| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
A Convenient Synthetic Method of a 5,7-Diarylcyclopenteno-[1,2-b]pyridine-6-carboxylate: A Key Intermediate for Potent Endothelin Receptor Antagonists
|
Niiyama, Kenji
|
|
2002
|
10 |
11 |
p. 3437-3444
8 p.
|
artikel
|
| 2 |
A convergent synthesis of core 2 branched sialylated and sulfated oligosaccharides
|
Xia, Jie
|
|
2002
|
10 |
11 |
p. 3673-3684
12 p.
|
artikel
|
| 3 |
Antitumor Agents. Part 214: † † For paper 213, see ref 1. Synthesis and Evaluation of Curcumin Analogues as Cytotoxic Agents
|
Ishida, Junko
|
|
2002
|
10 |
11 |
p. 3481-3487
7 p.
|
artikel
|
| 4 |
A structure–activity study of spermicidal and anti-HIV properties of hydroxylated cationic surfactants
|
Wong, Yue-Ling
|
|
2002
|
10 |
11 |
p. 3599-3608
10 p.
|
artikel
|
| 5 |
1,4-Benzothiazine and 1,4-Benzoxazine imidazole derivatives with antifungal activity: A docking study
|
Macchiarulo, Antonio
|
|
2002
|
10 |
11 |
p. 3415-3423
9 p.
|
artikel
|
| 6 |
Design and synthesis of an irreversible dopamine-sparing cocaine antagonist
|
Meltzer, Peter C.
|
|
2002
|
10 |
11 |
p. 3583-3591
9 p.
|
artikel
|
| 7 |
Design, Synthesis, and Biological Evaluation of a Series of β-Lactam-Based Prodrugs
|
Hakimelahi, Gholam Hossein
|
|
2002
|
10 |
11 |
p. 3489-3498
10 p.
|
artikel
|
| 8 |
Determination of the phamacophore of penclomedine, a clinically-evaluated antitumor pyridine derivative
|
Tiwari, Anita
|
|
2002
|
10 |
11 |
p. 3593-3598
6 p.
|
artikel
|
| 9 |
Development of a Purine-Scaffold Novel Class of Hsp90 Binders that Inhibit the Proliferation of Cancer Cells and Induce the Degradation of Her2 Tyrosine Kinase
|
Chiosis, Gabriela
|
|
2002
|
10 |
11 |
p. 3555-3564
10 p.
|
artikel
|
| 10 |
Editorial Board (Inside Front Cover)
|
|
|
2002
|
10 |
11 |
p. IFC-
1 p.
|
artikel
|
| 11 |
Erratum to “Novel potent 5-HT3 receptor ligands based on the pyrrolidone structure. effects of the quaternization of the basic nitrogen on the interaction with 5-HT3 receptor” [Bioorg. Med. Chem. 10 (2002) 2681]
|
Cappelli, Andrea
|
|
2002
|
10 |
11 |
p. 3693-
1 p.
|
artikel
|
| 12 |
Footprinting and circular dichroism studies on paromomycin binding to the packaging region of human immunodeficiency virus type-1
|
McPike, Mark P.
|
|
2002
|
10 |
11 |
p. 3663-3672
10 p.
|
artikel
|
| 13 |
Graphical Abstracts
|
|
|
2002
|
10 |
11 |
p. 3369-3377
9 p.
|
artikel
|
| 14 |
Halohydrin and Oxime Derivatives of Radicicol: Synthesis and Antitumor Activities
|
Agatsuma, Tsutomu
|
|
2002
|
10 |
11 |
p. 3445-3454
10 p.
|
artikel
|
| 15 |
Hemi-synthesis and Biological Activity of New Analogues of Podophyllotoxin
|
Roulland, Emmanuel
|
|
2002
|
10 |
11 |
p. 3463-3471
9 p.
|
artikel
|
| 16 |
Highly-Iodinated Fullerene as a Contrast Agent For X-ray Imaging
|
Wharton, Tim
|
|
2002
|
10 |
11 |
p. 3545-3554
10 p.
|
artikel
|
| 17 |
Inhibition of inosine monophosphate dehydrogenase (IMPDH) by the antiviral compound, 2-vinylinosine monophosphate
|
Pal, Suresh
|
|
2002
|
10 |
11 |
p. 3615-3618
4 p.
|
artikel
|
| 18 |
Methylation of l-trans-2,4-Pyrrolidine Dicarboxylate Converts the Glutamate Transport Inhibitor from a Substrate to a Non-substrate Inhibitor
|
Esslinger, C.Sean
|
|
2002
|
10 |
11 |
p. 3509-3515
7 p.
|
artikel
|
| 19 |
New dsDNA binding unnatural oligopeptides with pyrimidine selectivity
|
Zhang, Zhenyu
|
|
2002
|
10 |
11 |
p. 3401-3413
13 p.
|
artikel
|
| 20 |
Novel and Potent Anti-malarial Agents
|
Brinner, Kristin M
|
|
2002
|
10 |
11 |
p. 3649-3661
13 p.
|
artikel
|
| 21 |
Novel Branching Membrane Translocational Peptide as Gene Delivery Vector
|
Tung, Ching-Hsuan
|
|
2002
|
10 |
11 |
p. 3609-3614
6 p.
|
artikel
|
| 22 |
Novel peptidomimics as angiotensin-Converting enzyme inhibitors: A combinatorial approach
|
Bala, Manju
|
|
2002
|
10 |
11 |
p. 3685-3691
7 p.
|
artikel
|
| 23 |
Phospholipid-Bound Molecular Rotors: Synthesis and Characterization
|
Haidekker, Mark A.
|
|
2002
|
10 |
11 |
p. 3627-3636
10 p.
|
artikel
|
| 24 |
Prediction of lipophilicity of polyacenes using quantitative structure–Activity relationships
|
Khadikar, Padmakar V.
|
|
2002
|
10 |
11 |
p. 3499-3507
9 p.
|
artikel
|
| 25 |
QSAR study on narcotic mechanism of action and toxicity: a molecular connectivity approach to Vibrio fischeri toxicity testing
|
Agrawal, Vijay K.
|
|
2002
|
10 |
11 |
p. 3517-3522
6 p.
|
artikel
|
| 26 |
Quantitative structure–Activity relationship studies on 5-phenyl-3-ureido-1,5-benzodiazepine as cholecystokinin-A receptor antagonists
|
Agrawal, Vijay K.
|
|
2002
|
10 |
11 |
p. 3571-3581
11 p.
|
artikel
|
| 27 |
5-Substituted-1H-tetrazoles as carboxylic acid isosteres: medicinal chemistry and synthetic methods
|
Herr, R.Jason
|
|
2002
|
10 |
11 |
p. 3379-3393
15 p.
|
artikel
|
| 28 |
Synthesis and biological evaluation of a-Ring biaryl-carbamate analogues of rhazinilam
|
Baudoin, Olivier
|
|
2002
|
10 |
11 |
p. 3395-3400
6 p.
|
artikel
|
| 29 |
Synthesis and physical characterization of a P1 arginine combinatorial library, and its application to the determination of the substrate specificity of serine peptidases
|
Furlong, Stephen T.
|
|
2002
|
10 |
11 |
p. 3637-3647
11 p.
|
artikel
|
| 30 |
Synthesis and Structure–Activity Relationship of Diarylamide Derivatives as Selective Inhibitors of the Proliferation of Human Endothelial Cells
|
Ogita, Haruhisa
|
|
2002
|
10 |
11 |
p. 3473-3480
8 p.
|
artikel
|
| 31 |
Synthesis of (−)-5,8-Dihydroxy-3R-methyl-2R-(dipropylamino)-1,2,3,4-tetrahydronaphthalene: An Inhibitor of β-Amyloid1–42 Aggregation
|
Parker, Michael H
|
|
2002
|
10 |
11 |
p. 3565-3569
5 p.
|
artikel
|
| 32 |
Synthesis of 17β-N-Substituted 19-Nor-10-azasteroids as Inhibitors of Human 5α-Reductases I and II
|
Scarpi, Dina
|
|
2002
|
10 |
11 |
p. 3455-3461
7 p.
|
artikel
|
| 33 |
Tc and Re Chelates of 8α-Amino-6-methyl-ergoline: Synthesis and Affinity to the Dopamine D2 Receptor
|
Spies, H
|
|
2002
|
10 |
11 |
p. 3523-3528
6 p.
|
artikel
|
| 34 |
Tetrahydroisoquinoline-3-carboxylate based matrix-metalloproteinase inhibitors: design, synthesis and structure–activity relationship
|
Matter, Hans
|
|
2002
|
10 |
11 |
p. 3529-3544
16 p.
|
artikel
|
| 35 |
Thalassiolins A–C: new marine-derived inhibitors of HIV cDNA integrase
|
Rowley, David C
|
|
2002
|
10 |
11 |
p. 3619-3625
7 p.
|
artikel
|
| 36 |
The disaccharide anthracycline MEN 10755 binds human serum albumin to a non-classical drug binding site
|
Messori, Luigi
|
|
2002
|
10 |
11 |
p. 3425-3430
6 p.
|
artikel
|
| 37 |
Xanthones as inhibitors of microsomal lipid peroxidation and TNF-α induced ICAM-1 expression on human umbilical vein endothelial cells (HUVECs)
|
Madan, Babita
|
|
2002
|
10 |
11 |
p. 3431-3436
6 p.
|
artikel
|
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