| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
A comprehensive description of cyclin-dependent kinase 8 (CDK8) inhibitors as anticancer agents
|
Liu, Ying
|
|
|
128 |
C |
p.
|
artikel
|
| 2 |
Advances in MLKL-targeted inhibitors and PROTACs for necroptosis therapeutics
|
Dai, Pengcheng
|
|
|
128 |
C |
p.
|
artikel
|
| 3 |
An N-linked imidazo[1,2-a]pyridine benzoheterobicyclic hybrid inhibits mitosis and cancer cell proliferation by targeting tubulin
|
Sarkar, Tuhin
|
|
|
128 |
C |
p.
|
artikel
|
| 4 |
Brief analysis of Nav1.7 inhibitors: Mechanism of action and new research trends
|
Dong, Zhoujun
|
|
|
128 |
C |
p.
|
artikel
|
| 5 |
Comparative druggability of PD-1/PD-L1 inhibitors (A56, HD10): Cross-species differences in PD-L1 exposure and efficacy
|
Awadasseid, Annoor
|
|
|
128 |
C |
p.
|
artikel
|
| 6 |
Comprehensive insights into emodin compounds research in medicinal chemistry
|
Zhu, Liu-Xue
|
|
|
128 |
C |
p.
|
artikel
|
| 7 |
Contents continued
|
|
|
|
128 |
C |
p.
|
artikel
|
| 8 |
Design and synthesis of Sorafenib analogues and evaluation of their ferroptosis-inducing effects in tumor cells
|
Ning, Changxu
|
|
|
128 |
C |
p.
|
artikel
|
| 9 |
Design, synthesis, and anticancer evaluation of new pyrazolo[3,4-d]pyrimidine-based derivatives: CDK2 inhibition, apoptosis-inducing activity, molecular modelling studies
|
Hassan, Rasha A.
|
|
|
128 |
C |
p.
|
artikel
|
| 10 |
Design, synthesis, and biological evaluation of long-acting glucagon-like peptide-1 (GLP-1) conjugates modified with dual fatty acids and a proline-alanine-serine (PAS) polypeptide
|
Wang, Chengcheng
|
|
|
128 |
C |
p.
|
artikel
|
| 11 |
Design, synthesis, and biological evaluation of thioamide-linked spiropyrrolidine derivatives as novel 3CLpro inhibitors against SARS-CoV-2
|
Guma, Samuel Desta
|
|
|
128 |
C |
p.
|
artikel
|
| 12 |
Design, synthesis and structure-activity relationship studies of novel macrocyclic 2,4-diaminopyrimidines as HPK1 inhibitors
|
Wu, Feifei
|
|
|
128 |
C |
p.
|
artikel
|
| 13 |
Development of phenolic Mannich bases as α-glucosidase and aldose reductase inhibitors: In vitro and in silico approaches for managing diabetes mellitus and its complications
|
Tokalı, Feyzi Sinan
|
|
|
128 |
C |
p.
|
artikel
|
| 14 |
Drug discovery targeting protein arginine methyltransferase 5 (PRMT5): an update
|
Gu, Zhouyang
|
|
|
128 |
C |
p.
|
artikel
|
| 15 |
Editorial Board
|
|
|
|
128 |
C |
p.
|
artikel
|
| 16 |
Enhancing cyclic peptide functionality with hydrophilic diamino acids for improved APC-Asef interaction inhibition
|
He, Shipeng
|
|
|
128 |
C |
p.
|
artikel
|
| 17 |
Exploration of 4′-fluoro fleximer nucleoside analogues as potential broad-spectrum antiviral agents
|
Davis, Kyle A.
|
|
|
128 |
C |
p.
|
artikel
|
| 18 |
Graphical abstract TOC
|
|
|
|
128 |
C |
p.
|
artikel
|
| 19 |
Graphical abstract TOC
|
|
|
|
128 |
C |
p.
|
artikel
|
| 20 |
Innovative synthesis and purification method of fluorescent and bifunctional substrates for self-labelling protein tags
|
Sategna, Anna
|
|
|
128 |
C |
p.
|
artikel
|
| 21 |
Optimization of a naphthyl amide class identifies potent and selective reversible monoacylglycerol lipase (MAGL) inhibitors
|
Song, Chao
|
|
|
128 |
C |
p.
|
artikel
|
| 22 |
10PL8 and 2fPL8 inhibit gastric cancer cell proliferation by targeting degradation of CDK6 proteins to arrest the cell cycle
|
Zhang, Hao
|
|
|
128 |
C |
p.
|
artikel
|
| 23 |
Preparation of mitochondria-targeted camptothecin derivatives for the imaging and antiproliferation of colorectal cancer
|
Xu, Chenmeng
|
|
|
128 |
C |
p.
|
artikel
|
| 24 |
Recent achievements in molecular insights, anticancer activities, and comparative structure activity relationships of thiazolidin-4-one derivatives as EGFR inhibitors (2019-present)
|
Elsisi, Wessam I.
|
|
|
128 |
C |
p.
|
artikel
|
| 25 |
Recent breakthroughs in synthetic small molecules targeting SARS-CoV-2 Mpro from 2022 to 2024
|
Braconi, Laura
|
|
|
128 |
C |
p.
|
artikel
|
| 26 |
Structural evolution progress of orally bioavailable selective estrogen receptor degraders
|
Zhang, Jiahe
|
|
|
128 |
C |
p.
|
artikel
|
| 27 |
Structural optimization of phthalazine derivatives for anti-HBV activities to improve oral bioavailability
|
Yang, Yurong
|
|
|
128 |
C |
p.
|
artikel
|
| 28 |
Structure-activity relationship and crystallographic analyses of non-secosteroidal vitamin D receptor ligands bearing diphenylsilane core as a hydrophobic pharmacophore
|
Mudiyanselage, Hansaka Nirupama Thilakarathne Narasinghe
|
|
|
128 |
C |
p.
|
artikel
|
| 29 |
Structure-activity relationships and mechanism studies of novel 1, 2, 4-triazole-Schiff base derivatives as urease inhibitors: Synthesis, enzyme kinetics, spectroscopy, thermodynamics, and molecular docking
|
Lei, Yuji
|
|
|
128 |
C |
p.
|
artikel
|
| 30 |
Structure-based design of a novel series of cholesterol 24-hydroxylase (CH24H) inhibitors bearing 1,3-oxazole as a heme–iron binding group
|
Ito, Yoshiteru
|
|
|
128 |
C |
p.
|
artikel
|
| 31 |
Synthesis and anticancer activity evaluation of new linked/fused bioisosteric pyrazole-thiazole-bearing hybrid molecules
|
Yushyn, Ihor
|
|
|
128 |
C |
p.
|
artikel
|
| 32 |
Synthesis and anticancer activity of betulin-succinate derivatives in vitro and in the zebrafish xenograft tumor model
|
Ouyang, Ting
|
|
|
128 |
C |
p.
|
artikel
|
| 33 |
Synthesis and biological evaluation of indoline derivatives as CDGSH iron sulfur domain 2 activators
|
Yao, Chun-Hsu
|
|
|
128 |
C |
p.
|
artikel
|
| 34 |
Synthesis and multitarget inhibitory effect of indole-based ethyl cinnamate derivatives against SARS-CoV-2 Mpro and cathepsins for broad-spectrum anti-coronavirus activity
|
Citarella, Andrea
|
|
|
128 |
C |
p.
|
artikel
|
| 35 |
Synthesis of 20α/β-hydroxyprogesterone-trimethyl lock-triglyceride-mimetic prodrugs and its bioavailability study in rats
|
Li, Liangyun
|
|
|
128 |
C |
p.
|
artikel
|
| 36 |
Synthesis of novel naphtho[1,8-de]pyrimidine fused iminosugars and their anti-tumor activities
|
Yang, Yupeng
|
|
|
128 |
C |
p.
|
artikel
|
| 37 |
Tag-like cyclic peptides: Modular affinity elements for protein integration and bioengineering applications
|
Zhu, Zirui
|
|
|
128 |
C |
p.
|
artikel
|
| 38 |
Targeting MAP kinase for inhibiting Leishmania promastigotes and amastigotes stages by L-alanine derived molecules and their anticancer potential against PANC-1 cancer cell lines
|
Shahid, Misbah
|
|
|
128 |
C |
p.
|
artikel
|
| 39 |
Trifluoromethyl-substituted 3-selenylindol and 3-thiophenylindol induce metabolic alterations and impairment of cell cycle progression in hepatocarcinoma cells (HepG2)
|
Sbrana Serur dos Santos, Eduardo
|
|
|
128 |
C |
p.
|
artikel
|
| 40 |
Unveiling the medicinal diversity of benzoic acid containing molecules: Insights on druggable targets for type 2 diabetes mellitus
|
Rani, Kajal
|
|
|
128 |
C |
p.
|
artikel
|
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