| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
ACE inhibitors hypothesis generation for selective design, synthesis and biological evaluation of 3-mercapto-2-methyl-propanoyl-pyrrolidine-3-imine derivatives as antihypertensive agents
|
Ismail, Mohamed A.H.
|
|
2009
|
17 |
10 |
p. 3739-3746
8 p.
|
artikel
|
| 2 |
6-Amino-4-oxo-1,3-diphenyl-2-thioxo-1,2,3,4-tetrahydropyrimidine-5-carbonyl derivatives as a new class of potent inhibitors of Interleukin-8-induced neutrophil chemotaxis
|
Cesarini, Sara
|
|
2009
|
17 |
10 |
p. 3580-3587
8 p.
|
artikel
|
| 3 |
Antiplasmodial and antitrypanosomal activity of bicyclic amides and esters of dialkylamino acids
|
Faist, Johanna
|
|
2009
|
17 |
10 |
p. 3595-3603
9 p.
|
artikel
|
| 4 |
Carbonic anhydrase inhibitors. Inhibition of the human cytosolic isoforms I and II and transmembrane, tumor-associated isoforms IX and XII with boronic acids
|
Winum, Jean-Yves
|
|
2009
|
17 |
10 |
p. 3649-3652
4 p.
|
artikel
|
| 5 |
Chlorzoxazone esters of some non-steroidal anti-inflammatory (NSAI) carboxylic acids as mutual prodrugs: Design, synthesis, pharmacological investigations and docking studies
|
Abdel-Azeem, Ahmed Z.
|
|
2009
|
17 |
10 |
p. 3665-3670
6 p.
|
artikel
|
| 6 |
2′-Deoxy-1-methylpseudocytidine, a stable analog of 2′-deoxy-5-methylisocytidine
|
Kim, Hyo-Joong
|
|
2009
|
17 |
10 |
p. 3728-3732
5 p.
|
artikel
|
| 7 |
Design, synthesis, and biological evaluation of novel diarylalkyl amides as TRPV1 antagonists
|
Li, Fu-Nan
|
|
2009
|
17 |
10 |
p. 3557-3567
11 p.
|
artikel
|
| 8 |
1,3-Dialkyl-8-N-substituted benzyloxycarbonylamino-9-deazaxanthines as potent adenosine receptor ligands: Design, synthesis, structure–affinity and structure–selectivity relationships
|
Fernández, Franco
|
|
2009
|
17 |
10 |
p. 3618-3629
12 p.
|
artikel
|
| 9 |
2,4(5)-Diarylimidazoles as inhibitors of hNaV1.2 sodium channels: Pharmacological evaluation and structure–property relationships
|
Fantini, Marco
|
|
2009
|
17 |
10 |
p. 3642-3648
7 p.
|
artikel
|
| 10 |
Discovery and SAR of cinnolines/quinolines as liver X receptor (LXR) agonists with binding selectivity for LXRβ
|
Hu, Baihua
|
|
2009
|
17 |
10 |
p. 3519-3527
9 p.
|
artikel
|
| 11 |
Discovery, synthesis, and biological evaluation of piperidinol analogs with anti-tuberculosis activity
|
Sun, Dianqing
|
|
2009
|
17 |
10 |
p. 3588-3594
7 p.
|
artikel
|
| 12 |
3D QSAR of novel estrogen–RGD peptide conjugates: Getting insight into structural dependence of anti-osteoporosis activity and side effect of estrogen in ERT
|
Zhao, Ming
|
|
2009
|
17 |
10 |
p. 3680-3689
10 p.
|
artikel
|
| 13 |
Editorial board
|
|
|
2009
|
17 |
10 |
p. IFC-
1 p.
|
artikel
|
| 14 |
Enzymatic synthesis of perfluoroalkylated DNA
|
Holzberger, Bastian
|
|
2009
|
17 |
10 |
p. 3653-3658
6 p.
|
artikel
|
| 15 |
Graphical contents list
|
|
|
2009
|
17 |
10 |
p. 3511-3518
8 p.
|
artikel
|
| 16 |
Instructions to contributors
|
|
|
2009
|
17 |
10 |
p. I-
1 p.
|
artikel
|
| 17 |
Mechanism-based inhibitors of serine proteases with high selectivity through optimization of S′ subsite binding
|
Li, Yi
|
|
2009
|
17 |
10 |
p. 3536-3542
7 p.
|
artikel
|
| 18 |
Mechanism of action of N-phenyl-N′-(2-chloroethyl)ureas in the colchicine-binding site at the interface between α- and β-tubulin
|
Fortin, Sébastien
|
|
2009
|
17 |
10 |
p. 3690-3697
8 p.
|
artikel
|
| 19 |
New antituberculotics originated from salicylanilides with promising in vitro activity against atypical mycobacterial strains
|
Imramovský, Aleš
|
|
2009
|
17 |
10 |
p. 3572-3579
8 p.
|
artikel
|
| 20 |
On the inhibition of HIV-1 protease by hydrazino-ureas displaying the N→CO interaction
|
Waibel, Michael
|
|
2009
|
17 |
10 |
p. 3671-3679
9 p.
|
artikel
|
| 21 |
QSAR models for predicting enzymatic hydrolysis of new chemical entities in ‘soft-drug’ design
|
Massarelli, I.
|
|
2009
|
17 |
10 |
p. 3543-3556
14 p.
|
artikel
|
| 22 |
Steroidal bivalent ligands for the estrogen receptor: Design, synthesis, characterization and binding affinities
|
LaFrate, Andrew L.
|
|
2009
|
17 |
10 |
p. 3528-3535
8 p.
|
artikel
|
| 23 |
Structure–activity relationships of truncated adenosine derivatives as highly potent and selective human A3 adenosine receptor antagonists
|
Pal, Shantanu
|
|
2009
|
17 |
10 |
p. 3733-3738
6 p.
|
artikel
|
| 24 |
Studies on novel 2-imidazolidinones and tetrahydropyrimidin-2(1H)-ones as potential TACE inhibitors: Design, synthesis, molecular modeling, and preliminary biological evaluation
|
DasGupta, Shirshendu
|
|
2009
|
17 |
10 |
p. 3604-3617
14 p.
|
artikel
|
| 25 |
2-(Substituted phenyl)amino analogs of 1-methoxyspirobrassinol methyl ether: Synthesis and anticancer activity
|
Kutschy, Peter
|
|
2009
|
17 |
10 |
p. 3698-3712
15 p.
|
artikel
|
| 26 |
Synthesis and antirhinovirus activity of new 3-benzyl chromene and chroman derivatives
|
Conti, Cinzia
|
|
2009
|
17 |
10 |
p. 3720-3727
8 p.
|
artikel
|
| 27 |
Synthesis and evaluation of pharmacological profile of 1-aryl-6,7-dimethoxy-3,4-dihydroisoquinoline-2(1H)-sulfonamides
|
Gitto, Rosaria
|
|
2009
|
17 |
10 |
p. 3659-3664
6 p.
|
artikel
|
| 28 |
Synthesis, antiplatelet and in silico evaluations of novel N-substituted-phenylamino-5-methyl-1H-1,2,3-triazole-4-carbohydrazides
|
Jordão, Alessandro K.
|
|
2009
|
17 |
10 |
p. 3713-3719
7 p.
|
artikel
|
| 29 |
Synthesis of spirocyclic σ1 receptor ligands as potential PET radiotracers, structure–affinity relationships and in vitro metabolic stability
|
Große Maestrup, Eva
|
|
2009
|
17 |
10 |
p. 3630-3641
12 p.
|
artikel
|
| 30 |
Unique behavior of 2,6-bis(bromomethyl)naphthalene as a highly active organic DNA crosslinking molecule
|
Higashi, Toshinori
|
|
2009
|
17 |
10 |
p. 3568-3571
4 p.
|
artikel
|
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