and cytotoxic indoloquinoline alkaloids, and their tricyclic and bicyclic analogues
|
Van Baelen, Gitte
|
|
2009
|
17 |
20 |
p. 7209-7217
9 p.
|
artikel
|
| 24 |
Synthesis and antioxidant properties of new chromone derivatives
|
Gomes, Ana
|
|
2009
|
17 |
20 |
p. 7218-7226
9 p.
|
artikel
|
| 25 |
Synthesis and biological evaluation of 14-(aminoalkyl-aminomethyl)aromathecins as topoisomerase I inhibitors: Investigating the hypothesis of shared structure–activity relationships
|
Cinelli, Maris A.
|
|
2009
|
17 |
20 |
p. 7145-7155
11 p.
|
artikel
|
| 26 |
Synthesis and biological evaluation of flavan-3-ol derivatives as positive modulators of GABAA receptors
|
Mewett, Kenneth N.
|
|
2009
|
17 |
20 |
p. 7156-7173
18 p.
|
artikel
|
| 27 |
Synthesis and discovery of pyrazole-5-carbohydrazide N-glycosides as inducer of autophagy in A549 lung cancer cells
|
Lian, Song
|
|
2009
|
17 |
20 |
p. 7085-7092
8 p.
|
artikel
|
| 28 |
Synthesis and evaluation of benzo[b]thiophene derivatives as inhibitors of alkaline phosphatases
|
Li, Lina
|
|
2009
|
17 |
20 |
p. 7290-7300
11 p.
|
artikel
|
| 29 |
Synthesis and evaluation of non-hydrolyzable d-mannose 6-phosphate surrogates reveal 6-deoxy-6-dicarboxymethyl-d-mannose as a new strong inhibitor of phosphomannose isomerases
|
Foret, Johanna
|
|
2009
|
17 |
20 |
p. 7100-7107
8 p.
|
artikel
|
| 30 |
Synthesis and evaluation of novel α-heteroaryl-phenylpropanoic acid derivatives as PPARα/γ dual agonists
|
Casimiro-Garcia, Agustin
|
|
2009
|
17 |
20 |
p. 7113-7125
13 p.
|
artikel
|
| 31 |
Synthesis and hybridization of 2′-O-methyl-RNAs incorporating 2′-O-carbamoyluridine and unique participation of the carbamoyl group in U–G base pair
|
Seio, Kohji
|
|
2009
|
17 |
20 |
p. 7275-7280
6 p.
|
artikel
|
| 32 |
Synthesis and pharmacological exploitation of clioquinol-derived copper-binding apoptosis inducers triggering reactive oxygen species generation and MAPK pathway activation
|
Chen, Hui-Ling
|
|
2009
|
17 |
20 |
p. 7239-7247
9 p.
|
artikel
|
| 33 |
Synthesis and structure–activity relationships of dehydroaltenusin derivatives as selective DNA polymerase α inhibitors
|
Kuramochi, Kouji
|
|
2009
|
17 |
20 |
p. 7227-7238
12 p.
|
artikel
|
| 34 |
Synthesis of 2- and 17-substituted estrone analogs and their antiproliferative structure–activity relationships compared to 2-methoxyestradiol
|
Shah, Jamshed H.
|
|
2009
|
17 |
20 |
p. 7344-7352
9 p.
|
artikel
|
| 35 |
Tetraiodobenzimidazoles are potent inhibitors of protein kinase CK2
|
Gianoncelli, Alessandra
|
|
2009
|
17 |
20 |
p. 7281-7289
9 p.
|
artikel
|
| 36 |
The biological activity and metabolic stability of peptidic bifunctional compounds that are opioid receptor agonists and neurokinin-1 receptor antagonists with a cystine moiety
|
Yamamoto, Takashi
|
|
2009
|
17 |
20 |
p. 7337-7343
7 p.
|
artikel
|
| 37 |
Ursolic acid derivatives induce cell cycle arrest and apoptosis in NTUB1 cells associated with reactive oxygen species
|
Tu, Huang-Yao
|
|
2009
|
17 |
20 |
p. 7265-7274
10 p.
|
artikel
|
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