| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
5-Alkyl-2-alkylamino-6-(2,6-difluorophenylalkyl)-3,4-dihydropyrimidin-4(3H)-ones, a new series of potent, broad-spectrum non-nucleoside reverse transcriptase inhibitors belonging to the DABO family
|
Mai, Antonello
|
|
2005
|
13 |
6 |
p. 2065-2077
13 p.
|
artikel
|
| 2 |
3-Aminomethyl derivatives of 4,11-dihydroxynaphtho[2,3-f]indole-5,10-dione for circumvention of anticancer drug resistance
|
Shchekotikhin, Andrey E.
|
|
2005
|
13 |
6 |
p. 2285-2291
7 p.
|
artikel
|
| 3 |
A novel method of estimation of lipophilicity using distance-based topological indices: dominating role of equalized electronegativity
|
Agrawal, Vijay K.
|
|
2005
|
13 |
6 |
p. 2109-2120
12 p.
|
artikel
|
| 4 |
Antitumor agents 243. Syntheses and cytotoxicity of desmosdumotin C derivatives
|
Nakagawa-Goto, Kyoko
|
|
2005
|
13 |
6 |
p. 2325-2330
6 p.
|
artikel
|
| 5 |
A physically interpretable quantum-theoretic QSAR for some carbonic anhydrase inhibitors with diverse aromatic rings, obtained by a new QSAR procedure
|
Clare, Brian W.
|
|
2005
|
13 |
6 |
p. 2197-2211
15 p.
|
artikel
|
| 6 |
1-Aryl-4-(4-succinimidobutyl)piperazines and their conformationally constrained analogues: synthesis, binding to serotonin (5-HT1A, 5-HT2A, 5-HT7), α1-adrenergic, and dopaminergic D2 receptors, and in vivo 5-HT1A functional characteristics
|
Bojarski, Andrzej J.
|
|
2005
|
13 |
6 |
p. 2293-2303
11 p.
|
artikel
|
| 7 |
Comparative molecular similarity indices analysis (CoMSIA) studies of 1,2-naphthoquinone derivatives as PTP1B inhibitors
|
Sobhia, M. Elizabeth
|
|
2005
|
13 |
6 |
p. 2331-2338
8 p.
|
artikel
|
| 8 |
Conformational restrictions in ligand binding to the human intestinal di-/tripeptide transporter: implications for design of hPEPT1 targeted prodrugs
|
Våbenø, Jon
|
|
2005
|
13 |
6 |
p. 1977-1988
12 p.
|
artikel
|
| 9 |
Contributors to this issue
|
|
|
2005
|
13 |
6 |
p. I-II
nvt p.
|
artikel
|
| 10 |
Cooperative lectin recognition of periodical glycoclusters along DNA duplexes: alternate hybridization and full hybridization
|
Yamada, Yoshinao
|
|
2005
|
13 |
6 |
p. 1913-1922
10 p.
|
artikel
|
| 11 |
Core-modified porphyrins. Part 4: Steric effects on photophysical and biological properties in vitro
|
You, Youngjae
|
|
2005
|
13 |
6 |
p. 2235-2251
17 p.
|
artikel
|
| 12 |
Design and synthesis of an optimized positional scanning library of peptoids: identification of novel multidrug resistance reversal agents
|
Masip, Isabel
|
|
2005
|
13 |
6 |
p. 1923-1929
7 p.
|
artikel
|
| 13 |
Design and synthesis of new antimalarial agents from 4-aminoquinoline
|
Solomon, V. Raja
|
|
2005
|
13 |
6 |
p. 2157-2165
9 p.
|
artikel
|
| 14 |
Design, synthesis, antibacterial and QSAR studies of benzimidazole and imidazole chloroaryloxyalkyl derivatives
|
Khalafi-Nezhad, A.
|
|
2005
|
13 |
6 |
p. 1931-1938
8 p.
|
artikel
|
| 15 |
Development of α-keto-based inhibitors of cruzain, a cysteine protease implicated in Chagas disease
|
Choe, Youngchool
|
|
2005
|
13 |
6 |
p. 2141-2156
16 p.
|
artikel
|
| 16 |
2,7-Dihydro-3H-pyridazino[5,4,3-kl]acridin-3-one derivatives, novel type of cytotoxic agents active on multidrug-resistant cell lines. Synthesis and biological evaluation
|
Stefańska, Barbara
|
|
2005
|
13 |
6 |
p. 1969-1975
7 p.
|
artikel
|
| 17 |
Dipeptide alcohol-based inhibitors of eukaryotic DNA polymerase α
|
Kuriyama, Isoko
|
|
2005
|
13 |
6 |
p. 2187-2196
10 p.
|
artikel
|
| 18 |
Editorial board
|
|
|
2005
|
13 |
6 |
p. IFC-
1 p.
|
artikel
|
| 19 |
Fluorosubstitution and 7-alkylation as prospective modifications of biologically active 6-aryl derivatives of tricyclic acyclovir and ganciclovir analogues
|
Ostrowski, Tomasz
|
|
2005
|
13 |
6 |
p. 2089-2096
8 p.
|
artikel
|
| 20 |
General synthesis and biological evaluation of α-1-C-substituted derivatives of fagomine (2-deoxynojirimycin-α-C-glycosides)
|
Goujon, Jean-Yves
|
|
2005
|
13 |
6 |
p. 2313-2324
12 p.
|
artikel
|
| 21 |
Graphical contents list
|
|
|
2005
|
13 |
6 |
p. 1881-1891
11 p.
|
artikel
|
| 22 |
Heterocyclic inhibitors of dihydrodipicolinate synthase are not competitive
|
Turner, Jennifer J.
|
|
2005
|
13 |
6 |
p. 2133-2140
8 p.
|
artikel
|
| 23 |
1H NMR studies of homo and mixed ligand complexes of Tl+ ion with several polyazamacrocycles
|
Bordbar, Maryam
|
|
2005
|
13 |
6 |
p. 2253-2262
10 p.
|
artikel
|
| 24 |
Inhibition of secretory phospholipase A2. 2-Synthesis and structure–activity relationship studies of 4,5-dihydro-3-(4-tetradecyloxybenzyl)-1,2,4-4H-oxadiazol-5-one (PMS1062) derivatives specific for group II enzyme
|
Dong, Chang-Zhi
|
|
2005
|
13 |
6 |
p. 1989-2007
19 p.
|
artikel
|
| 25 |
Inhibitory effects of 2-substituted-1-naphthol derivatives on cyclooxygenase I and II
|
Kongkathip, Boonsong
|
|
2005
|
13 |
6 |
p. 2167-2175
9 p.
|
artikel
|
| 26 |
Instructions to contributors
|
|
|
2005
|
13 |
6 |
p. III-VII
nvt p.
|
artikel
|
| 27 |
Microbial transformation of (−)-isolongifolol and butyrylcholinesterase inhibitory activity of transformed products
|
Choudhary, M. Iqbal
|
|
2005
|
13 |
6 |
p. 1939-1944
6 p.
|
artikel
|
| 28 |
Molecular docking and 3D-QSAR studies on the binding mechanism of statine-based peptidomimetics with β-secretase
|
Zuo, Zhili
|
|
2005
|
13 |
6 |
p. 2121-2131
11 p.
|
artikel
|
| 29 |
New naphthylcombretastatins. Modifications on the ethylene bridge
|
Sánchez Maya, Ana B.
|
|
2005
|
13 |
6 |
p. 2097-2107
11 p.
|
artikel
|
| 30 |
Novel acetylcholinesterase inhibitor as increasing agent on rhythmic bladder contractions: SAR of 8-{3-[1-(3-fluorobenzyl)piperidin-4-yl]propanoyl}-1,2,5,6-tetrahydro-4H-pyrrolo[3,2,1-ij]quinolin-4-one (TAK-802) and related compounds
|
Ishichi, Yuji
|
|
2005
|
13 |
6 |
p. 1901-1911
11 p.
|
artikel
|
| 31 |
Oxathiolene oxide synthesis via chelation-controlled addition of organometallic reagents to alkynols followed by addition of sulfur electrophiles and evaluation of oxathiolene oxides as anticarcinogenic enzyme inducers
|
Franks, Marion A.
|
|
2005
|
13 |
6 |
p. 2221-2233
13 p.
|
artikel
|
| 32 |
Parallel synthesis and dopamine D3/D2 receptor screening of novel {4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl}carboxamides
|
Heidler, Philipp
|
|
2005
|
13 |
6 |
p. 2009-2014
6 p.
|
artikel
|
| 33 |
Properties and structure–activity studies of cyclic β-hairpin peptidomimetics based on the cationic antimicrobial peptide protegrin I
|
Robinson, John A.
|
|
2005
|
13 |
6 |
p. 2055-2064
10 p.
|
artikel
|
| 34 |
Structure–activity relationship for aryl and heteroaryl boronic acid inhibitors of hormone-sensitive lipase
|
Ebdrup, Søren
|
|
2005
|
13 |
6 |
p. 2305-2312
8 p.
|
artikel
|
| 35 |
Structure–activity study of epi-gallocatechin gallate (EGCG) analogs as proteasome inhibitors
|
Wan, Sheng Biao
|
|
2005
|
13 |
6 |
p. 2177-2185
9 p.
|
artikel
|
| 36 |
Synthesis and antiamoebic activities of 1-N-substituted cyclised pyrazoline analogues of thiosemicarbazones
|
Abid, Mohammad
|
|
2005
|
13 |
6 |
p. 2213-2220
8 p.
|
artikel
|
| 37 |
Synthesis and anticancer activity of new pyrrolocarbazoles and pyrrolo-β-carbolines
|
Laronze, M.
|
|
2005
|
13 |
6 |
p. 2263-2283
21 p.
|
artikel
|
| 38 |
Synthesis and biological activity of fluoroquinolone-pyrrolo[2,1-c][1,4]benzodiazepine conjugates
|
Kamal, Ahmed
|
|
2005
|
13 |
6 |
p. 2021-2029
9 p.
|
artikel
|
| 39 |
Synthesis and biological evaluation of 2-aminothiazoles and their amide derivatives on human adenosine receptors. Lack of effect of 2-aminothiazoles as allosteric enhancers
|
Göblyös, Anikó
|
|
2005
|
13 |
6 |
p. 2079-2087
9 p.
|
artikel
|
| 40 |
Synthesis and biological evaluation of new symmetrical derivatives as cytotoxic agents and apoptosis inducers
|
Sanmartín, Carmen
|
|
2005
|
13 |
6 |
p. 2031-2044
14 p.
|
artikel
|
| 41 |
Synthesis, conformational analysis, and biological activity of new analogues of thiazole-4-carboxamide adenine dinucleotide (TAD) as IMP dehydrogenase inhibitors
|
Franchetti, Palmarisa
|
|
2005
|
13 |
6 |
p. 2045-2053
9 p.
|
artikel
|
| 42 |
Synthesis of brequinar analogue inhibitors of malaria parasite dihydroorotate dehydrogenase
|
Boa, Andrew N.
|
|
2005
|
13 |
6 |
p. 1945-1967
23 p.
|
artikel
|
| 43 |
2,4,6-Trisubstituted pyrimidine derivatives as pregnancy interceptive agents
|
Agarwal, Anu
|
|
2005
|
13 |
6 |
p. 1893-1899
7 p.
|
artikel
|
| 44 |
UV-B protective effect of a polyacylated anthocyanin, HBA, in flower petals of the blue morning glory, Ipomoea tricolor cv. Heavenly Blue
|
Mori, Mihoko
|
|
2005
|
13 |
6 |
p. 2015-2020
6 p.
|
artikel
|
Tijdschrift beschrijving