| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
Analysis of structure–activity relationships with the N-(3-acyloxy-2-benzylpropyl)-N ′-[4-(methylsulfonylamino)benzyl]thiourea template for vanilloid receptor 1 antagonism
|
Lee, Jeewoo
|
|
2004
|
12 |
13 |
p. 3411-3420
10 p.
|
artikel
|
| 2 |
A study of the stability of tri(glucosyloxyphenyl)chlorin, a sensitizer for photodynamic therapy, in human colon tumoural cells: a liquid chromatography and MALDI-TOF mass spectrometry analysis
|
Laville, I
|
|
2004
|
12 |
13 |
p. 3673-3682
10 p.
|
artikel
|
| 3 |
Benzamides and benzamidines as specific inhibitors of epidermal growth factor receptor and v-Src protein tyrosine kinases
|
Asano, Toru
|
|
2004
|
12 |
13 |
p. 3529-3542
14 p.
|
artikel
|
| 4 |
Contributors to this issue
|
|
|
2004
|
12 |
13 |
p. I-II
nvt p.
|
artikel
|
| 5 |
Corrigendum to “S1 subsite in snake venom thrombin-like enzymes: can S1 subsite lipophilicity be used to sort binding affinities of trypsin-like enzymes to small-molecule inhibitors?” [Bioorg. Med. Chem. 12 (2004) 2571]
|
Silva Jr., Floriano P.
|
|
2004
|
12 |
13 |
p. 3755-
1 p.
|
artikel
|
| 6 |
3-Deazaadenosine analogues of p5′A2′p5′A2′p5′A: synthesis, stereochemistry, and the roles of adenine ring nitrogen-3 in the interaction with RNase L
|
Kalinichenko, Elena N
|
|
2004
|
12 |
13 |
p. 3637-3647
11 p.
|
artikel
|
| 7 |
Design of 1-substituted 2-arylmethyl-4,5-methylenedioxybenzene derivatives as antiseizure agents
|
Micale, Nicola
|
|
2004
|
12 |
13 |
p. 3703-3709
7 p.
|
artikel
|
| 8 |
Design, synthesis, and structure–activity relationships of novel tetracyclic compounds as peripheral benzodiazepine receptor ligands
|
Okubo, Taketoshi
|
|
2004
|
12 |
13 |
p. 3569-3580
12 p.
|
artikel
|
| 9 |
Development of CoMFA, advance CoMFA and CoMSIA models in pyrroloquinazolines as thrombin receptor antagonist
|
Dixit, Anshuman
|
|
2004
|
12 |
13 |
p. 3591-3598
8 p.
|
artikel
|
| 10 |
Discovery and SAR of indole-2-carboxylic acid benzylidene-hydrazides as a new series of potent apoptosis inducers using a cell-based HTS assay
|
Zhang, Han-Zhong
|
|
2004
|
12 |
13 |
p. 3649-3655
7 p.
|
artikel
|
| 11 |
Editorial board
|
|
|
2004
|
12 |
13 |
p. IFC-
1 p.
|
artikel
|
| 12 |
Evaluation of hesperetin 7-O-lauryl ether as lipid-lowering agent in high-cholesterol-fed rats
|
Choi, Gab-Sun
|
|
2004
|
12 |
13 |
p. 3599-3605
7 p.
|
artikel
|
| 13 |
15-Fluoro prostaglandin FP agonists: a new class of topical ocular hypotensives
|
Klimko, Peter
|
|
2004
|
12 |
13 |
p. 3451-3469
19 p.
|
artikel
|
| 14 |
Graphical contents list
|
|
|
2004
|
12 |
13 |
p. 3401-3410
10 p.
|
artikel
|
| 15 |
GRIND/ALMOND investigations on CysLT1 receptor antagonists of the quinolinyl(bridged)aryl type
|
Benedetti, Paolo
|
|
2004
|
12 |
13 |
p. 3607-3617
11 p.
|
artikel
|
| 16 |
Inhibition of the Staphylococcus aureus sortase transpeptidase SrtA by phosphinic peptidomimetics
|
Kruger, Ryan G
|
|
2004
|
12 |
13 |
p. 3723-3729
7 p.
|
artikel
|
| 17 |
Instructions to contributors
|
|
|
2004
|
12 |
13 |
p. III-VII
nvt p.
|
artikel
|
| 18 |
Isolation of quercetin's salts and studies of their physicochemical properties and antioxidant relationships
|
Milane, Hadi A.
|
|
2004
|
12 |
13 |
p. 3627-3635
9 p.
|
artikel
|
| 19 |
Nitro and amino substitution within the A-ring of 5H-8,9-dimethoxy-5-(2-N,N-dimethylaminoethyl)dibenzo[c,h][1,6]naphthyridin-6-ones: influence on topoisomerase I-targeting activity and cytotoxicity
|
Ruchelman, Alexander L
|
|
2004
|
12 |
13 |
p. 3731-3742
12 p.
|
artikel
|
| 20 |
Novel iodine-124 labeled EGFR inhibitors as potential PET agents for molecular imaging in cancer
|
Shaul, Mazal
|
|
2004
|
12 |
13 |
p. 3421-3429
9 p.
|
artikel
|
| 21 |
Novel ketolide antibiotics with a fused five-membered lactone ring––synthesis, physicochemical and antimicrobial properties
|
Hunziker, Daniel
|
|
2004
|
12 |
13 |
p. 3503-3519
17 p.
|
artikel
|
| 22 |
Phenolic acid derivatives with potential anticancer properties––a structure–activity relationship study. Part 1: Methyl, propyl and octyl esters of caffeic and gallic acids
|
Fiuza, S.M.
|
|
2004
|
12 |
13 |
p. 3581-3589
9 p.
|
artikel
|
| 23 |
Probing the aglycon binding site of a β-glucosidase: a collection of C-1-modified 2,5-dideoxy-2,5-imino-d-mannitol derivatives and their structure–activity relationships as competitive inhibitors
|
Wrodnigg, Tanja M.
|
|
2004
|
12 |
13 |
p. 3485-3495
11 p.
|
artikel
|
| 24 |
Solution-phase combinatorial synthesis of nonpeptide bradykinin antagonists
|
Kam, Yoo Lim
|
|
2004
|
12 |
13 |
p. 3543-3552
10 p.
|
artikel
|
| 25 |
Study of the green tea polyphenols catechin-3-gallate (CG) and epicatechin-3-gallate (ECG) as proteasome inhibitors
|
Wan, Sheng Biao
|
|
2004
|
12 |
13 |
p. 3521-3527
7 p.
|
artikel
|
| 26 |
Synthesis and anticancer activity evaluation of new 2-alkylcarbonyl and 2-benzoyl-3-trifluoromethyl-quinoxaline 1,4-di-N-oxide derivatives
|
Zarranz, Belén
|
|
2004
|
12 |
13 |
p. 3711-3721
11 p.
|
artikel
|
| 27 |
Synthesis and antileishmanial activity of novel buparvaquone oxime derivatives
|
Mäntylä, Antti
|
|
2004
|
12 |
13 |
p. 3497-3502
6 p.
|
artikel
|
| 28 |
Synthesis and antitumor activity of 20-O-linked nitrogen-based camptothecin ester derivatives
|
Wang, Cun-ying
|
|
2004
|
12 |
13 |
p. 3657-3662
6 p.
|
artikel
|
| 29 |
Synthesis and cytotoxicity of 1-substituted 2-methyl-1H-imidazo[4,5-g]phthalazine-4,9-dione derivatives
|
Sung Kim, Jin
|
|
2004
|
12 |
13 |
p. 3683-3686
4 p.
|
artikel
|
| 30 |
Synthesis and evaluation of 6-methylene-bridged uracil derivatives. Part 1: Discovery of novel orally active inhibitors of human thymidine phosphorylase
|
Yano, Shingo
|
|
2004
|
12 |
13 |
p. 3431-3441
11 p.
|
artikel
|
| 31 |
Synthesis and evaluation of 6-methylene-bridged uracil derivatives. Part 2: Optimization of inhibitors of human thymidine phosphorylase and their selectivity with uridine phosphorylase
|
Yano, Shingo
|
|
2004
|
12 |
13 |
p. 3443-3450
8 p.
|
artikel
|
| 32 |
Synthesis and functional activity of (2-aryl-1-piperazinyl)-N-(3-methylphenyl)acetamides: selective dopamine D4 receptor agonists
|
Matulenko, Mark A
|
|
2004
|
12 |
13 |
p. 3471-3483
13 p.
|
artikel
|
| 33 |
Synthesis and fungicidal activity of enantiomerically pure (R)- and (S)-silicon-containing azole fungicides
|
Itoh, Hiroyuki
|
|
2004
|
12 |
13 |
p. 3561-3567
7 p.
|
artikel
|
| 34 |
Synthesis and immunochemical characterization of protein conjugates of carbohydrate and carbohydrate-mimetic peptides as experimental vaccines
|
Hossany, Rehana B
|
|
2004
|
12 |
13 |
p. 3743-3754
12 p.
|
artikel
|
| 35 |
Synthesis and neuropharmacological evaluation of R(−)-N-alkyl-11-hydroxynoraporphines and their esters
|
Csutoras, Csaba
|
|
2004
|
12 |
13 |
p. 3553-3559
7 p.
|
artikel
|
| 36 |
Synthesis and photocytotoxic activity of new α-methylene-γ-butyrolactone-psoralen heterodimers
|
Ropp, Sandrine
|
|
2004
|
12 |
13 |
p. 3619-3625
7 p.
|
artikel
|
| 37 |
Synthesis, antiviral, and anti-HIV-1 integrase activities of 3-aroyl-1,1-dioxo-1,4,2-benzodithiazines
|
Brzozowski, Zdzislaw
|
|
2004
|
12 |
13 |
p. 3663-3672
10 p.
|
artikel
|
| 38 |
Synthesis of carbamate-type caged derivatives of a novel glutamate transporter blocker
|
Takaoka, Kiyo
|
|
2004
|
12 |
13 |
p. 3687-3694
8 p.
|
artikel
|
| 39 |
Topological models for prediction of anti-inflammatory activity of N-arylanthranilic acids
|
Bajaj, Sanjay
|
|
2004
|
12 |
13 |
p. 3695-3701
7 p.
|
artikel
|
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