| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
Allele-specific inhibition of divergent protein tyrosine phosphatases with a single small molecule
|
Zhang, Xin-Yu
|
|
2008
|
16 |
17 |
p. 8090-8097
8 p.
|
artikel
|
| 2 |
A new synthetic access to furo[3,2-f]chromene analogues of an antimycobacterial
|
Alvey, Luke
|
|
2008
|
16 |
17 |
p. 8264-8272
9 p.
|
artikel
|
| 3 |
Antibacterial profile against drug-resistant Staphylococcus epidermidis clinical strain and structure–activity relationship studies of 1H-pyrazolo[3,4-b]pyridine and thieno[2,3-b]pyridine derivatives
|
Leal, Bruno
|
|
2008
|
16 |
17 |
p. 8196-8204
9 p.
|
artikel
|
| 4 |
Antifungal activity of synthetic di(hetero)arylamines based on the benzo[b]thiophene moiety
|
Pinto, Eugénia
|
|
2008
|
16 |
17 |
p. 8172-8177
6 p.
|
artikel
|
| 5 |
Anti-HIV-1 activity of phloroglucinol derivative, 6,6′-bieckol, from Ecklonia cava
|
Artan, Murat
|
|
2008
|
16 |
17 |
p. 7921-7926
6 p.
|
artikel
|
| 6 |
Antiproliferative and apoptosis-inducing activities of alkyl gallate and gallamide derivatives related to (−)-epigallocatechin gallate
|
Dodo, Kosuke
|
|
2008
|
16 |
17 |
p. 7975-7982
8 p.
|
artikel
|
| 7 |
Characterization of the binding properties of SIRT2 inhibitors with a N-(3-phenylpropenoyl)-glycine tryptamide backbone
|
Kiviranta, Päivi H.
|
|
2008
|
16 |
17 |
p. 8054-8062
9 p.
|
artikel
|
| 8 |
Chemoenzymatic syntheses of prenylated aromatic small molecules using Streptomyces prenyltransferases with relaxed substrate specificities
|
Kumano, Takuto
|
|
2008
|
16 |
17 |
p. 8117-8126
10 p.
|
artikel
|
| 9 |
5-(4-Chlorophenyl)-5,6-dihydro-1,3-oxazepin-7(4H)-one derivatives as lipophilic cyclic analogues of baclofen: Design, synthesis, and neuropharmacological evaluation
|
Abdel-Hafez, Atef A.
|
|
2008
|
16 |
17 |
p. 7983-7991
9 p.
|
artikel
|
| 10 |
Comparative docking studies of labdane-type diterpenes with forskolin at the active site of adenylyl cyclase
|
Koukoulitsa, Catherine
|
|
2008
|
16 |
17 |
p. 8237-8243
7 p.
|
artikel
|
| 11 |
Computer based design, synthesis and biological evaluation of novel indole derivatives as HCV NS3-4A serine protease inhibitors
|
Ismail, Nasser S.M.
|
|
2008
|
16 |
17 |
p. 7877-7887
11 p.
|
artikel
|
| 12 |
Cyclic voltammetric analysis of 2-styrylchromones: Relationship with the antioxidant activity
|
Gomes, Ana
|
|
2008
|
16 |
17 |
p. 7939-7943
5 p.
|
artikel
|
| 13 |
Design and SAR of new substituted purines bearing aryl groups at N9 position as HIV-1 Tat–TAR interaction inhibitors
|
Pang, Ruifang
|
|
2008
|
16 |
17 |
p. 8178-8186
9 p.
|
artikel
|
| 14 |
Design and synthesis of a metabolically stable and potent antitussive agent, a novel δ opioid receptor antagonist, TRK-851
|
Sakami, Satoshi
|
|
2008
|
16 |
17 |
p. 7956-7967
12 p.
|
artikel
|
| 15 |
Design and synthesis of carborane-containing androgen receptor (AR) antagonist bearing a pyridine ring
|
Ohta, Kiminori
|
|
2008
|
16 |
17 |
p. 8022-8028
7 p.
|
artikel
|
| 16 |
Design, synthesis, and acetylcholinesterase inhibitory activity of novel coumarin analogues
|
Zhou, Xiang
|
|
2008
|
16 |
17 |
p. 8011-8021
11 p.
|
artikel
|
| 17 |
Design, synthesis, and antitumor activity of new bis-aminomethylnaphthalenes
|
Bollini, Mariela
|
|
2008
|
16 |
17 |
p. 8003-8010
8 p.
|
artikel
|
| 18 |
Design, synthesis and biological evaluation of dihydronaphthalene and benzosuberene analogs of the combretastatins as inhibitors of tubulin polymerization in cancer chemotherapy
|
Sriram, Madhavi
|
|
2008
|
16 |
17 |
p. 8161-8171
11 p.
|
artikel
|
| 19 |
Design, synthesis and biological evaluation of novel compounds with conjugated structure as anti-tumor agents
|
Su, Hong
|
|
2008
|
16 |
17 |
p. 7992-8002
11 p.
|
artikel
|
| 20 |
Editorial board
|
|
|
2008
|
16 |
17 |
p. IFC-
1 p.
|
artikel
|
| 21 |
Furoxan-, alkylnitrate-derivatives and related compounds as anti-trypanosomatid agents: Mechanism of action studies
|
Boiani, Lucı´a
|
|
2008
|
16 |
17 |
p. 7900-7907
8 p.
|
artikel
|
| 22 |
Graphical contents list
|
|
|
2008
|
16 |
17 |
p. 7863-7876
14 p.
|
artikel
|
| 23 |
Hybridization-dependent fluorescence of oligodeoxynucleotides incorporating new pyrene-modified adenosine residues
|
Seio, Kohji
|
|
2008
|
16 |
17 |
p. 8287-8293
7 p.
|
artikel
|
| 24 |
Identification of SVM-based classification model, synthesis and evaluation of prenylated flavonoids as vasorelaxant agents
|
Dong, Xiaowu
|
|
2008
|
16 |
17 |
p. 8151-8160
10 p.
|
artikel
|
| 25 |
Instructions to contributors
|
|
|
2008
|
16 |
17 |
p. I-
1 p.
|
artikel
|
| 26 |
In vitro antifungal activity of polyfunctionalized 2-(hetero)arylquinolines prepared through imino Diels–Alder reactions
|
Meléndez Gómez, Carlos M.
|
|
2008
|
16 |
17 |
p. 7908-7920
13 p.
|
artikel
|
| 27 |
Molecular modeling and dynamics studies of Shikimate Kinase from Bacillus anthracis
|
Pauli, Ivani
|
|
2008
|
16 |
17 |
p. 8098-8108
11 p.
|
artikel
|
| 28 |
Monoquaternary pyridinium salts with modified side chain—synthesis and evaluation on model of tabun- and paraoxon-inhibited acetylcholinesterase
|
Musilek, Kamil
|
|
2008
|
16 |
17 |
p. 8218-8223
6 p.
|
artikel
|
| 29 |
New QSPR study for the prediction of aqueous solubility of drug-like compounds
|
Duchowicz, Pablo R.
|
|
2008
|
16 |
17 |
p. 7944-7955
12 p.
|
artikel
|
| 30 |
NO-donors. Part 17 1 : Synthesis and antimicrobial activity of novel ketoconazole–NO-donor hybrid compounds
|
Konter, Joerg
|
|
2008
|
16 |
17 |
p. 8294-8300
7 p.
|
artikel
|
| 31 |
Novel azolyl-(phenylmethyl)]aryl/heteroarylamines: Potent CYP26 inhibitors and enhancers of all-trans retinoic acid activity in neuroblastoma cells
|
Gomaa, Mohamed Sayed
|
|
2008
|
16 |
17 |
p. 8301-8313
13 p.
|
artikel
|
| 32 |
Novel synthesis and pharmacological evaluation as α2-adrenoceptor ligands of O-phenylisouronium salts
|
Goonan, Áine
|
|
2008
|
16 |
17 |
p. 8210-8217
8 p.
|
artikel
|
| 33 |
N-Propynyl analogs of β-phenylethylidenehydrazines: Synthesis and evaluation of effects on glycine, GABA, and monoamine oxidase
|
MacKenzie, Erin M.
|
|
2008
|
16 |
17 |
p. 8254-8263
10 p.
|
artikel
|
| 34 |
Pestalachlorides A–C, antifungal metabolites from the plant endophytic fungus Pestalotiopsis adusta
|
Li, Erwei
|
|
2008
|
16 |
17 |
p. 7894-7899
6 p.
|
artikel
|
| 35 |
Potent CCR4 antagonists: Synthesis, evaluation, and docking study of 2,4-diaminoquinazolines
|
Yokoyama, Kazuhiro
|
|
2008
|
16 |
17 |
p. 7968-7974
7 p.
|
artikel
|
| 36 |
Quantitative structure–activity relationship studies on nitrofuranyl anti-tubercular agents
|
Hevener, Kirk E.
|
|
2008
|
16 |
17 |
p. 8042-8053
12 p.
|
artikel
|
| 37 |
Spin trapping experiments with different carbamoyl-substituted EMPO derivatives
|
Stolze, Klaus
|
|
2008
|
16 |
17 |
p. 8082-8089
8 p.
|
artikel
|
| 38 |
Stress-driven discovery of metabolites from the phytopathogenic fungus Leptosphaeria maculans: Structure and activity of leptomaculins A–E
|
Pedras, M. Soledade C.
|
|
2008
|
16 |
17 |
p. 8063-8071
9 p.
|
artikel
|
| 39 |
Structure–activity relationships of new inhibitors of breast cancer resistance protein (ABCG2)
|
Pick, Anne
|
|
2008
|
16 |
17 |
p. 8224-8236
13 p.
|
artikel
|
| 40 |
Syntheses and anti-depressant activity of 5-amino-1, 3, 4-thiadiazole-2-thiol imines and thiobenzyl derivatives
|
Yusuf, Mohammad
|
|
2008
|
16 |
17 |
p. 8029-8034
6 p.
|
artikel
|
| 41 |
Synthesis and antimicrobial activity of dermaseptin S1 analogues
|
Savoia, Dianella
|
|
2008
|
16 |
17 |
p. 8205-8209
5 p.
|
artikel
|
| 42 |
Synthesis and antiproliferative activity in vitro of novel (2-butynyl)thioquinolines
|
Mól, W.
|
|
2008
|
16 |
17 |
p. 8136-8141
6 p.
|
artikel
|
| 43 |
Synthesis and bio-evaluation of a new fatty acid derivative for myocardial imaging
|
Mathur, Anupam
|
|
2008
|
16 |
17 |
p. 7927-7931
5 p.
|
artikel
|
| 44 |
Synthesis and biological evaluation of glucuronide prodrugs of the histone deacetylase inhibitor CI-994 for application in selective cancer chemotherapy
|
Thomas, Mickaël
|
|
2008
|
16 |
17 |
p. 8109-8116
8 p.
|
artikel
|
| 45 |
Synthesis and elastase-inhibiting activity of 2-pyridinyl-isothiazol-3(2H)-one 1,1-dioxides
|
Eilfeld, Alexander
|
|
2008
|
16 |
17 |
p. 8127-8135
9 p.
|
artikel
|
| 46 |
Synthesis and evaluation of curcumin analogues as potential thioredoxin reductase inhibitors
|
Qiu, Xu
|
|
2008
|
16 |
17 |
p. 8035-8041
7 p.
|
artikel
|
| 47 |
Synthesis and structure–activity relationship studies of theophylline analogs on population responses in the rat hippocampus in vitro
|
Ananthalakshmi, Kethireddy V.V.
|
|
2008
|
16 |
17 |
p. 8142-8150
9 p.
|
artikel
|
| 48 |
Synthesis, in vitro, and in vivo biological evaluation and molecular docking simulations of chiral alcohol and ether derivatives of the 1,5-diarylpyrrole scaffold as novel anti-inflammatory and analgesic agents
|
Biava, Mariangela
|
|
2008
|
16 |
17 |
p. 8072-8081
10 p.
|
artikel
|
| 49 |
Synthesis of both enantiomers of hydroxypipecolic acid derivatives equivalent to 5-azapyranuronic acids and evaluation of their inhibitory activities against glycosidases
|
Yoshimura, Yuichi
|
|
2008
|
16 |
17 |
p. 8273-8286
14 p.
|
artikel
|
| 50 |
Synthesis of new sulfonyl pyrrolidine derivatives as matrix metalloproteinase inhibitors
|
Cheng, Xian-Chao
|
|
2008
|
16 |
17 |
p. 7932-7938
7 p.
|
artikel
|
| 51 |
Synthesis, structural studies and biological properties of new TBA analogues containing an acyclic nucleotide
|
Coppola, Teresa
|
|
2008
|
16 |
17 |
p. 8244-8253
10 p.
|
artikel
|
| 52 |
The efficacy and selectivity of tumor cell killing by Akt inhibitors are substantially increased by chloroquine
|
Hu, Changkun
|
|
2008
|
16 |
17 |
p. 7888-7893
6 p.
|
artikel
|
| 53 |
Thiazolidinone CFTR inhibitors with improved water solubility identified by structure–activity analysis
|
Sonawane, N.D.
|
|
2008
|
16 |
17 |
p. 8187-8195
9 p.
|
artikel
|
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