| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
6-Amino-2-mercapto-3H-pyrimidin-4-one derivatives as new candidates for the antagonism at the P2Y12 receptors
|
Crepaldi, Pamela
|
|
2009
|
17 |
13 |
p. 4612-4621
10 p.
|
artikel
|
| 2 |
Analysis of binding parameters of HIV-1 integrase inhibitors: Correlates of drug inhibition and resistance
|
Loizidou, Eriketi Z.
|
|
2009
|
17 |
13 |
p. 4806-4818
13 p.
|
artikel
|
| 3 |
Antimycobacterial activity of new 3,5-disubstituted 1,3,4-oxadiazol-2(3H)-one derivatives. Molecular modeling investigations
|
Zampieri, Daniele
|
|
2009
|
17 |
13 |
p. 4693-4707
15 p.
|
artikel
|
| 4 |
Antiviral and cytotoxic activities of aminoarylazo compounds and aryltriazene derivatives
|
Tonelli, Michele
|
|
2009
|
17 |
13 |
p. 4425-4440
16 p.
|
artikel
|
| 5 |
A versatile photoactivatable probe designed to label the diphosphate binding site of farnesyl diphosphate utilizing enzymes
|
Henry, Olivier
|
|
2009
|
17 |
13 |
p. 4797-4805
9 p.
|
artikel
|
| 6 |
Benzhydrylquinazolinediones: Novel cytosolic phospholipase A2α inhibitors with improved physicochemical properties
|
Kirincich, Steven J.
|
|
2009
|
17 |
13 |
p. 4383-4405
23 p.
|
artikel
|
| 7 |
Carbonic anhydrase inhibitors. Inhibition and homology modeling studies of the fungal β-carbonic anhydrase from Candida albicans with sulfonamides
|
Innocenti, Alessio
|
|
2009
|
17 |
13 |
p. 4503-4509
7 p.
|
artikel
|
| 8 |
Chemistry of renieramycins. Part 8: Synthesis and cytotoxicity evaluation of renieramycin M–jorunnamycin A analogues
|
Charupant, Kornvika
|
|
2009
|
17 |
13 |
p. 4548-4558
11 p.
|
artikel
|
| 9 |
Cytotoxic activity and inhibitory effect on nitric oxide production of triterpene saponins from the roots of Physospermum verticillatum (Waldst & Kit) (Apiaceae)
|
Tundis, Rosa
|
|
2009
|
17 |
13 |
p. 4542-4547
6 p.
|
artikel
|
| 10 |
Design and synthesis of ten biphenyl-neolignan derivatives and their in vitro inhibitory potency against cyclooxygenase-1/2 activity and 5-lipoxygenase-mediated LTB4-formation
|
Schühly, Wolfgang
|
|
2009
|
17 |
13 |
p. 4459-4465
7 p.
|
artikel
|
| 11 |
Design of Ga–DOTA-based bifunctional radiopharmaceuticals: Two functional moieties can be conjugated to radiogallium–DOTA without reducing the complex stability
|
Mukai, Takahiro
|
|
2009
|
17 |
13 |
p. 4285-4289
5 p.
|
artikel
|
| 12 |
Design, synthesis and biological evaluation of novel triazole, urea and thiourea derivatives of quinoline against Mycobacterium tuberculosis
|
Upadhayaya, Ram Shankar
|
|
2009
|
17 |
13 |
p. 4681-4692
12 p.
|
artikel
|
| 13 |
Design, synthesis and dopamine D4 receptor binding activities of new N-heteroaromatic 5/6-ring Mannich bases
|
Linz, Sabine
|
|
2009
|
17 |
13 |
p. 4448-4458
11 p.
|
artikel
|
| 14 |
Design, synthesis and primary activity evaluation of l-arginine derivatives as amino-peptidase N/CD13 inhibitors
|
Mou, Jiajia
|
|
2009
|
17 |
13 |
p. 4666-4673
8 p.
|
artikel
|
| 15 |
Discovery, characterization and comparison of inhibitors of Bacillus anthracis and Staphylococcus aureus replicative DNA helicases
|
Aiello, Daniel
|
|
2009
|
17 |
13 |
p. 4466-4476
11 p.
|
artikel
|
| 16 |
Discovery of novel P3 sulfonamide-capped inhibitors of HCV NS3 protease. Inhibitors with improved cellular potencies
|
Venkatraman, Srikanth
|
|
2009
|
17 |
13 |
p. 4486-4495
10 p.
|
artikel
|
| 17 |
Discovery of tetrahydrotetramethylnaphthalene analogs as adult T-cell leukemia cell-selective proliferation inhibitors in a small chemical library constructed based on multi-template hypothesis
|
Nakamura, Masahiko
|
|
2009
|
17 |
13 |
p. 4740-4746
7 p.
|
artikel
|
| 18 |
Editorial board
|
|
|
2009
|
17 |
13 |
p. IFC-
1 p.
|
artikel
|
| 19 |
Efficient solid-phase synthesis of oligodeoxynucleotides having a 5′-terminal 2,2,7-trimethylguanosine pyrophosphate linkage
|
Ohkubo, Akihiro
|
|
2009
|
17 |
13 |
p. 4819-4824
6 p.
|
artikel
|
| 20 |
Enhanced cytotoxicity of a polymer–drug conjugate with triple payload of paclitaxel
|
Erez, Rotem
|
|
2009
|
17 |
13 |
p. 4327-4335
9 p.
|
artikel
|
| 21 |
Evaluation of anti-inflammatory effect of synthetic 1,5-bis(4-acetoxy-3-methoxyphenyl)-1,4-pentadien-3-one, HB2
|
Paulino, Niraldo
|
|
2009
|
17 |
13 |
p. 4290-4295
6 p.
|
artikel
|
| 22 |
Glycogen phosphorylase inhibitory effects of 2-oxo-1,2-dihydropyridin-3-yl amide derivatives
|
Karis, N. David
|
|
2009
|
17 |
13 |
p. 4724-4733
10 p.
|
artikel
|
| 23 |
Graphical contents list
|
|
|
2009
|
17 |
13 |
p. 4257-4273
17 p.
|
artikel
|
| 24 |
Human sialidase inhibitors: Design, synthesis, and biological evaluation of 4-acetamido-5-acylamido-2-fluoro benzoic acids
|
Magesh, Sadagopan
|
|
2009
|
17 |
13 |
p. 4595-4603
9 p.
|
artikel
|
| 25 |
Identification of novel serotonin 2C receptor ligands by sequential virtual screening
|
Ahmed, Asif
|
|
2009
|
17 |
13 |
p. 4559-4568
10 p.
|
artikel
|
| 26 |
Inhibitory effects of phloroglucinol derivatives isolated from Ecklonia stolonifera on FcεRI expression
|
Shim, Sun-Yup
|
|
2009
|
17 |
13 |
p. 4734-4739
6 p.
|
artikel
|
| 27 |
Instructions to contributors
|
|
|
2009
|
17 |
13 |
p. I-
1 p.
|
artikel
|
| 28 |
In vitro and in vivo studies of 6,8-(diaryl)imidazo[1,2-a]pyrazin-3(7H)-ones as new antioxidants
|
De Wael, Frederic
|
|
2009
|
17 |
13 |
p. 4336-4344
9 p.
|
artikel
|
| 29 |
Lathyrane diterpenes from Euphorbia lathyris as modulators of multidrug resistance and their crystal structures
|
Jiao, Wei
|
|
2009
|
17 |
13 |
p. 4786-4792
7 p.
|
artikel
|
| 30 |
Minor structural differences of monomethine cyanine derivatives yield strong variation in their interactions with DNA, RNA as well as on their in vitro antiproliferative activity
|
Glavaš-Obrovac, Ljubica
|
|
2009
|
17 |
13 |
p. 4747-4755
9 p.
|
artikel
|
| 31 |
Molecular encapsulation of 5-nitroindazole derivatives in 2,6-dimethyl-β-cyclodextrin: Electrochemical and spectroscopic studies
|
Pérez-Cruz, Fernanda
|
|
2009
|
17 |
13 |
p. 4604-4611
8 p.
|
artikel
|
| 32 |
Novel and potent small-molecule urotensin II receptor agonists
|
Lehmann, Fredrik
|
|
2009
|
17 |
13 |
p. 4657-4665
9 p.
|
artikel
|
| 33 |
Novel hyaluronic acid–methotrexate conjugates for osteoarthritis treatment
|
Homma, Akie
|
|
2009
|
17 |
13 |
p. 4647-4656
10 p.
|
artikel
|
| 34 |
N-Substituted-2-alkyl- and 2-arylnorapomorphines: Novel, highly active D2 agonists
|
Herm, Laura
|
|
2009
|
17 |
13 |
p. 4756-4762
7 p.
|
artikel
|
| 35 |
2-Oxoamide inhibitors of phospholipase A2 activity and cellular arachidonate release based on dipeptides and pseudodipeptides
|
Barbayianni, Efrosini
|
|
2009
|
17 |
13 |
p. 4833-4843
11 p.
|
artikel
|
| 36 |
Phage display screening against a set of targets to establish peptide-based sugar mimetics and molecular docking to predict binding site
|
Yu, Limin
|
|
2009
|
17 |
13 |
p. 4825-4832
8 p.
|
artikel
|
| 37 |
Potential antioxidants and tyrosinase inhibitors from synthetic polyphenolic deoxybenzoins
|
Ng, Lean-Teik
|
|
2009
|
17 |
13 |
p. 4360-4366
7 p.
|
artikel
|
| 38 |
p-Terphenyls from the fruiting bodies of Paxillus curtisii and their antioxidant properties
|
Lee, In-Kyoung
|
|
2009
|
17 |
13 |
p. 4674-4680
7 p.
|
artikel
|
| 39 |
QSAR study on maximal inhibition (I max) of quaternary ammonium antagonists for S-(−)-nicotine-evoked dopamine release from dopaminergic nerve terminals in rat striatum
|
Zheng, Fang
|
|
2009
|
17 |
13 |
p. 4477-4485
9 p.
|
artikel
|
| 40 |
Quinazolindione derivatives as potent 5-HT3A receptor antagonists
|
Lee, Byung-Hwan
|
|
2009
|
17 |
13 |
p. 4793-4796
4 p.
|
artikel
|
| 41 |
Retinoid receptor subtype-selective modulators through synthetic modifications of RARγ agonists
|
Álvarez, Susana
|
|
2009
|
17 |
13 |
p. 4345-4359
15 p.
|
artikel
|
| 42 |
9,11-Secosterols with antiproliferative activity from the gorgonian Eunicella cavolini
|
Ioannou, Efstathia
|
|
2009
|
17 |
13 |
p. 4537-4541
5 p.
|
artikel
|
| 43 |
Synthesis and antimicrobial activity of 4-hydroxy-4-(pyridyl)alk-3-en-2-ones
|
Riahi, Abdolmajid
|
|
2009
|
17 |
13 |
p. 4323-4326
4 p.
|
artikel
|
| 44 |
Synthesis and biological activities of aminopyrimidyl-indoles structurally related to meridianins
|
Akue-Gedu, Rufine
|
|
2009
|
17 |
13 |
p. 4420-4424
5 p.
|
artikel
|
| 45 |
Synthesis and biological activity of a fluorescent schweinfurthin analogue
|
Kuder, Craig H.
|
|
2009
|
17 |
13 |
p. 4718-4723
6 p.
|
artikel
|
| 46 |
Synthesis and biological evaluation of febrifugine analogues as potential antimalarial agents
|
Zhu, Shuren
|
|
2009
|
17 |
13 |
p. 4496-4502
7 p.
|
artikel
|
| 47 |
Synthesis and biological evaluation of novel 4-azaindolyl-indolyl-maleimides as glycogen synthase kinase-3β (GSK-3β) inhibitors
|
Ye, Qing
|
|
2009
|
17 |
13 |
p. 4302-4312
11 p.
|
artikel
|
| 48 |
Synthesis and biological evaluation of novel carbon-11 labeled pyridyl ethers: candidate ligands for in vivo imaging of α4β2 nicotinic acetylcholine receptors (α4β2-nAChRs) in the brain with positron emission tomography
|
Gao, Yongjun
|
|
2009
|
17 |
13 |
p. 4367-4377
11 p.
|
artikel
|
| 49 |
Synthesis and cytotoxic activity of 5,6-heteroaromatically annulated pyridine-2,4-diamines
|
Willemann, C.
|
|
2009
|
17 |
13 |
p. 4406-4419
14 p.
|
artikel
|
| 50 |
Synthesis and DNA cleavage activity of 2-hydrazinyl-1,4,5,6-tetrahydropyrimidine containing hydroxy group
|
Shao, Ying
|
|
2009
|
17 |
13 |
p. 4274-4279
6 p.
|
artikel
|
| 51 |
Synthesis and evaluation of novel 7-azaindazolyl-indolyl-maleimide derivatives as antitumor agents and protein kinase C inhibitors
|
Ye, Qing
|
|
2009
|
17 |
13 |
p. 4763-4772
10 p.
|
artikel
|
| 52 |
Synthesis and in vitro anti-hepatitis B virus activity of 6H-[1]benzothiopyrano[4,3-b]quinolin-9-ols
|
Jia, Wei
|
|
2009
|
17 |
13 |
p. 4569-4574
6 p.
|
artikel
|
| 53 |
Synthesis and in vitro antiplasmodial evaluation of 4-anilino-2-trichloromethylquinazolines
|
Verhaeghe, Pierre
|
|
2009
|
17 |
13 |
p. 4313-4322
10 p.
|
artikel
|
| 54 |
Synthesis and pharmacological evaluation of 1,2,3,4-tetrahydropyrazino[1,2-a]indole and 2-[(phenylmethylamino)methyl]-1H-indole analogues as novel melatoninergic ligands
|
Markl, Christian
|
|
2009
|
17 |
13 |
p. 4583-4594
12 p.
|
artikel
|
| 55 |
Synthesis and structure–activity relationship of a novel series of heterocyclic sulfonamide γ-secretase inhibitors
|
Pu, Jun
|
|
2009
|
17 |
13 |
p. 4708-4717
10 p.
|
artikel
|
| 56 |
Synthesis and structure–activity relationship of Huprine derivatives as human acetylcholinesterase inhibitors
|
Ronco, Cyril
|
|
2009
|
17 |
13 |
p. 4523-4536
14 p.
|
artikel
|
| 57 |
Synthesis and structure–activity relationships of C-glycosylated oxadiazoles as inhibitors of glycogen phosphorylase
|
Tóth, Marietta
|
|
2009
|
17 |
13 |
p. 4773-4785
13 p.
|
artikel
|
| 58 |
Synthesis and structure–activity relationships of N-(4-amino-2,6-diisopropylphenyl)-N’-(1,4-diarylpiperidine-4-yl)methylureas as anti-hyperlipidemic agents
|
Asano, Shigehiro
|
|
2009
|
17 |
13 |
p. 4636-4646
11 p.
|
artikel
|
| 59 |
Synthesis and structure–activity relationships of radicicol derivatives and WNT-5A expression inhibitory activity
|
Shinonaga, Hideki
|
|
2009
|
17 |
13 |
p. 4622-4635
14 p.
|
artikel
|
| 60 |
Synthesis of hybrid analogues of caffeine and eudistomin D and its affinity for adenosine receptors
|
Ishiyama, Haruaki
|
|
2009
|
17 |
13 |
p. 4280-4284
5 p.
|
artikel
|
| 61 |
Synthesis of 2α-propoxy-1α,25-dihydroxyvitamin D3 and comparison of its metabolism by human CYP24A1 and rat CYP24A1
|
Saito, Nozomi
|
|
2009
|
17 |
13 |
p. 4296-4301
6 p.
|
artikel
|
| 62 |
Synthesis of quinolinyl and isoquinolinyl phenyl ketones as novel agonists for the cannabinoid CB2 receptor
|
Reux, Bastien
|
|
2009
|
17 |
13 |
p. 4441-4447
7 p.
|
artikel
|
| 63 |
Synthesis, structural characterisation and biological evaluation of fluorinated analogues of resveratrol
|
Moran, Brian W.
|
|
2009
|
17 |
13 |
p. 4510-4522
13 p.
|
artikel
|
| 64 |
Synthetic resveratrol aliphatic acid inhibits TLR2-mediated apoptosis and an involvement of Akt/GSK3β pathway
|
Chen, Lin
|
|
2009
|
17 |
13 |
p. 4378-4382
5 p.
|
artikel
|
| 65 |
The structure-based design, synthesis, and biological evaluation of DNA-binding amide linked bisintercalating bisanthrapyrazole anticancer compounds
|
Hasinoff, Brian B.
|
|
2009
|
17 |
13 |
p. 4575-4582
8 p.
|
artikel
|
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