nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
1 |
A comparative molecular field and comparative molecular similarity indices analyses (CoMFA and CoMSIA) of N-phenyl-N′-(2-chloroethyl)ureas targeting the colchicine-binding site as anticancer agents
|
Fortin, Sébastien |
|
2008 |
16 |
4 |
p. 1914-1926 13 p. |
artikel |
2 |
An expeditious one-pot synthesis of 1,6-dideoxy-N-alkylated nojirimycin derivatives and their inhibitory effects on the secretion of IFN-γ and IL-4
|
Zhou, Jian |
|
2008 |
16 |
4 |
p. 1605-1612 8 p. |
artikel |
3 |
A novel series of parenteral cephalosporins exhibiting potent activities against both Pseudomonas aeruginosa and other Gram-negative pathogens. Part 2: Synthesis and structure–activity relationships
|
Yamawaki, Kenji |
|
2008 |
16 |
4 |
p. 1632-1647 16 p. |
artikel |
4 |
A novel sesquiterpenoid dimer parviflorene F induces apoptosis by up-regulating the expression of TRAIL-R2 and a caspase-dependent mechanism
|
Ohtsuki, Takashi |
|
2008 |
16 |
4 |
p. 1756-1763 8 p. |
artikel |
5 |
Anti-Plasmodium activity of tetrazolium salts
|
Cui, Xilin |
|
2008 |
16 |
4 |
p. 1927-1947 21 p. |
artikel |
6 |
Antiproliferative effects on human tumor cells and rat aortic smooth muscular cells of 2,3-heteroarylmaleimides and heterofused imides
|
Ferri, Nicola |
|
2008 |
16 |
4 |
p. 1691-1701 11 p. |
artikel |
7 |
Aryl azoles with neuroprotective activity—Parallel synthesis and attempts at target identification
|
Cocconcelli, Giuseppe |
|
2008 |
16 |
4 |
p. 2043-2052 10 p. |
artikel |
8 |
Biomimetic synthesis of xuxuarines Eα and Eβ: Structure revision of Rzedowskia bistriterpenoids
|
Jacobsen, Neil E. |
|
2008 |
16 |
4 |
p. 1884-1889 6 p. |
artikel |
9 |
Bioorganic & Medicinal Chemistry Reviews and Perspectives
|
|
|
2008 |
16 |
4 |
p. 2131-2133 3 p. |
artikel |
10 |
Conception of myeloperoxidase inhibitors derived from flufenamic acid by computational docking and structure modification
|
Van Antwerpen, Pierre |
|
2008 |
16 |
4 |
p. 1702-1720 19 p. |
artikel |
11 |
Corrugoside, a new immunostimulatory α-galactoglycosphingolipid from the marine sponge Axinella corrugata
|
Costantino, Valeria |
|
2008 |
16 |
4 |
p. 2077-2085 9 p. |
artikel |
12 |
Design and synthesis of a siderophore conjugate as a potent PSMA inhibitor and potential diagnostic agent for prostate cancer
|
Ding, Pingyu |
|
2008 |
16 |
4 |
p. 1648-1657 10 p. |
artikel |
13 |
Design and synthesis of DPP-IV inhibitors lacking the electrophilic nitrile group
|
Kondo, Takashi |
|
2008 |
16 |
4 |
p. 1613-1631 19 p. |
artikel |
14 |
Design of azidoproline containing gluten peptides to suppress CD4+ T-cell responses associated with Celiac disease
|
Kapoerchan, Varsha V. |
|
2008 |
16 |
4 |
p. 2053-2062 10 p. |
artikel |
15 |
Design, Synthesis and Evaluation of Antiinflammatory, Analgesic and Ulcerogenicity studies of Novel S-Substituted phenacyl-1,3,4-oxadiazole-2-thiol and Schiff bases of Diclofenac acid as Nonulcerogenic Derivatives
|
Bhandari, Shashikant V. |
|
2008 |
16 |
4 |
p. 1822-1831 10 p. |
artikel |
16 |
Editorial board
|
|
|
2008 |
16 |
4 |
p. IFC- 1 p. |
artikel |
17 |
Estradiol and estrone C-16 derivatives as inhibitors of type 1 17β-hydroxysteroid dehydrogenase: Blocking of ER+ breast cancer cell proliferation induced by estrone
|
Laplante, Yannick |
|
2008 |
16 |
4 |
p. 1849-1860 12 p. |
artikel |
18 |
5,5,6-Fused tricycles bearing imidazole and pyrazole 6-methylidene penems as broad-spectrum inhibitors of β-lactamases
|
Venkatesan, Aranapakam M. |
|
2008 |
16 |
4 |
p. 1890-1902 13 p. |
artikel |
19 |
Graphical contents list
|
|
|
2008 |
16 |
4 |
p. 1549-1561 13 p. |
artikel |
20 |
Influence of heterocyclic and oxime-containing farnesol analogs on quorum sensing and pathogenicity in Candida albicans
|
Shchepin, Roman |
|
2008 |
16 |
4 |
p. 1842-1848 7 p. |
artikel |
21 |
Influence of sulfur oxidation state and steric bulk upon trifluoromethyl ketone (TFK) binding kinetics to carboxylesterases and fatty acid amide hydrolase (FAAH)
|
Wheelock, Craig E. |
|
2008 |
16 |
4 |
p. 2114-2130 17 p. |
artikel |
22 |
Inhibitors of proteases and amide hydrolases that employ an α-ketoheterocycle as a key enabling functionality
|
Maryanoff, Bruce E. |
|
2008 |
16 |
4 |
p. 1562-1595 34 p. |
artikel |
23 |
Instructions to contributors
|
|
|
2008 |
16 |
4 |
p. I- 1 p. |
artikel |
24 |
Iromycins from Streptomyces sp. and from synthesis: New inhibitors of the mitochondrial electron transport chain
|
Surup, Frank |
|
2008 |
16 |
4 |
p. 1738-1746 9 p. |
artikel |
25 |
New QSAR combined strategy for the design of A1 adenosine receptor agonists
|
González, Maykel Pérez |
|
2008 |
16 |
4 |
p. 1658-1675 18 p. |
artikel |
26 |
New 1,2,3,4-tetrahydroisoquinoline derivatives as modulators of proteolytic cleavage of amyloid precursor proteins
|
Hu, Ming-Kuan |
|
2008 |
16 |
4 |
p. 1957-1965 9 p. |
artikel |
27 |
Novel anti-HIV cyclotriazadisulfonamide derivatives as modeled by ligand- and receptor-based approaches
|
Pinheiro, Júlia R. |
|
2008 |
16 |
4 |
p. 1683-1690 8 p. |
artikel |
28 |
N6-substituted C5′-modified adenosines as A1 adenosine receptor agonists
|
Ashton, T.D. |
|
2008 |
16 |
4 |
p. 1861-1873 13 p. |
artikel |
29 |
Orally active 1,2,4-trioxepanes: Synthesis and antimalarial activity of a series of 7-arylvinyl-1,2,4-trioxepanes against multidrug-resistant Plasmodium yoelii in Swiss mice
|
Singh, Chandan |
|
2008 |
16 |
4 |
p. 1816-1821 6 p. |
artikel |
30 |
Oxazaborolidine derivatives inducing autoinducer-2 signal transduction in Vibrio harveyi
|
Aharoni, R. |
|
2008 |
16 |
4 |
p. 1596-1604 9 p. |
artikel |
31 |
Phenylalanine-containing hydroxamic acids as selective inhibitors of class IIb histone deacetylases (HDACs)
|
Schäfer, Stefan |
|
2008 |
16 |
4 |
p. 2011-2033 23 p. |
artikel |
32 |
Potent and selective small molecule NS3 serine protease inhibitors of Hepatitis C virus with dichlorocyclopropylproline as P2 residue
|
Chen, Kevin X. |
|
2008 |
16 |
4 |
p. 1874-1883 10 p. |
artikel |
33 |
Properties of flaky affinity resin with co-continuous structure
|
Mori, Tomoko |
|
2008 |
16 |
4 |
p. 1983-1991 9 p. |
artikel |
34 |
Protein phosphatase inhibitory activity of tautomycin photoaffinity probes evaluated at femto-molar level
|
Sydnes, Magne O. |
|
2008 |
16 |
4 |
p. 1747-1755 9 p. |
artikel |
35 |
Selection and characterization of human antibodies neutralizing Bacillus anthracis toxin
|
Zhou, Bin |
|
2008 |
16 |
4 |
p. 1903-1913 11 p. |
artikel |
36 |
Synthesis, adenosine receptor binding and 3D-QSAR of 4-substituted 2-(2′-furyl)-1,2,4-triazolo[1,5-a]quinoxalines
|
Martínez, Ana |
|
2008 |
16 |
4 |
p. 2103-2113 11 p. |
artikel |
37 |
Synthesis and cyclooxygenase inhibitory activities of linear 1-(methanesulfonylphenyl or benzenesulfonamido)-2-(pyridyl)acetylene regioisomers
|
Chowdhury, Morshed Alam |
|
2008 |
16 |
4 |
p. 1948-1956 9 p. |
artikel |
38 |
Synthesis and structure–activity relationships of a series of substituted 2-(1H-furo[2,3-g]indazol-1-yl)ethylamine derivatives as 5-HT2C receptor agonists
|
Shimada, Itsuro |
|
2008 |
16 |
4 |
p. 1966-1982 17 p. |
artikel |
39 |
Synthesis and structure–activity relationships of 16-ene-22-thia-1α,25-dihydroxy-26,27-dimethyl-19-norvitamin D3 analogs having side chains of different sizes
|
Takaku, Hajime |
|
2008 |
16 |
4 |
p. 1796-1815 20 p. |
artikel |
40 |
Synthesis, biological evaluation and molecular modelling studies of methyleneimidazole substituted biaryls as inhibitors of human 17α-hydroxylase-17,20-lyase (CYP17). Part I: Heterocyclic modifications of the core structure
|
Jagusch, Carsten |
|
2008 |
16 |
4 |
p. 1992-2010 19 p. |
artikel |
41 |
Synthesis, characterization and antiproliferative studies of the enantiomers of cis-[(1,2-camphordiamine)dichloro]platinum(II) complexes
|
Montaña, Ángel M. |
|
2008 |
16 |
4 |
p. 1721-1737 17 p. |
artikel |
42 |
Synthesis, metal ion binding, and biological evaluation of new anticancer 2-(2′-hydroxyphenyl)benzoxazole analogs of UK-1
|
McKee, Mireya L. |
|
2008 |
16 |
4 |
p. 1775-1783 9 p. |
artikel |
43 |
Synthesis of (nor)tropeine (di)esters and allosteric modulation of glycine receptor binding
|
Maksay, Gábor |
|
2008 |
16 |
4 |
p. 2086-2092 7 p. |
artikel |
44 |
Synthesis of novel spirostanic saponins and their cytotoxic activity
|
Hernández, Juan C. |
|
2008 |
16 |
4 |
p. 2063-2076 14 p. |
artikel |
45 |
Targeting the inverted CCAAT Box-2 of the topoisomerase IIα gene: DNA sequence selective recognition by a polyamide–intercalator as a staggered dimer
|
Mackay, Hilary |
|
2008 |
16 |
4 |
p. 2093-2102 10 p. |
artikel |
46 |
The effect of flavonoid derivatives on doxorubicin transport and metabolism
|
Václavíková, Radka |
|
2008 |
16 |
4 |
p. 2034-2042 9 p. |
artikel |
47 |
The synthesis of bivalent 2β-carbomethoxy-3β-(3,4-dichlorophenyl)-8-heterobicyclo[3.2.1]octanes as probes for proximal binding sites on the dopamine and serotonin transporters
|
Meltzer, Peter C. |
|
2008 |
16 |
4 |
p. 1832-1841 10 p. |
artikel |
48 |
Toward the development of chemoprevention agents (III): Synthesis and anti-inflammatory activities of a new class of 5-glycylamino-2-substituted-phenyl-1,3-dioxacycloalkanes
|
Bi, Lanrong |
|
2008 |
16 |
4 |
p. 1764-1774 11 p. |
artikel |
49 |
Trypanocidal activity of a new pterocarpan and other secondary metabolites of plants from Northeastern Brazil flora
|
Vieira, Nashira Campos |
|
2008 |
16 |
4 |
p. 1676-1682 7 p. |
artikel |
50 |
Virtual screening approaches for the identification of non-lipid autotaxin inhibitors
|
Parrill, Abby L. |
|
2008 |
16 |
4 |
p. 1784-1795 12 p. |
artikel |