Discovery, preclinical validation and early human imaging with [11C]AZ14193391 – the first blood-brain barrier permeable and subtype selective PARP1 PET radioligand
Title:
Discovery, preclinical validation and early human imaging with [11C]AZ14193391 – the first blood-brain barrier permeable and subtype selective PARP1 PET radioligand
Author:
Cortes Gonzalez, Miguel Angel Jucaite, Aurelija Cselenyi, Zsolt Johnstrom, Peter Pike, Andy Högnäsbacka, Antonia Dahl, Kenneth Balazs, Amber Degorce, Sébastien Ghosh, Avipsa Hande, Sudir Johannes, Jeffrey Staniewska, Anna Leo, Elizabetta Hammerlik, Petra Davies, Barry Cosulich, Sabrina Swales, John Lawrence, Rachel Stenkrona, Per Farde, Lars Halldin, Christer Schou, Magnus