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Discovery of orally efficacious RORγt inverse agonists, part 1: Identification of novel phenylglycinamides as lead scaffolds |
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Titel: |
Discovery of orally efficacious RORγt inverse agonists, part 1: Identification of novel phenylglycinamides as lead scaffolds |
Auteur: |
Shirai, Junya Tomata, Yoshihide Kono, Mitsunori Ochida, Atsuko Fukase, Yoshiyuki Sato, Ayumu Masada, Shinichi Kawamoto, Tetsuji Yonemori, Kazuko Koyama, Ryoukichi Nakagawa, Hideyuki Nakayama, Masaharu Uga, Keiko Shibata, Akira Koga, Keiko Okui, Toshitake Shirasaki, Mikio Skene, Robert Sang, BiChing Hoffman, Isaac Lane, Wes Fujitani, Yasushi Yamasaki, Masashi Yamamoto, Satoshi |
Verschenen in: |
Bioorganic & medicinal chemistry |
Paginering: |
Jaargang 26 () nr. 2 pagina's 483-500 |
Jaar: |
2018 |
Inhoud: |
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Uitgever: |
Elsevier Ltd |
Bronbestand: |
Elektronische Wetenschappelijke Tijdschriften |
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