Discovery of isoquinolinone and naphthyridinone-based inhibitors of poly(ADP-ribose) polymerase-1 (PARP1) as anticancer agents: Structure activity relationship and preclinical characterization
Titel:
Discovery of isoquinolinone and naphthyridinone-based inhibitors of poly(ADP-ribose) polymerase-1 (PARP1) as anticancer agents: Structure activity relationship and preclinical characterization
Auteur:
Karche, Navnath P. Bhonde, Mandar Sinha, Neelima Jana, Gourhari Kukreja, Gagan Kurhade, Sanjay P. Jagdale, Arun R. Tilekar, Ajay R. Hajare, Anil K. Jadhav, Ganesh R. Gupta, Nishant R. Limaye, Rohan Khedkar, Nilesh Thube, Baban R. Shaikh, Javed S. Rao Irlapati, Nageswara Phukan, Samiron Gole, Gopal Bommakanti, Apparao Khanwalkar, Harshal Pawar, Yogesh Kale, Ramesh Kumar, Rakesh Gupta, Rajesh Praveen Kumar, V.R. Wahid, Saif Francis, Albi Bhat, Tariq Kamble, Nivrutti Patil, Vinod Nigade, Prashant B. Modi, Dipak Pawar, Shashikant Naidu, Sneha Volam, Harish Pagdala, Vamsi Mallurwar, Sadanand Goyal, Hemant Bora, Pushpak Ahirrao, Prajakta Singh, Minakshi Kamalakannan, Prabhakaran Naik, Kumar Ram Kumar, Pradipta Powar, Rajendra G. Shankar, Rajesh B. Bernstein, Peter R. Gundu, Jayasagar Nemmani, Kumar Narasimham, Lakshmi George, Kochumalayil Shaji Sharma, Sharad Bakhle, Dhananjay Kamboj, Rajender Kumar Palle, Venkata P.