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Discovery of Pyrazolo[1,5-a]pyrazin-4-ones as Potent and Brain Penetrant GluN2A-Selective Positive Allosteric Modulators Reducing AMPA Receptor Binding Activity |
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Titel: |
Discovery of Pyrazolo[1,5-a]pyrazin-4-ones as Potent and Brain Penetrant GluN2A-Selective Positive Allosteric Modulators Reducing AMPA Receptor Binding Activity |
Auteur: |
Sakurai, Fumie Yukawa, Takafumi Kina, Asato Murakami, Masataka Takami, Kazuaki Morimoto, Sachie Seto, Masaki Kamata, Makoto Yamashita, Tohru Nakashima, Kosuke Narita, Naohiro Bettini, Ezio Ugolini, Annarosa Corsi, Mauro Hasui, Tomoaki |
Verschenen in: |
Bioorganic & medicinal chemistry |
Paginering: |
Jaargang 56 () nr. C pagina's p. |
Jaar: |
2022 |
Inhoud: |
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Uitgever: |
The Author(s) |
Bronbestand: |
Elektronische Wetenschappelijke Tijdschriften |
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