| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
A novel Syk family kinase inhibitor: Design, synthesis, and structure–activity relationship of 1,2,4-triazolo[4,3-c]pyrimidine and 1,2,4-triazolo[1,5-c]pyrimidine derivatives
|
Hirabayashi, Akihito
|
|
2008
|
16 |
15 |
p. 7347-7357
11 p.
|
artikel
|
| 2 |
Anticonvulsant activity of some xanthone derivatives
|
Marona, Henryk
|
|
2008
|
16 |
15 |
p. 7234-7244
11 p.
|
artikel
|
| 3 |
Aromatic 2-chloroethyl urea derivatives and bioisosteres. Part 2: Cytocidal activity and effects on the nuclear translocation of thioredoxin-1, and the cell cycle progression
|
Fortin, Jessica S.
|
|
2008
|
16 |
15 |
p. 7477-7488
12 p.
|
artikel
|
| 4 |
Baicalin, a prodrug able to reach the CNS, is a prolyl oligopeptidase inhibitor
|
Tarragó, Teresa
|
|
2008
|
16 |
15 |
p. 7516-7524
9 p.
|
artikel
|
| 5 |
Bis(sulfonamide) isosters of mycophenolic adenine dinucleotide analogues: Inhibition of inosine monophosphate dehydrogenase
|
Chen, Liqiang
|
|
2008
|
16 |
15 |
p. 7462-7469
8 p.
|
artikel
|
| 6 |
Carbonic anhydrase inhibitors: Inhibition of mammalian isoforms I–XIV with a series of substituted phenols including paracetamol and salicylic acid
|
Innocenti, Alessio
|
|
2008
|
16 |
15 |
p. 7424-7428
5 p.
|
artikel
|
| 7 |
Characterization of the PON1 active site using modeling simulation, in relation to PON1 lactonase activity
|
Tavori, Hagai
|
|
2008
|
16 |
15 |
p. 7504-7509
6 p.
|
artikel
|
| 8 |
Cinnamoyl- and hydroxycinnamoyl amides of glaucine and their antioxidative and antiviral activities
|
Spasova, Maya
|
|
2008
|
16 |
15 |
p. 7457-7461
5 p.
|
artikel
|
| 9 |
Comparative molecular dynamics simulations of the potent synthetic classical cannabinoid ligand AMG3 in solution and at binding site of the CB1 and CB2 receptors
|
Durdagi, Serdar
|
|
2008
|
16 |
15 |
p. 7377-7387
11 p.
|
artikel
|
| 10 |
Design and synthesis of novel oxazole containing 1,3-Dioxane-2-carboxylic acid derivatives as PPAR α/γ dual agonists
|
Pingali, Harikishore
|
|
2008
|
16 |
15 |
p. 7117-7127
11 p.
|
artikel
|
| 11 |
Design, synthesis, and biological evaluation of Mannich bases of heterocyclic chalcone analogs as cytotoxic agents
|
Reddy, M. Vijaya Bhaskar
|
|
2008
|
16 |
15 |
p. 7358-7370
13 p.
|
artikel
|
| 12 |
Design, synthesis, and biological evaluation of pirenzepine analogs bearing a 1,2-cyclohexanediamine and perhydroquinoxaline units in exchange for the piperazine ring as antimuscarinics
|
Minarini, Anna
|
|
2008
|
16 |
15 |
p. 7311-7320
10 p.
|
artikel
|
| 13 |
Design, synthesis, and evaluation of 3C protease inhibitors as anti-enterovirus 71 agents
|
Kuo, Chih-Jung
|
|
2008
|
16 |
15 |
p. 7388-7398
11 p.
|
artikel
|
| 14 |
Discovery and stereoselective synthesis of the novel isochroman neurokinin-1 receptor antagonist ‘CJ-17,493’
|
Shishido, Yuji
|
|
2008
|
16 |
15 |
p. 7193-7205
13 p.
|
artikel
|
| 15 |
Editorial board
|
|
|
2008
|
16 |
15 |
p. IFC-
1 p.
|
artikel
|
| 16 |
Enhanced affinity of ketotifen toward tamarind seed polysaccharide in comparison with hydroxyethylcellulose and hyaluronic acid: A nuclear magnetic resonance investigation
|
Uccello-Barretta, Gloria
|
|
2008
|
16 |
15 |
p. 7371-7376
6 p.
|
artikel
|
| 17 |
Fluorinated phenylcyclopropylamines. Part 5: Effects of electron-withdrawing or -donating aryl substituents on the inhibition of monoamine oxidases A and B by 2-aryl-2-fluoro-cyclopropylamines
|
Hruschka, Svenja
|
|
2008
|
16 |
15 |
p. 7148-7166
19 p.
|
artikel
|
| 18 |
Functionalized pyrrolidine inhibitors of human type II α-mannosidases as anti-cancer agents: Optimizing the fit to the active site
|
Fiaux, Hélène
|
|
2008
|
16 |
15 |
p. 7337-7346
10 p.
|
artikel
|
| 19 |
Graphical contents list
|
|
|
2008
|
16 |
15 |
p. 7081-7094
14 p.
|
artikel
|
| 20 |
Hanultarin, a cytotoxic lignan as an inhibitor of actin cytoskeleton polymerization from the seeds of Trichosanthes kirilowii
|
Moon, Surk-Sik
|
|
2008
|
16 |
15 |
p. 7264-7269
6 p.
|
artikel
|
| 21 |
Homo- and hetero-bivalent edrophonium-like ammonium salts as highly potent, dual binding site AChE inhibitors
|
Leonetti, Francesco
|
|
2008
|
16 |
15 |
p. 7450-7456
7 p.
|
artikel
|
| 22 |
Identification of a butyrophenone analog as a potential atypical antipsychotic agent: 4-[4-(4-Chlorophenyl)-1,4-diazepan-1-yl]-1-(4-fluorophenyl)butan-1-one
|
Ablordeppey, Seth Y.
|
|
2008
|
16 |
15 |
p. 7291-7301
11 p.
|
artikel
|
| 23 |
Identification of a methotrexate-binding peptide from a T7 phage display screen using a QCM device
|
Takakusagi, Yoichi
|
|
2008
|
16 |
15 |
p. 7410-7414
5 p.
|
artikel
|
| 24 |
Illudalic acid as a potential LAR inhibitor: Synthesis, SAR, and preliminary studies on the mechanism of action
|
Ling, Qing
|
|
2008
|
16 |
15 |
p. 7399-7409
11 p.
|
artikel
|
| 25 |
Instructions to contributors
|
|
|
2008
|
16 |
15 |
p. I-
1 p.
|
artikel
|
| 26 |
In vitro inhibition of glycogen-degrading enzymes and glycosidases by six-membered sugar mimics and their evaluation in cell cultures
|
Kuriyama, Chinami
|
|
2008
|
16 |
15 |
p. 7330-7336
7 p.
|
artikel
|
| 27 |
Lack of aquaporin-4 water transport inhibition by antiepileptics and arylsulfonamides
|
Yang, Baoxue
|
|
2008
|
16 |
15 |
p. 7489-7493
5 p.
|
artikel
|
| 28 |
Major sperm protein as a diagnostic antigen for onchocerciasis
|
Park, Junguk
|
|
2008
|
16 |
15 |
p. 7206-7209
4 p.
|
artikel
|
| 29 |
Molecular features of the prazosin molecule required for activation of Transport-P
|
da Silva, Joaquim Fernando Mendes
|
|
2008
|
16 |
15 |
p. 7254-7263
10 p.
|
artikel
|
| 30 |
Muscarinic receptor 1 agonist activity of novel N-arylthioureas substituted 3-morpholino arecoline derivatives in Alzheimer’s presenile dementia models
|
Malviya, Manish
|
|
2008
|
16 |
15 |
p. 7095-7101
7 p.
|
artikel
|
| 31 |
Nitrogen-containing flavonoid analogues as CDK1/cyclin B inhibitors: Synthesis, SAR analysis, and biological activity
|
Zhang, Shixuan
|
|
2008
|
16 |
15 |
p. 7127-7132
6 p.
|
artikel
|
| 32 |
Novel inhibitors of anthrax edema factor
|
Chen, Deliang
|
|
2008
|
16 |
15 |
p. 7225-7233
9 p.
|
artikel
|
| 33 |
Novel N1-substituted 1,3-dihydro-2H-benzimidazol-2-ones as potent non-nucleoside reverse transcriptase inhibitors
|
Monforte, Anna-Maria
|
|
2008
|
16 |
15 |
p. 7429-7435
7 p.
|
artikel
|
| 34 |
Novel sterically hindered cannabinoid CB1 receptor ligands
|
Urbani, Paolo
|
|
2008
|
16 |
15 |
p. 7510-7515
6 p.
|
artikel
|
| 35 |
Phenyl phosphotriester derivatives of AZT: Variations upon the SATE moiety
|
Villard, Anne-Laure
|
|
2008
|
16 |
15 |
p. 7321-7329
9 p.
|
artikel
|
| 36 |
QSAR prediction of inhibition of aldose reductase for flavonoids
|
Mercader, Andrew G.
|
|
2008
|
16 |
15 |
p. 7470-7476
7 p.
|
artikel
|
| 37 |
QSAR study of imidazoline antihypertensive drugs
|
Nikolic, Katarina
|
|
2008
|
16 |
15 |
p. 7134-7140
7 p.
|
artikel
|
| 38 |
Remarkable DNA binding affinity and potential anticancer activity of pyrrolo[2,1-c][1,4]benzodiazepine–naphthalimide conjugates linked through piperazine side-armed alkane spacers
|
Kamal, Ahmed
|
|
2008
|
16 |
15 |
p. 7218-7224
7 p.
|
artikel
|
| 39 |
Selective alkylation of βII-tubulin and thioredoxin-1 by structurally related subsets of aryl chloroethylureas leading to either anti-microtubules or redox modulating agents
|
Fortin, Jessica S.
|
|
2008
|
16 |
15 |
p. 7277-7290
14 p.
|
artikel
|
| 40 |
Single-stranded DNA aptamers specific for antibiotics tetracyclines
|
Niazi, Javed H.
|
|
2008
|
16 |
15 |
p. 7245-7253
9 p.
|
artikel
|
| 41 |
Structure–activity correlations for β-phenethylamines at human trace amine receptor 1
|
Lewin, Anita H.
|
|
2008
|
16 |
15 |
p. 7415-7423
9 p.
|
artikel
|
| 42 |
Structure–activity relationship of flavonoids as influenza virus neuraminidase inhibitors and their in vitro anti-viral activities
|
Liu, Ai-Lin
|
|
2008
|
16 |
15 |
p. 7141-7147
7 p.
|
artikel
|
| 43 |
Sulfur-substituted naphthalimides as photoactivatable anticancer agents: DNA interaction, fluorescence imaging, and phototoxic effects in cultured tumor cells
|
Ott, Ingo
|
|
2008
|
16 |
15 |
p. 7107-7116
10 p.
|
artikel
|
| 44 |
Syntheses of phosphatidyl-β-d-glucoside analogues to probe antigen selectivity of monoclonal antibody ‘DIM21’
|
Greimel, Peter
|
|
2008
|
16 |
15 |
p. 7210-7217
8 p.
|
artikel
|
| 45 |
Synthesis and antiviral evaluation of some new pyrazole and fused pyrazolopyrimidine derivatives
|
Rashad, Aymn E.
|
|
2008
|
16 |
15 |
p. 7102-7106
5 p.
|
artikel
|
| 46 |
Synthesis and biological evaluation of new disubstituted analogues of 6-methoxy-3-(3′,4′,5′-trimethoxybenzoyl)-1H-indole (BPR0L075), as potential antivascular agents
|
Ty, Nancy
|
|
2008
|
16 |
15 |
p. 7494-7503
10 p.
|
artikel
|
| 47 |
Synthesis and cytotoxic, anti-inflammatory, and anti-oxidant activities of 2′,5′-dialkoxylchalcones as cancer chemopreventive agents
|
Cheng, Jen-Hao
|
|
2008
|
16 |
15 |
p. 7270-7276
7 p.
|
artikel
|
| 48 |
Synthesis and evaluation of pyrazolo[3,4-b]pyridines and its structural analogues as TNF-α and IL-6 inhibitors
|
Bharate, Sandip B.
|
|
2008
|
16 |
15 |
p. 7167-7176
10 p.
|
artikel
|
| 49 |
Synthesis, DNA binding, and cytotoxic evaluation of new analogs of diallyldisulfide, an active principle of garlic
|
Rai, Santosh Kumar
|
|
2008
|
16 |
15 |
p. 7302-7310
9 p.
|
artikel
|
| 50 |
Synthesis, inhibitory activities, and QSAR study of xanthone derivatives as α-glucosidase inhibitors
|
Liu, Yan
|
|
2008
|
16 |
15 |
p. 7185-7192
8 p.
|
artikel
|
| 51 |
Synthesis of 3′-deoxy-3′-C-methyl nucleoside derivatives
|
Aljarah, Mohamed
|
|
2008
|
16 |
15 |
p. 7436-7442
7 p.
|
artikel
|
| 52 |
Synthesis of scyllo-inositol derivatives and their effects on amyloid beta peptide aggregation
|
Sun, Yedi
|
|
2008
|
16 |
15 |
p. 7177-7184
8 p.
|
artikel
|
| 53 |
The discovery of small molecule chemical probes of Bcl-XL and Mcl-1
|
Prakesch, Michael
|
|
2008
|
16 |
15 |
p. 7443-7449
7 p.
|
artikel
|
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