Cyclic AMP Analog Blocks Kinase Activation by Stabilizing Inactive Conformation: Conformational Selection Highlights a New Concept in Allosteric Inhibitor Design*
Titel:
Cyclic AMP Analog Blocks Kinase Activation by Stabilizing Inactive Conformation: Conformational Selection Highlights a New Concept in Allosteric Inhibitor Design*
Auteur:
Badireddy, Suguna Yunfeng, Gao Ritchie, Mark Akamine, Pearl Wu, Jian Kim, Choel W. Taylor, Susan S. Qingsong, Lin Swaminathan, Kunchithapadam Anand, Ganesh S.