| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
Analysis of stereoelectronic properties, mechanism of action and pharmacophore of synthetic indolo[2,1-b]quinazoline-6,12-dione derivatives in relation to antileishmanial activity using quantum chemical, cyclic voltammetry and 3-D-QSAR CATALYST procedures
|
Bhattacharjee, Apurba K
|
|
2002
|
10 |
6 |
p. 1979-1989
11 p.
|
artikel
|
| 2 |
Anti-Candida albicans Properties of Novel Benzoxazine Analogues
|
Fringuelli, Renata
|
|
2002
|
10 |
6 |
p. 1681-1686
6 p.
|
artikel
|
| 3 |
A Practical Synthesis and Biological Evaluation of 9-Halogenated PGF Analogues
|
Tani, Kousuke
|
|
2002
|
10 |
6 |
p. 1883-1894
12 p.
|
artikel
|
| 4 |
Arbutin synthase, a novel member of the NRD1β glycosyltransferase family, is a unique multifunctional enzyme converting various natural products and xenobiotics
|
Hefner, Tobias
|
|
2002
|
10 |
6 |
p. 1731-1741
11 p.
|
artikel
|
| 5 |
Chemical Modification of the β-Glucocerebrosidase Inhibitor N-Octyl-β-valienamine: Synthesis and Biological Evaluation of 4-Epimeric and 4-O-(β-d-Galactopyranosyl) Derivatives
|
Ogawa, Seiichiro
|
|
2002
|
10 |
6 |
p. 1967-1972
6 p.
|
artikel
|
| 6 |
Comparison of the Inhibition of Human and Trypanosoma cruzi Prolyl Endopeptidases
|
Vendeville, Sandrine
|
|
2002
|
10 |
6 |
p. 1719-1729
11 p.
|
artikel
|
| 7 |
Design and synthesis of a selective EP4-receptor agonist. Part 3: 16-phenyl-5-thiaPGE1 and 9-β-halo derivatives with improved stability
|
Maruyama, Toru
|
|
2002
|
10 |
6 |
p. 1743-1759
17 p.
|
artikel
|
| 8 |
Design and Synthesis of Novel Tetra-Peptide Motilin Agonists
|
Haramura, Masayuki
|
|
2002
|
10 |
6 |
p. 1805-1811
7 p.
|
artikel
|
| 9 |
Determination of a sugar chain and its linkage site on a glycoprotein TIME-EA4 from silkworm diapause eggs by means of LC-ESI-Q-TOF-MS and MS/MS
|
Kurahashi, Takuya
|
|
2002
|
10 |
6 |
p. 1703-1710
8 p.
|
artikel
|
| 10 |
Discovery of 4,5-Diphenyl-1,2,4-triazole Derivatives as a Novel Class of Selective Antagonists for the Human V1A Receptor
|
Kakefuda, Akio
|
|
2002
|
10 |
6 |
p. 1905-1912
8 p.
|
artikel
|
| 11 |
Efficient and highly stereoselective synthesis of a β-Lactam inhibitor of the serine protease prostate-specific antigen
|
Annunziata, Rita
|
|
2002
|
10 |
6 |
p. 1813-1818
6 p.
|
artikel
|
| 12 |
Efficient Synthesis of ‘Redox-Switched’ Naphthoquinone Thiol-Crown Ethers and Their Biological Activity Evaluation
|
Huang, Sheng-Tung
|
|
2002
|
10 |
6 |
p. 1947-1952
6 p.
|
artikel
|
| 13 |
Erratum to “sequence-specific delivery of a quinone methide intermediate to the major groove of DNA” [Bioorg. Med. Chem. 9 (2001) 2347]
|
Zhou, Qibing
|
|
2002
|
10 |
6 |
p. 2089-
1 p.
|
artikel
|
| 14 |
Exploration of the DTrp-NMeLys Motif in the Search for potent somatostatin antagonists
|
Rajeswaran, W.G
|
|
2002
|
10 |
6 |
p. 2023-2029
7 p.
|
artikel
|
| 15 |
Graphical Abstracts
|
|
|
2002
|
10 |
6 |
p. xi-xxi
nvt p.
|
artikel
|
| 16 |
Higher acyclic nitrogen containing deoxy sugar derivatives: A new lead in the generation of antimycobacterial chemotherapeutics
|
Pathak, Rashmi
|
|
2002
|
10 |
6 |
p. 1695-1702
8 p.
|
artikel
|
| 17 |
Insight into the stereochemistry in the inhibition of carboxypeptidase A with N-(hydroxyaminocarbonyl)phenylalanine: binding modes of an enantiomeric pair of the inhibitor to carboxypeptidase A
|
Cho, Jae Hyun
|
|
2002
|
10 |
6 |
p. 2015-2022
8 p.
|
artikel
|
| 18 |
linckosides A and B, two new neuritogenic steroid glycosides from the okinawan starfish linckia laevigata
|
Qi, Jianhua
|
|
2002
|
10 |
6 |
p. 1961-1966
6 p.
|
artikel
|
| 19 |
Major histocompatibility complex class II binding characteristics of peptoid–peptide hybrids
|
de Haan, Ellen C
|
|
2002
|
10 |
6 |
p. 1939-1945
7 p.
|
artikel
|
| 20 |
Metabolites of Orally Active NO-Independent Pyrazolopyridine Stimulators of Soluble Guanylate Cyclase
|
Straub, Alexander
|
|
2002
|
10 |
6 |
p. 1711-1717
7 p.
|
artikel
|
| 21 |
Molecular recognition by Kluyveromyces of amphotericin B-loaded, galactose-tagged, poly (lactic acid) microspheres
|
Kassab, Rima
|
|
2002
|
10 |
6 |
p. 1767-1775
9 p.
|
artikel
|
| 22 |
N-3(9)-Arylpropenyl-N-9(3)-propionyl-3,9-diazabicyclo[3.3.1]nonanes as μ-Opioid receptor agonists. Effects on μ-Affinity of arylalkenyl chain modifications
|
Pinna, Gérard A.
|
|
2002
|
10 |
6 |
p. 1929-1937
9 p.
|
artikel
|
| 23 |
New apratoxins of marine cyanobacterial origin from guam and palau
|
Luesch, Hendrik
|
|
2002
|
10 |
6 |
p. 1973-1978
6 p.
|
artikel
|
| 24 |
New synthetic siderophores and Their β-Lactam conjugates based on diamino acids and dipeptides
|
Wittmann, S
|
|
2002
|
10 |
6 |
p. 1659-1670
12 p.
|
artikel
|
| 25 |
Novel 4,5-Diaryl-3-hydroxy-2(5H)-furanones as Anti-Oxidants and Anti-Inflammatory Agents
|
Weber, Valérie
|
|
2002
|
10 |
6 |
p. 1647-1658
12 p.
|
artikel
|
| 26 |
Novel Morpholinone-Based d-Phe-Pro-Arg Mimics as Potential Thrombin Inhibitors: Design, Synthesis, and X-ray Crystal Structure of an Enzyme Inhibitor Complex
|
Dahlgren, Anders
|
|
2002
|
10 |
6 |
p. 1829-1839
11 p.
|
artikel
|
| 27 |
Novel tacrine derivatives that block neuronal calcium channels
|
de los Rı́os, Cristóbal
|
|
2002
|
10 |
6 |
p. 2077-2088
12 p.
|
artikel
|
| 28 |
Oligomers of glycamino acid
|
Suhara, Yoshitomo
|
|
2002
|
10 |
6 |
p. 1999-2013
15 p.
|
artikel
|
| 29 |
2-O-Substituted Cyclodextrins as Reversal Agents for the Neuromuscular Blocker Rocuronium Bromide
|
Tarver, Gary J
|
|
2002
|
10 |
6 |
p. 1819-1827
9 p.
|
artikel
|
| 30 |
3-Oxa-15-cyclohexyl prostaglandin DP receptor agonists as topical antiglaucoma agents
|
Hellberg, Mark R.
|
|
2002
|
10 |
6 |
p. 2031-2049
19 p.
|
artikel
|
| 31 |
Phenylpiperazinylmethylindolecarboxylates and derivatives as selective D4-Ligands
|
Moll, Annette
|
|
2002
|
10 |
6 |
p. 1671-1679
9 p.
|
artikel
|
| 32 |
Photo-Control of nitric oxide synthase activity using a caged isoform specific inhibitor
|
Montgomery, Heather J.
|
|
2002
|
10 |
6 |
p. 1919-1927
9 p.
|
artikel
|
| 33 |
Potent DNA photocleavage by zinc(II) complexes of cationic bis-porphyrins linked with aliphatic diamine
|
Ishikawa, Yoshinobu
|
|
2002
|
10 |
6 |
p. 1953-1960
8 p.
|
artikel
|
| 34 |
Structure–Activity Relationships of seco-Prezizaane Terpenoids in γ-Aminobutyric Acid Receptors of Houseflies and Rats
|
Kuriyama, Tadahiko
|
|
2002
|
10 |
6 |
p. 1873-1881
9 p.
|
artikel
|
| 35 |
Study on quantitative structure–toxicity relationships of benzene derivatives acting by narcosis
|
Khadikar, Padmakar V.
|
|
2002
|
10 |
6 |
p. 1761-1766
6 p.
|
artikel
|
| 36 |
Syntheses, biological evaluation and QSAR study on antitumor activity of 1,5-N,N′-disubstituted-2-(substituted benzenesulphonyl) glutamamides
|
Srikanth, K.
|
|
2002
|
10 |
6 |
p. 1841-1854
14 p.
|
artikel
|
| 37 |
Synthesis and antimicrotubule activity of combretatropone derivatives
|
Janik, Mark E.
|
|
2002
|
10 |
6 |
p. 1895-1903
9 p.
|
artikel
|
| 38 |
Synthesis and biological evaluation of aroylguanidines related to amiloride as inhibitors of the human platelet Na+/H+ exchanger
|
Laeckmann, Didier
|
|
2002
|
10 |
6 |
p. 1793-1804
12 p.
|
artikel
|
| 39 |
Synthesis and In Vitro Antitumor Activity of Thiophene Analogues of 5-Chloro-5,8-dideazafolic Acid and 2-Methyl-2-desamino-5-chloro-5,8-dideazafolic Acid
|
Forsch, Ronald A.
|
|
2002
|
10 |
6 |
p. 2067-2076
10 p.
|
artikel
|
| 40 |
Synthesis and In vitro characterization of a tissue-Selective fullerene: vectoring C60(OH)16AMBP to mineralized bone
|
Gonzalez, Kelly A
|
|
2002
|
10 |
6 |
p. 1991-1997
7 p.
|
artikel
|
| 41 |
Synthesis and SAR of N-Benzoyl-l-Biphenylalanine Derivatives: Discovery of TR-14035, A Dual α4β7/α4β1 Integrin Antagonist
|
Sircar, Ila
|
|
2002
|
10 |
6 |
p. 2051-2066
16 p.
|
artikel
|
| 42 |
Synthesis and structure–activity relationship of diarylamide urea derivatives as selective inhibitors of the proliferation of human coronary artery smooth muscle cells
|
Ogita, Haruhisa
|
|
2002
|
10 |
6 |
p. 1865-1871
7 p.
|
artikel
|
| 43 |
Synthesis of a novel quinoline derivative, 2-(2-methylquinolin-4-ylamino)-N-phenylacetamide—a potential antileishmanial agent
|
Sahu, Niranjan P.
|
|
2002
|
10 |
6 |
p. 1687-1693
7 p.
|
artikel
|
| 44 |
Synthesis of Feruloyl-myo-insitol derivatives and their inhibitory effects on phorbol ester-induced superoxide generation and esptein–barr virus activation
|
Hosoda, Asao
|
|
2002
|
10 |
6 |
p. 1855-1863
9 p.
|
artikel
|
| 45 |
Synthesis of (1S,2R)-1-Phenyl-2-[(S)-1-aminopropyl]-N,N-diethylcyclopropanecarboxamide (PPDC) Derivatives Modified at the Carbamoyl Moiety As a New Class of NMDA Receptor Antagonists
|
Kazuta, Yuji
|
|
2002
|
10 |
6 |
p. 1777-1791
15 p.
|
artikel
|
| 46 |
Vomilenine Reductase — a novel Enzyme catalyzing a crucial Step in the Biosynthesis of the Therapeutically applied Antiarrhythmic Alkaloid Ajmaline
|
von Schumann, Gerald
|
|
2002
|
10 |
6 |
p. 1913-1918
6 p.
|
artikel
|
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