nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
1 |
Absolute Stereostructure of Potent α-Glucosidase Inhibitor, Salacinol, with Unique Thiosugar Sulfonium Sulfate Inner Salt Structure from Salacia reticulata
|
Yoshikawa, Masayuki |
|
2002 |
10 |
5 |
p. 1547-1554 8 p. |
artikel |
2 |
Acetamidoquinone and acetamidohydroxy derivatives as inhibitors for both dihydroxyacetamido epoxidase and dehydrogenase
|
Whiteley, Chris G. |
|
2002 |
10 |
5 |
p. 1221-1227 7 p. |
artikel |
3 |
A Convenient Synthesis and Hepatoprotective Activity of Imidazo[1,2-c]pyrimido[5,4-e]pyrimidine, Tetraazaacenaphthene and Tetraazaphenalene from Cyclic Ketene Aminals Through Tandem Addition-Cyclization Reactions ‡ ‡ CDRI communication number 5986.
|
Ram, Vishnu J |
|
2002 |
10 |
5 |
p. 1275-1280 6 p. |
artikel |
4 |
5′-Alkyl-benzothiadiazides: A New Subgroup of AMPA Receptor Modulators with Improved Affinity
|
Phillips, Dean |
|
2002 |
10 |
5 |
p. 1229-1248 20 p. |
artikel |
5 |
An Analysis of the Binding of Cocaine Analogues to the Monoamine Transporters Using Tensor Decomposition 3-D QSAR
|
Appell, Michael |
|
2002 |
10 |
5 |
p. 1197-1206 10 p. |
artikel |
6 |
A Novel Approach towards Studying Non-Genotoxic Enediynes as Potential Anticancer Therapeutics
|
Hakimelahi, Gholam Hossein |
|
2002 |
10 |
5 |
p. 1321-1328 8 p. |
artikel |
7 |
Antioxidant activity of synthetic cytokinin analogues: 6-alkynyl- and 6-alkenylpurines as novel 15-Lipoxygenase inhibitors
|
Bråthe, Anders |
|
2002 |
10 |
5 |
p. 1581-1586 6 p. |
artikel |
8 |
Aryl Cyclopentadienyl Tricarbonyl Rhenium Complexes: Novel Ligands for the Estrogen Receptor with Potential Use as Estrogen Radiopharmaceuticals
|
Mull, Eric S |
|
2002 |
10 |
5 |
p. 1381-1398 18 p. |
artikel |
9 |
Benzoyl and cinnamoyl nitrogen mustard derivatives of benzoheterocyclic analogues of the tallimustine: synthesis and antitumour activity
|
Baraldi, Pier Giovanni |
|
2002 |
10 |
5 |
p. 1611-1618 8 p. |
artikel |
10 |
Binding of 1-Benzopyran-4-one Derivatives to Aldose Reductase: A Free Energy Perturbation Study
|
Rastelli, Giulio |
|
2002 |
10 |
5 |
p. 1427-1436 10 p. |
artikel |
11 |
9-Carboxymethyl-5H,10H-imidazo[1,2-a]indeno[1,2-e]pyrazin-4-one-2-carbocylic Acid (RPR117824): Selective Anticonvulsive and Neuroprotective AMPA Antagonist
|
Mignani, Serge |
|
2002 |
10 |
5 |
p. 1627-1637 11 p. |
artikel |
12 |
Certification of the Critical Importance of l-3-(2-Naphthyl)alanine at Position 3 of a Specific CXCR4 Inhibitor, T140, Leads to an Exploratory Performance of Its Downsizing Study
|
Tamamura, Hirokazu |
|
2002 |
10 |
5 |
p. 1417-1426 10 p. |
artikel |
13 |
Coupling of Isoprenoid Triflates with Organoboron Nucleophiles: Synthesis and Biological Evaluation of Geranylgeranyl Diphosphate Analogues
|
Mu, YongQi |
|
2002 |
10 |
5 |
p. 1207-1219 13 p. |
artikel |
14 |
Discovery of diaminobutane derivatives as Ca2+-permeable AMPA receptor antagonists
|
Yoneda, Yoshiyuki |
|
2002 |
10 |
5 |
p. 1347-1359 13 p. |
artikel |
15 |
Discovery of new inhibitors of aldose reductase from molecular docking and database screening
|
Rastelli, Giulio |
|
2002 |
10 |
5 |
p. 1437-1450 14 p. |
artikel |
16 |
3-D-QSAR Analysis of N-(3-Acyloxy-2-benzylpropyl)-N′-dihydroxytetrahydrobenzazepine and Tetrahydroisoquinoline and N-(3-Acyloxy-2-benzylpropyl)-N′-(4-hydroxy-3-methoxybenzyl) Thioureas Analogues as Potent Vanilloid Receptor Ligands
|
Kim, Ki H. |
|
2002 |
10 |
5 |
p. 1367-1372 6 p. |
artikel |
17 |
Experimental and Calculated Shift in pK a upon Binding of Phosphotyrosine Peptide to the SH2 Domain of p56lck
|
de Mol, Nico J. |
|
2002 |
10 |
5 |
p. 1477-1482 6 p. |
artikel |
18 |
Fatty Acid Esters of Juvenoid Alcohols as Insect Hormonogen Agents (Juvenogens)
|
Wimmer, Zdeněk |
|
2002 |
10 |
5 |
p. 1305-1312 8 p. |
artikel |
19 |
Graphical Abstracts
|
|
|
2002 |
10 |
5 |
p. xi-xxi nvt p. |
artikel |
20 |
I2-Imidazoline Binding Site Affinity of a Structurally Different Type of Ligands
|
Dardonville, Christophe |
|
2002 |
10 |
5 |
p. 1525-1533 9 p. |
artikel |
21 |
Mapping of Possible Binding Sequences of Two Beta-Sheet Breaker Peptides on Beta Amyloid Peptide of Alzheimer's Disease
|
Hetényi, Csaba |
|
2002 |
10 |
5 |
p. 1587-1593 7 p. |
artikel |
22 |
Molecular Orbital Calculation for the Model Compounds of Kainoid Amino Acids, Agonists of Excitatory Amino Acid Receptors. Does the Kainoid C4-Substituent Directly Interact with the Receptors?
|
Hashimoto, Kimiko |
|
2002 |
10 |
5 |
p. 1373-1379 7 p. |
artikel |
23 |
Novel anthracycline oligosaccharides: influence of chemical modifications of the carbohydrate moiety on biological activity
|
Cipollone, A |
|
2002 |
10 |
5 |
p. 1459-1470 12 p. |
artikel |
24 |
Novel Irreversible Butyrylcholinesterase Inhibitors: 2-Chloro-1-(substituted-phenyl)ethylphosphonic Acids
|
Zhang, Nanjing |
|
2002 |
10 |
5 |
p. 1281-1290 10 p. |
artikel |
25 |
Novel Non-Steroidal/Non-Anilide Type Androgen Antagonists with an Isoxazolone Moiety
|
Ishioka, Toshiyasu |
|
2002 |
10 |
5 |
p. 1555-1566 12 p. |
artikel |
26 |
Novel Tn antigen-containing neoglycopeptides: synthesis and evaluation as anti tumor vaccines
|
Cipolla, Laura |
|
2002 |
10 |
5 |
p. 1639-1646 8 p. |
artikel |
27 |
Orally Active Cephalosporins. Part 4: Synthesis, Structure–Activity Relationships and Oral Absorption of Novel 3-(4-Pyrazolylmethylthio)cephalosporins with Various C-7 Side Chains
|
Yamamoto, Hirofumi |
|
2002 |
10 |
5 |
p. 1535-1545 11 p. |
artikel |
28 |
Polyene substrates with unusual methylation patterns to probe the active sites of three catalytic antibodies
|
Kim, Geun Tae |
|
2002 |
10 |
5 |
p. 1249-1262 14 p. |
artikel |
29 |
Powerful antioxidative agents based on garcinoic acid from Garcinia kola
|
Terashima, Kenji |
|
2002 |
10 |
5 |
p. 1619-1625 7 p. |
artikel |
30 |
QSAR of HIV-1 integrase inhibitors by genetic function approximation method
|
Makhija, Mahindra T. |
|
2002 |
10 |
5 |
p. 1483-1497 15 p. |
artikel |
31 |
QSAR Studies on Antimalarial Substituted Phenyl Analogues and Their Nω-Oxides
|
Agrawal, Vijay K. |
|
2002 |
10 |
5 |
p. 1361-1366 6 p. |
artikel |
32 |
Recognition of Bulged DNA by a Neocarzinostatin Product via an Induced Fit Mechanism
|
Yang, Catherine F. |
|
2002 |
10 |
5 |
p. 1329-1335 7 p. |
artikel |
33 |
Resolution of (RS)-Proglumide using Lipase from Candida cylindraceae
|
Muralidhar, R.V |
|
2002 |
10 |
5 |
p. 1471-1475 5 p. |
artikel |
34 |
Structure–Activity relationships among novel phenoxybenzamine-Related β-Chloroethylamines
|
Giardinà, Dario |
|
2002 |
10 |
5 |
p. 1291-1303 13 p. |
artikel |
35 |
Structure–Activity Relationships of 1β-Methyl-2-(5-phenylpyrrolidin-3-ylthio)carbapenems
|
Sato, Hiroki |
|
2002 |
10 |
5 |
p. 1595-1610 16 p. |
artikel |
36 |
Substituted Indoloquinolines as New Antifungal Agents
|
Ablordeppey, Seth Y |
|
2002 |
10 |
5 |
p. 1337-1346 10 p. |
artikel |
37 |
Synthesis and Biological Activity of 1-Phenylsulfonyl-4-Phenylsulfonylaminopyrrolidine Derivatives as Thromboxane A2 Receptor Antagonists
|
Marusawa, Hiroshi |
|
2002 |
10 |
5 |
p. 1399-1415 17 p. |
artikel |
38 |
Synthesis and biological evaluation of novel thioapio dideoxynucleosides
|
Moon, Hyung Ryong |
|
2002 |
10 |
5 |
p. 1499-1507 9 p. |
artikel |
39 |
Synthesis and Biological Properties of Amino Acid Amide Ligand-Based Pyridinioalkanoyl Thioesters as Anti-HIV Agents
|
Song, Yongsheng |
|
2002 |
10 |
5 |
p. 1263-1273 11 p. |
artikel |
40 |
Synthesis and 31P NMR characterization of new low toxic highly sensitive pH probes designed for in vivo acidic pH studies
|
Martel, Sophie |
|
2002 |
10 |
5 |
p. 1451-1458 8 p. |
artikel |
41 |
Synthesis of Potential Thrombin Inhibitors. Incorporation of Tartaric Acid Templates as P2 Proline Mimetics
|
Dahlgren, Anders |
|
2002 |
10 |
5 |
p. 1567-1580 14 p. |
artikel |
42 |
The Discovery of YM-60828: A Potent, Selective and Orally-Bioavailable Factor Xa Inhibitor
|
Hirayama, Fukushi |
|
2002 |
10 |
5 |
p. 1509-1523 15 p. |
artikel |
43 |
The 1.76 Å Resolution Crystal Structure of Glycogen Phosphorylase b Complexed with Glucose, and CP320626, a Potential Antidiabetic Drug
|
Oikonomakos, Nikos G |
|
2002 |
10 |
5 |
p. 1313-1319 7 p. |
artikel |