| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
A biaryl peptide crosslink in a MetJ peptide model confers cooperative, nonspecific binding to DNA that ablates both repressor binding and In vitro transcription
|
Yoburn, Joshua C
|
|
2003
|
11 |
6 |
p. 811-816
6 p.
|
artikel
|
| 2 |
A frame shifted disulfide bridged analogue of angiotensin II
|
Schmidt, Boris
|
|
2003
|
11 |
6 |
p. 985-990
6 p.
|
artikel
|
| 3 |
Antitumor agents 220. Antitumor-Promoting effects of cimigenol and related compounds on Epstein–Barr virus activation and two-stage mouse skin carcinogenesis
|
Sakurai, Nobuko
|
|
2003
|
11 |
6 |
p. 1137-1140
4 p.
|
artikel
|
| 4 |
A substrate variant as a high-affinity, reversible inhibitor: insight from the X-ray structure of cilastatin bound to membrane dipeptidase
|
Smyth, Timothy P
|
|
2003
|
11 |
6 |
p. 991-998
8 p.
|
artikel
|
| 5 |
Bis-4-aminoquinolines: novel triple-helix DNA intercalators and antagonists of immunostimulatory CpG-oligodeoxynucleotides
|
Strekowski, Lucjan
|
|
2003
|
11 |
6 |
p. 1079-1085
7 p.
|
artikel
|
| 6 |
Chiral 3,3′-(1,2-Ethanediyl)-bis[2-(3,4-dimethoxyphenyl)-4-thiazolidinones] with anti-inflammatory activity. Part 11: Evaluation of COX-2 selectivity and modelling
|
Vigorita, M.G
|
|
2003
|
11 |
6 |
p. 999-1006
8 p.
|
artikel
|
| 7 |
Curcumin differentially modulates mRNA profiles in Jurkat T and human peripheral blood mononuclear cells
|
Gertsch, Jürg
|
|
2003
|
11 |
6 |
p. 1057-1063
7 p.
|
artikel
|
| 8 |
Design and synthesis of HIV-1 protease inhibitors. Novel tetrahydrofuran P2/P2′-groups interacting with Asp29/30 of the HIV-1 protease. Determination of binding from X-ray crystal structure of inhibitor protease complex
|
Oscarsson, Karin
|
|
2003
|
11 |
6 |
p. 1107-1115
9 p.
|
artikel
|
| 9 |
6-Dimethylamino 1H-Pyrazolo[3,4-d]pyrimidine derivatives as new inhibitors of inflammatory mediators in intact cells
|
Quintela, José M
|
|
2003
|
11 |
6 |
p. 863-868
6 p.
|
artikel
|
| 10 |
2,3-Disubstituted quinuclidines as a novel class of dopamine transporter inhibitors
|
Sakamuri, Sukumar
|
|
2003
|
11 |
6 |
p. 1123-1136
14 p.
|
artikel
|
| 11 |
Editorial Board
|
|
|
2003
|
11 |
6 |
p. IFC-
1 p.
|
artikel
|
| 12 |
Graphical Abstracts
|
|
|
2003
|
11 |
6 |
p. 801-809
9 p.
|
artikel
|
| 13 |
Ibogaine analogues. Synthesis and preliminary pharmacological evaluation of 7-heteroaryl-2-azabicyclo[2.2.2]oct-7-enes
|
Passarella, Daniele
|
|
2003
|
11 |
6 |
p. 1007-1014
8 p.
|
artikel
|
| 14 |
Inhibition of nucleoside transport By new analogues of nitrobenzylthioinosine
|
Deghati, Paymaneh Y.F
|
|
2003
|
11 |
6 |
p. 899-908
10 p.
|
artikel
|
| 15 |
Mechanism of biochemical action of substituted 4-methylbenzopyran-2-ones. Part 10: identification of inhibitors for the liver microsomal acetoxycoumarin: protein transacetylase
|
Raj, Hanumantharao G
|
|
2003
|
11 |
6 |
p. 1015-1019
5 p.
|
artikel
|
| 16 |
Modes of antifungal action of alkanols against Saccharomyces cerevisiae
|
Kubo, Isao
|
|
2003
|
11 |
6 |
p. 1117-1122
6 p.
|
artikel
|
| 17 |
New fluorinated derivatives as esterase inhibitors. Synthesis, hydration and crossed specificity studies
|
Quero, Carmen
|
|
2003
|
11 |
6 |
p. 1047-1055
9 p.
|
artikel
|
| 18 |
New insights into protein crosslinking via the Maillard reaction: structural requirements, the effect on enzyme function, and predicted efficacy of crosslinking inhibitors as anti-ageing therapeutics
|
Miller, Antonia G
|
|
2003
|
11 |
6 |
p. 843-852
10 p.
|
artikel
|
| 19 |
N-Morpholino- and N-diethyl-analogues of palmitoylethanolamide increase the sensitivity of transfected human vanilloid receptors to activation by anandamide without affecting fatty acid amidohydrolase activity
|
Vandevoorde, Séverine
|
|
2003
|
11 |
6 |
p. 817-825
9 p.
|
artikel
|
| 20 |
ortho-Halogen naphthaleins as specific inhibitors of Lactobacillus casei thymidylate synthase. Conformational properties and biological activity
|
Ghelli, Stefano
|
|
2003
|
11 |
6 |
p. 951-963
13 p.
|
artikel
|
| 21 |
Prodrugs of biologically active phosphate esters
|
Schultz, Carsten
|
|
2003
|
11 |
6 |
p. 885-898
14 p.
|
artikel
|
| 22 |
Purification and characterization of an alkaline lipase from a newly isolated Pseudomonas mendocina PK-12CS and chemoselective hydrolysis of fatty acid ester † † CDRI Communication No. 6212.
|
Jinwal, Umesh K
|
|
2003
|
11 |
6 |
p. 1041-1046
6 p.
|
artikel
|
| 23 |
Role of solution conformation and flexibility of short peptide ligands that bind to the p56lck SH2 domain
|
Dekker, Frank J
|
|
2003
|
11 |
6 |
p. 941-949
9 p.
|
artikel
|
| 24 |
Solid-phase library synthesis of reversed-statine type inhibitors of the malarial aspartyl proteases plasmepsin I and II
|
Dahlgren, Anders
|
|
2003
|
11 |
6 |
p. 827-841
15 p.
|
artikel
|
| 25 |
Structure–activity relationships of xanthene carboxamides, novel CCR1 receptor antagonists
|
Naya, Akira
|
|
2003
|
11 |
6 |
p. 875-884
10 p.
|
artikel
|
| 26 |
Substituted heterocyclic thiourea compounds as a new class of anti-allergic agents inhibiting IgE/FcεRI receptor mediated mast cell leukotriene release
|
Venkatachalam, T.K
|
|
2003
|
11 |
6 |
p. 1095-1105
11 p.
|
artikel
|
| 27 |
Synthesis and antioxidant properties of a new lipophilic ascorbic acid analogue
|
Cotelle, Philippe
|
|
2003
|
11 |
6 |
p. 1087-1093
7 p.
|
artikel
|
| 28 |
Synthesis and anti-tumor-promoting activity of glycoglycerolipid analogues lacking the glycerol backbone
|
Colombo, Diego
|
|
2003
|
11 |
6 |
p. 909-912
4 p.
|
artikel
|
| 29 |
Synthesis and bioactivity of 4,10-dimethyl-pyridino[2,3-h]quinolin-2(1H)-one-9-carboxylic acid and its esters
|
Zhang, Qian
|
|
2003
|
11 |
6 |
p. 1031-1034
4 p.
|
artikel
|
| 30 |
Synthesis and biological activity of 3,3-Diamino-sulfonylacrylonitriles as novel inhibitors of glucose induced insulin secretion from beta cells
|
Tagmose, Tina M
|
|
2003
|
11 |
6 |
p. 931-940
10 p.
|
artikel
|
| 31 |
Synthesis and cytotoxicity of dihydroartemisinin ethers containing cyanoarylmethyl group
|
Li, Ying
|
|
2003
|
11 |
6 |
p. 977-984
8 p.
|
artikel
|
| 32 |
Synthesis and DNA binding studies of a new asymmetric cyanine dye binding in the minor groove of [poly(dA-dT)]2
|
Karlsson, H.Jonas
|
|
2003
|
11 |
6 |
p. 1035-1040
6 p.
|
artikel
|
| 33 |
Synthesis and evaluation of trans 3,4-cyclopropyl l-arginine analogues as isoform selective inhibitors of nitric oxide synthase
|
Fishlock, Dan
|
|
2003
|
11 |
6 |
p. 869-873
5 p.
|
artikel
|
| 34 |
Synthesis and growth inhibition activity of α-Bromoacrylic heterocyclic and benzoheterocyclic derivatives of distamycin A modified on the amidino moiety
|
Baraldi, Pier Giovanni
|
|
2003
|
11 |
6 |
p. 965-975
11 p.
|
artikel
|
| 35 |
Synthesis and structure–affinity relationship investigations of 5-aminomethyl and 5-carbamoyl analogues of the antipsychotic sertindole. A new class of selective α1 adrenoceptor antagonists
|
Balle, Thomas
|
|
2003
|
11 |
6 |
p. 1065-1078
14 p.
|
artikel
|
| 36 |
Synthesis, characterization and in vitro anti-invasive activity screening of polyphenolic and heterocyclic compounds
|
Parmar, Virinder S
|
|
2003
|
11 |
6 |
p. 913-929
17 p.
|
artikel
|
| 37 |
The role of dicarbonyl compounds in non-enzymatic crosslinking: a structure–activity study
|
Meade, Susie J
|
|
2003
|
11 |
6 |
p. 853-862
10 p.
|
artikel
|
| 38 |
Water soluble prodrugs of the antitumor agent 3-[(3-amino-4-methoxy)phenyl]-2-(3,4,5-trimethoxyphenyl)cyclopent-2-ene-1-one
|
Nam, Nguyen-Hai
|
|
2003
|
11 |
6 |
p. 1021-1029
9 p.
|
artikel
|
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