Exploiting a water network to achieve enthalpy-driven, bromodomain-selective BET inhibitors
Title:
Exploiting a water network to achieve enthalpy-driven, bromodomain-selective BET inhibitors
Author:
Shadrick, William R. Slavish, Peter J. Chai, Sergio C. Waddell, Brett Connelly, Michele Low, Jonathan A. Tallant, Cynthia Young, Brandon M. Bharatham, Nagakumar Knapp, Stefan Boyd, Vincent A. Morfouace, Marie Roussel, Martine F. Chen, Taosheng Lee, Richard E. Kiplin Guy, R. Shelat, Anang A. Potter, Philip M.