| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
A new small molecule that directly inhibits the DNA binding of NF-κB
|
Kobayashi, Takanobu
|
|
2009
|
17 |
14 |
p. 5293-5297
5 p.
|
artikel
|
| 2 |
An extended study of dimeric phenyl tropanes
|
Nielsen, Susan
|
|
2009
|
17 |
14 |
p. 4900-4909
10 p.
|
artikel
|
| 3 |
Anti-tumor and anti-angiogenic activity of novel hydantoin derivatives: Inhibition of VEGF secretion in liver metastatic osteosarcoma cells
|
Basappa,
|
|
2009
|
17 |
14 |
p. 4928-4934
7 p.
|
artikel
|
| 4 |
Bioactive conformation analysis of cyclic imides as protoporphyrinogen oxidase inhibitor by combining DFT calculations, QSAR and molecular dynamic simulations
|
Zhang, Li
|
|
2009
|
17 |
14 |
p. 4935-4942
8 p.
|
artikel
|
| 5 |
Bioorganic & Medicinal Chemistry Reviews and Perspectives
|
|
|
2009
|
17 |
14 |
p. 5353-5355
3 p.
|
artikel
|
| 6 |
Carbonic anhydrase inhibitors. Aromatic/heterocyclic sulfonamides incorporating phenacetyl, pyridylacetyl and thienylacetyl tails act as potent inhibitors of human mitochondrial isoforms VA and VB
|
Güzel, Özlen
|
|
2009
|
17 |
14 |
p. 4894-4899
6 p.
|
artikel
|
| 7 |
Carbonic anhydrase inhibitors. Inhibition studies of a coral secretory isoform by sulfonamides
|
Bertucci, Anthony
|
|
2009
|
17 |
14 |
p. 5054-5058
5 p.
|
artikel
|
| 8 |
Characterization and synthetic application of a novel β1,3-galactosyltransferase from Escherichia coli O55:H7
|
Liu, Xian-wei
|
|
2009
|
17 |
14 |
p. 4910-4915
6 p.
|
artikel
|
| 9 |
‘Click’ D1 receptor agonists with a 5-HT1A receptor pharmacophore producing D2 receptor activity
|
Zhang, Jing
|
|
2009
|
17 |
14 |
p. 4873-4880
8 p.
|
artikel
|
| 10 |
Combining selectivity and affinity predictions using an integrated Support Vector Machine (SVM) approach: An alternative tool to discriminate between the human adenosine A2A and A3 receptor pyrazolo-triazolo-pyrimidine antagonists binding sites
|
Michielan, Lisa
|
|
2009
|
17 |
14 |
p. 5259-5274
16 p.
|
artikel
|
| 11 |
Computational selection of inhibitors of Aβ aggregation and neuronal toxicity
|
Chen, Deliang
|
|
2009
|
17 |
14 |
p. 5189-5197
9 p.
|
artikel
|
| 12 |
Design and synthesis of 3,5-diarylisoxazole derivatives as novel class of anti-hyperglycemic and lipid lowering agents
|
Kumar, Atul
|
|
2009
|
17 |
14 |
p. 5285-5292
8 p.
|
artikel
|
| 13 |
Design and synthesis of membrane fusion inhibitors against the feline immunodeficiency virus
|
Oishi, Shinya
|
|
2009
|
17 |
14 |
p. 4916-4920
5 p.
|
artikel
|
| 14 |
Diazen-1-ium-1,2-diolated nitric oxide donor ester prodrugs of 5-(4-carboxymethylphenyl)-1-(4-methanesulfonylphenyl)-3-trifluoromethyl-1H-pyrazole and its aminosulfonyl analog: Synthesis, biological evaluation and nitric oxide release studies
|
Abdellatif, Khaled R.A.
|
|
2009
|
17 |
14 |
p. 5182-5188
7 p.
|
artikel
|
| 15 |
Diketoacid-genre HIV-1 integrase inhibitors containing enantiomeric arylamide functionality
|
Zhao, Xue Zhi
|
|
2009
|
17 |
14 |
p. 5318-5324
7 p.
|
artikel
|
| 16 |
2D-QSAR and 3D-QSAR/CoMFA analyses of the N-terminal substituted anthranilic acid based CCK1 receptor antagonists: ‘Hic Rhodus, hic saltus’
|
Hadjipavlou-Litina, Dimitra
|
|
2009
|
17 |
14 |
p. 5198-5206
9 p.
|
artikel
|
| 17 |
Editorial board
|
|
|
2009
|
17 |
14 |
p. IFC-
1 p.
|
artikel
|
| 18 |
Efficient synthesis of the first betulonic acid–acetylene hybrids and their hepatoprotective and anti-inflammatory activity
|
Vasilevsky, Sergey F.
|
|
2009
|
17 |
14 |
p. 5164-5169
6 p.
|
artikel
|
| 19 |
Enaminones 10. Molecular modeling aspects of the 5-methylcyclohexenone derivatives
|
Gibson, Ainsley
|
|
2009
|
17 |
14 |
p. 5342-5346
5 p.
|
artikel
|
| 20 |
Fluorescence quenching properties of multiple pyrene-modified RNAs
|
Maie, Kenji
|
|
2009
|
17 |
14 |
p. 4996-5000
5 p.
|
artikel
|
| 21 |
Graphical contents list
|
|
|
2009
|
17 |
14 |
p. 4845-4860
16 p.
|
artikel
|
| 22 |
Identification of a bioactive compound isolated from Brazilian propolis type 6
|
Castro, Myrella Lessio
|
|
2009
|
17 |
14 |
p. 5332-5335
4 p.
|
artikel
|
| 23 |
Identification of PDE4B Over 4D subtype-selective inhibitors revealing an unprecedented binding mode
|
Kranz, Michael
|
|
2009
|
17 |
14 |
p. 5336-5341
6 p.
|
artikel
|
| 24 |
Inhibition of human vascular NADPH oxidase by apocynin derived oligophenols
|
Mora-Pale, Mauricio
|
|
2009
|
17 |
14 |
p. 5146-5152
7 p.
|
artikel
|
| 25 |
Inhibitors of VIM-2 by screening pharmacologically active and click-chemistry compound libraries
|
Minond, Dmitriy
|
|
2009
|
17 |
14 |
p. 5027-5037
11 p.
|
artikel
|
| 26 |
Instructions to contributors
|
|
|
2009
|
17 |
14 |
p. I-
1 p.
|
artikel
|
| 27 |
In vitro biological activity and structural analysis of 2,4-diamino-5-(2′-arylpropargyl)pyrimidine inhibitors of Candida albicans
|
Paulsen, Janet L.
|
|
2009
|
17 |
14 |
p. 4866-4872
7 p.
|
artikel
|
| 28 |
In vitro erythrocytic uptake studies of artemisinin and selected derivatives using LC–MS and 2D-QSAR analysis of uptake in parasitized erythrocytes
|
Shah, Falgun
|
|
2009
|
17 |
14 |
p. 5325-5331
7 p.
|
artikel
|
| 29 |
Mannosylated saponins based on oleanolic and glycyrrhizic acids. Towards synthetic colloidal antigen delivery systems
|
Daines, Alison M.
|
|
2009
|
17 |
14 |
p. 5207-5218
12 p.
|
artikel
|
| 30 |
Molecular modifications on carboxylic acid derivatives as potent histone deacetylase inhibitors: Activity and docking studies
|
Bora-Tatar, Gamze
|
|
2009
|
17 |
14 |
p. 5219-5228
10 p.
|
artikel
|
| 31 |
Molecular recognition in the P2Y14 receptor: Probing the structurally permissive terminal sugar moiety of uridine-5′-diphosphoglucose
|
Ko, Hyojin
|
|
2009
|
17 |
14 |
p. 5298-5311
14 p.
|
artikel
|
| 32 |
New furanoflavanoids, intestinal α-glucosidase inhibitory and free-radical (DPPH) scavenging, activity from antihyperglycemic root extract of Derris indica (Lam.)
|
Ranga Rao, R.
|
|
2009
|
17 |
14 |
p. 5170-5175
6 p.
|
artikel
|
| 33 |
NFκB decoy delivery using dendritic poly(l-lysine) for treatment of endotoxin-induced hepatitis in mice
|
Sugao, Yusuke
|
|
2009
|
17 |
14 |
p. 4990-4995
6 p.
|
artikel
|
| 34 |
Novel 1-aminoethyl-3-arylsulfonyl-1H-pyrrolo[2,3-b]pyridines are potent 5-HT6 agonists
|
Bernotas, Ronald C.
|
|
2009
|
17 |
14 |
p. 5153-5163
11 p.
|
artikel
|
| 35 |
Novel l-adenosine analogs as cardioprotective agents
|
Kasiganesan, Harinath
|
|
2009
|
17 |
14 |
p. 5347-5352
6 p.
|
artikel
|
| 36 |
Novel 3α-methoxyserrat-14-en-21β-ol (PJ-1) and 3β-methoxyserrat-14-en-21β-ol (PJ-2)-curcumin, kojic acid, quercetin, and baicalein conjugates as HIV agents
|
Tanaka, Reiko
|
|
2009
|
17 |
14 |
p. 5238-5246
9 p.
|
artikel
|
| 37 |
Novel orally active NPY Y5 receptor antagonists: Synthesis and structure–activity relationship of spiroindoline class compounds
|
Sakamoto, Toshihiro
|
|
2009
|
17 |
14 |
p. 5015-5026
12 p.
|
artikel
|
| 38 |
Nucleoside–amino acid conjugates: An alternative route to the design of ribonuclease A inhibitors
|
Debnath, Joy
|
|
2009
|
17 |
14 |
p. 4921-4927
7 p.
|
artikel
|
| 39 |
Optimization of peptide-based inhibitors of prostate-specific antigen (PSA) as targeted imaging agents for prostate cancer
|
LeBeau, Aaron M.
|
|
2009
|
17 |
14 |
p. 4888-4893
6 p.
|
artikel
|
| 40 |
Proteochemometrics mapping of the interaction space for retroviral proteases and their substrates
|
Kontijevskis, Aleksejs
|
|
2009
|
17 |
14 |
p. 5229-5237
9 p.
|
artikel
|
| 41 |
Purinergic P2X7 receptor antagonists: Chemistry and fundamentals of biological screening
|
Gunosewoyo, Hendra
|
|
2009
|
17 |
14 |
p. 4861-4865
5 p.
|
artikel
|
| 42 |
Quantitative high-throughput screening identifies inhibitors of anthrax-induced cell death
|
Zhu, Ping Jun
|
|
2009
|
17 |
14 |
p. 5139-5145
7 p.
|
artikel
|
| 43 |
Reaction of the antitumor antibiotic olivomycin I with aryl diazonium salts. Synthesis, cytotoxic and antiretroviral potency of 5-aryldiazenyl-6-O-deglycosyl derivatives of olivomycin I
|
Tevyashova, Anna N.
|
|
2009
|
17 |
14 |
p. 4961-4967
7 p.
|
artikel
|
| 44 |
Ruthenium complexes endowed with potent anti-Trypanosoma cruzi activity: Synthesis, biological characterization and structure–activity relationships
|
Donnici, Claudio Luis
|
|
2009
|
17 |
14 |
p. 5038-5043
6 p.
|
artikel
|
| 45 |
SAR and biological evaluation of SEN12333/WAY-317538: Novel alpha 7 nicotinic acetylcholine receptor agonist
|
Haydar, Simon N.
|
|
2009
|
17 |
14 |
p. 5247-5258
12 p.
|
artikel
|
| 46 |
Separation of α-glucosidase-inhibitory and liver X receptor-antagonistic activities of phenethylphenyl phthalimide analogs and generation of LXRα-selective antagonists
|
Motoshima, Kazunori
|
|
2009
|
17 |
14 |
p. 5001-5014
14 p.
|
artikel
|
| 47 |
Structure–activity studies on the nociceptin/orphanin FQ receptor antagonist 1-benzyl-N-{3-[spiroisobenzofuran-1(3H),4′-piperidin-1-yl]propyl} pyrrolidine-2-carboxamide
|
Trapella, Claudio
|
|
2009
|
17 |
14 |
p. 5080-5095
16 p.
|
artikel
|
| 48 |
Structure-based shape pharmacophore modeling for the discovery of novel anesthetic compounds
|
Ebalunode, Jerry O.
|
|
2009
|
17 |
14 |
p. 5133-5138
6 p.
|
artikel
|
| 49 |
Synthesis and antiproliferative activity of 2,4-disubstituted 6-aryl-7H-pyrrolo[3,2-d]pyrimidin-7-one 5-oxides
|
Pudziuvelyte, Erika
|
|
2009
|
17 |
14 |
p. 4955-4960
6 p.
|
artikel
|
| 50 |
Synthesis and biological evaluation of 11C-labeled β-galactosyl triazoles as potential PET tracers for in vivo LacZ reporter gene imaging
|
Celen, Sofie
|
|
2009
|
17 |
14 |
p. 5117-5125
9 p.
|
artikel
|
| 51 |
Synthesis and biological evaluation of new 4-carboxyl quinoline derivatives as cyclooxygenase-2 inhibitors
|
Zarghi, Afshin
|
|
2009
|
17 |
14 |
p. 5312-5317
6 p.
|
artikel
|
| 52 |
Synthesis and biological evaluation of SANT-2 and analogues as inhibitors of the hedgehog signaling pathway
|
Büttner, Anita
|
|
2009
|
17 |
14 |
p. 4943-4954
12 p.
|
artikel
|
| 53 |
Synthesis and investigations of double-pharmacophore ligands for treatment of chronic and neuropathic pain
|
Vardanyan, Ruben
|
|
2009
|
17 |
14 |
p. 5044-5053
10 p.
|
artikel
|
| 54 |
Synthesis and multidrug resistance reversal activity of dihydroptychantol A and its novel derivatives
|
Sun, Bin
|
|
2009
|
17 |
14 |
p. 4981-4989
9 p.
|
artikel
|
| 55 |
Synthesis and structure–activity relationship of 3β-(4-alkylthio, -methylsulfinyl, and -methylsulfonylphenyl)tropane and 3β-(4-alkylthiophenyl)nortropane derivatives for monoamine transporters
|
Jin, Chunyang
|
|
2009
|
17 |
14 |
p. 5126-5132
7 p.
|
artikel
|
| 56 |
Synthesis, antioxidant properties and radioprotective effects of new benzothiazoles and thiadiazoles
|
Cressier, Damien
|
|
2009
|
17 |
14 |
p. 5275-5284
10 p.
|
artikel
|
| 57 |
Synthesis, antitumor evaluation, molecular modeling and quantitative structure–activity relationship (QSAR) of some novel arylazopyrazolodiazine and triazine analogs
|
El-Shafei, Ahmed
|
|
2009
|
17 |
14 |
p. 5096-5105
10 p.
|
artikel
|
| 58 |
Synthesis, biological evaluation and docking studies of novel benzopyranone congeners for their expected activity as anti-inflammatory, analgesic and antipyretic agents
|
Eissa, Amal A.M.
|
|
2009
|
17 |
14 |
p. 5059-5070
12 p.
|
artikel
|
| 59 |
Synthesis of amyloid β peptide 1–42 (E22Δ) click peptide: pH-triggered in situ production of its native form
|
Wang, Hui
|
|
2009
|
17 |
14 |
p. 4881-4887
7 p.
|
artikel
|
| 60 |
Synthesis of novel purine nucleosides towards a selective inhibition of human butyrylcholinesterase
|
Marcelo, Filipa
|
|
2009
|
17 |
14 |
p. 5106-5116
11 p.
|
artikel
|
| 61 |
Synthesis of uracil nucleotide analogs with a modified, acyclic ribose moiety as P2Y2 receptor antagonists
|
Sauer, Roland
|
|
2009
|
17 |
14 |
p. 5071-5079
9 p.
|
artikel
|
| 62 |
Tetrahydroisoquinolines as dopaminergic ligands: 1-Butyl-7-chloro-6-hydroxy-tetrahydroisoquinoline, a new compound with antidepressant-like activity in mice
|
Berenguer, Inmaculada
|
|
2009
|
17 |
14 |
p. 4968-4980
13 p.
|
artikel
|
| 63 |
Toward preparation of antibody-based imaging probe libraries for dual-modality positron emission tomography and fluorescence imaging
|
Xu, Heng
|
|
2009
|
17 |
14 |
p. 5176-5181
6 p.
|
artikel
|
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