nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
1 |
A cell-penetrating peptide from a novel pVII–pIX phage-displayed random peptide library
|
Gao, Changshou |
|
2002 |
10 |
12 |
p. 4057-4065 9 p. |
artikel |
2 |
1-Alkoxycarbonyl-3-halogenoazetidin-2-ones as elastase (PPE) inhibitors
|
Gérard, Stéphane |
|
2002 |
10 |
12 |
p. 3955-3964 10 p. |
artikel |
3 |
A novel class of endothelin-A receptor antagonists, (R)-2-(benzo[1,3]dioxol-5-yl)-6-isopropyloxy-2H-chromene-3-carboxylic acids (S-1255). Conformational analysis of basic structure, crucial for ETA antagonism, in solution and solid states
|
Ishizuka, Natsuki |
|
2002 |
10 |
12 |
p. 3965-3972 8 p. |
artikel |
4 |
Anti-HIV-1 peptides derived from partial amino acid sequences of CC-Chemokine RANTES
|
Nishiyama, Yasuhiro |
|
2002 |
10 |
12 |
p. 4113-4117 5 p. |
artikel |
5 |
Author Index
|
|
|
2002 |
10 |
12 |
p. VII-XXI nvt p. |
artikel |
6 |
Binding affinity prediction of novel estrogen receptor ligands using receptor-based 3-D QSAR methods
|
Sippl, Wolfgang |
|
2002 |
10 |
12 |
p. 3741-3755 15 p. |
artikel |
7 |
Characterization of a Binding Site for Template Competitive Inhibitors of HIV-1 Reverse Transcriptase Using Photolabeling Derivatives
|
Lin, Weiying |
|
2002 |
10 |
12 |
p. 4131-4141 11 p. |
artikel |
8 |
Combining molecular modeling with experimental methodologies: mechanism of membrane permeation and accumulation of ofloxacin
|
Fresta, Massimo |
|
2002 |
10 |
12 |
p. 3871-3889 19 p. |
artikel |
9 |
Design and synthesis of novel imidazole derivatives as potent inhibitors of allene oxide synthase(CYP74)
|
Oh, Keimei |
|
2002 |
10 |
12 |
p. 3707-3711 5 p. |
artikel |
10 |
Design of Inhibitors of Scytalone Dehydratase: Probing Interactions with an Asparagine Carboxamide
|
Basarab, Gregory S |
|
2002 |
10 |
12 |
p. 4143-4154 12 p. |
artikel |
11 |
Design, synthesis and antitumor activities of novel 7-arylseleno-7-deoxydaunomycinone derivatives
|
Zhang, Shu-Jia |
|
2002 |
10 |
12 |
p. 3899-3904 6 p. |
artikel |
12 |
Design, Synthesis, Conformational Analysis, and Biological Studies of Urotensin-II Lactam Analogues
|
Grieco, Paolo |
|
2002 |
10 |
12 |
p. 3731-3739 9 p. |
artikel |
13 |
Development of 3D-QSAR models for 5-Lipoxygenase antagonists: chalcones
|
Arockia Babu, M |
|
2002 |
10 |
12 |
p. 4035-4041 7 p. |
artikel |
14 |
Discovery of Novel Phosphonic Acid Derivatives as New Chemical Leads for Inhibitors of TNF-α production
|
Matsui, Toshiaki |
|
2002 |
10 |
12 |
p. 3807-3815 9 p. |
artikel |
15 |
2D-QSAR in hydroxamic acid derivatives as peptide deformylase inhibitors and antibacterial agents
|
Gupta, Manish K |
|
2002 |
10 |
12 |
p. 3713-3716 4 p. |
artikel |
16 |
Erratum to “A simple method for the preparation of (5Z,8Z,11Z,14Z)-16-Hydroxyeicosa-5,8,11,14-tetraenoic acid enantiomers and the corresponding 14,15-Dehydro analogues: role of the 16-Hydroxy group for the lipoxygenase reaction”
|
Ivanov, Igor V |
|
2002 |
10 |
12 |
p. 4193- 1 p. |
artikel |
17 |
Facile synthesis of stable lipid analogues possessing a range of alkyl groups: application to artificial glycolipids
|
Azefu, Yasuo |
|
2002 |
10 |
12 |
p. 4013-4022 10 p. |
artikel |
18 |
Folded conformation of an immunostimulating tetrapeptide Rigin: high temperature molecular dynamics simulation study
|
Ashish, A. |
|
2002 |
10 |
12 |
p. 4083-4090 8 p. |
artikel |
19 |
Graphical Abstracts
|
|
|
2002 |
10 |
12 |
p. 3695-3706 12 p. |
artikel |
20 |
Highly potent inhibitors of TNF-α production. Part I
|
Matsui, Toshiaki |
|
2002 |
10 |
12 |
p. 3757-3786 30 p. |
artikel |
21 |
Highly potent inhibitors of tnf-α production. Part II: metabolic stabilization of a newly found chemical lead and conformational analysis of an active diastereoisomer
|
Matsui, Toshiaki |
|
2002 |
10 |
12 |
p. 3787-3805 19 p. |
artikel |
22 |
Inhibitors of nitric oxide production from the bark of Myrica rubra: structures of new biphenyl type diarylheptanoid glycosides and taraxerane type triterpene
|
Tao, Jing |
|
2002 |
10 |
12 |
p. 4005-4012 8 p. |
artikel |
23 |
Inside Front Cover
|
|
|
2002 |
10 |
12 |
p. IFC- 1 p. |
artikel |
24 |
Mapping of the active site of rat kidney γ-glutamyl transpeptidase using activated esters and their amide derivatives
|
Castonguay, Roselyne |
|
2002 |
10 |
12 |
p. 4185-4191 7 p. |
artikel |
25 |
Mechanism of biochemical action of substituted 4-methylbenzopyran-2-ones. Part 9: Comparison of acetoxy 4-methylcoumarins and other polyphenolic acetates reveal the specificity to acetoxy drug: protein transacetylase for pyran carbonyl group in proximity to the oxygen heteroatom
|
Singh, Ishwar |
|
2002 |
10 |
12 |
p. 4103-4111 9 p. |
artikel |
26 |
Membrane-Permeant derivatives of mannose-1-phosphate
|
Rutschow, Synke |
|
2002 |
10 |
12 |
p. 4043-4049 7 p. |
artikel |
27 |
1-Methoxy-, 1-deoxy-11-hydroxy- and 11-Hydroxy-1-methoxy-Δ8-tetrahydrocannabinols: new selective ligands for the CB2 receptor
|
Huffman, John W |
|
2002 |
10 |
12 |
p. 4119-4129 11 p. |
artikel |
28 |
New water-soluble prodrugs of HIV protease inhibitors based on O→N intramolecular acyl migration
|
Hamada, Yoshio |
|
2002 |
10 |
12 |
p. 4155-4167 13 p. |
artikel |
29 |
Nitrophenyl Derivatives as Aldose Reductase Inhibitors
|
Costantino, Luca |
|
2002 |
10 |
12 |
p. 3923-3931 9 p. |
artikel |
30 |
Novel (bisarylmethoxy)butylpiperidine analogues as neurotransmitter transporter inhibitors with activity at dopamine receptor sites
|
Choi, Sung-Woon |
|
2002 |
10 |
12 |
p. 4091-4102 12 p. |
artikel |
31 |
On the topological evidences for modelling lipophilicity
|
Agrawal, Vijay K. |
|
2002 |
10 |
12 |
p. 3981-3996 16 p. |
artikel |
32 |
Progress in arylpiperazine synthesis by the catalytic amination reaction
|
Torisawa, Yasuhiro |
|
2002 |
10 |
12 |
p. 4023-4027 5 p. |
artikel |
33 |
QSAR studies of HIV-1 integrase inhibition
|
Yuan, Hongbin |
|
2002 |
10 |
12 |
p. 4169-4183 15 p. |
artikel |
34 |
Stereoselectivity in reactions of amino acids catalyzed by pyridoxal derivatives carrying rigidly-Attached chirally-Mounted basic groups—transamination, racemization, decarboxylation, retro-Aldol reaction, and aldol condensation
|
Liu, Lei |
|
2002 |
10 |
12 |
p. 3973-3979 7 p. |
artikel |
35 |
Straightforward Syntheses of Furanomycin Derivatives and their Biological Evaluation
|
Kazmaier, Uli |
|
2002 |
10 |
12 |
p. 3905-3913 9 p. |
artikel |
36 |
Study on the multiple mechanisms underlying the reaction between hydroxyl radical and phenolic compounds by qualitative structure and activity relationship
|
Cheng, Zhiyong |
|
2002 |
10 |
12 |
p. 4067-4073 7 p. |
artikel |
37 |
Sulfamoyloxy-substituted 2-phenylindoles
|
Golob, Thomas |
|
2002 |
10 |
12 |
p. 3941-3953 13 p. |
artikel |
38 |
Synthesis and biological evaluation of new mannose 6-phosphate analogues
|
Vidal, Sébastien |
|
2002 |
10 |
12 |
p. 4051-4056 6 p. |
artikel |
39 |
Synthesis and Biological Studies of Novel Neurotensin(8–13) Mimetics
|
Hong, Feng |
|
2002 |
10 |
12 |
p. 3849-3858 10 p. |
artikel |
40 |
Synthesis and estrogen receptor affinity of a 4-hydroxytamoxifen-Labeled ligand for diagnostic imaging
|
Lashley, Matthew R |
|
2002 |
10 |
12 |
p. 4075-4082 8 p. |
artikel |
41 |
Synthesis and evaluation of anticancer benzoxazoles and benzimidazoles related to UK-1
|
Kumar, Devinder |
|
2002 |
10 |
12 |
p. 3997-4004 8 p. |
artikel |
42 |
Synthesis and pharmacological evaluation of new arylpiperazines. 3-{4-[4-(3-chlorophenyl)-1-piperazinyl]butyl}-quinazolidin-4-one — a dual serotonin 5-HT1A/5-HT2A receptor ligand with an anxiolytic-like activity
|
Bojarski, Andrzej J |
|
2002 |
10 |
12 |
p. 3817-3827 11 p. |
artikel |
43 |
Synthesis and Structure–Activity Relationship of Dehydroxymethylepoxyquinomicin Analogues as Inhibitors of NF-κB Functions
|
Chaicharoenpong, Chanya |
|
2002 |
10 |
12 |
p. 3933-3939 7 p. |
artikel |
44 |
Synthesis, Conformation and T-Helper Cell Stimulation of an O-Linked Glycopeptide Epitope Containing Extended Carbohydrate Side-Chains
|
Cudic, Mare |
|
2002 |
10 |
12 |
p. 3859-3870 12 p. |
artikel |
45 |
Synthesis of 3-alkyl(Aryl)-4-alkylidenamino-4,5-dihydro-1H-1,2,4-triazol-5-ones and 3-alkyl-4-alkylamino-4,5-dihydro-1H-1,2,4-triazol-5-ones as antitumor agents
|
Demirbaş, Neslihan |
|
2002 |
10 |
12 |
p. 3717-3723 7 p. |
artikel |
46 |
Synthesis of derivatives of (1S,2R)-1-phenyl-2-[(S)-1-aminopropyl]-N,N-diethylcyclopropanecarboxamide (PPDC) modified at the 1-aromatic moiety as novel NMDA receptor antagonists: the aromatic group is essential for the activity
|
Kazuta, Yuji |
|
2002 |
10 |
12 |
p. 3829-3848 20 p. |
artikel |
47 |
Synthesis of silicon-containing azole derivatives with magnesium bromide diethyl etherate, and an investigation of their fungicidal activities
|
Itoh, Hiroyuki |
|
2002 |
10 |
12 |
p. 4029-4034 6 p. |
artikel |
48 |
Tetrapeptides as potent protease inhibitors of hepatitis C virus full-Length NS3 (Protease-Helicase/NTPase)
|
Johansson, Anja |
|
2002 |
10 |
12 |
p. 3915-3922 8 p. |
artikel |
49 |
The product of the natural reaction catalyzed by 4-oxalocrotonate tautomerase becomes an affinity label of its mutant
|
Brik, Ashraf |
|
2002 |
10 |
12 |
p. 3891-3897 7 p. |
artikel |
50 |
Volume Contents 2002
|
|
|
2002 |
10 |
12 |
p. XXIII-LII nvt p. |
artikel |
51 |
Xanthones as inhibitors of growth of human cancer cell lines and Their effects on the proliferation of human lymphocytes In Vitro
|
Pedro, Madalena |
|
2002 |
10 |
12 |
p. 3725-3730 6 p. |
artikel |