Optimization of potency and pharmacokinetics of tricyclic indole derived inhibitors of HCV NS5B polymerase. Identification of ester prodrugs with improved oral pharmacokinetics
Titel:
Optimization of potency and pharmacokinetics of tricyclic indole derived inhibitors of HCV NS5B polymerase. Identification of ester prodrugs with improved oral pharmacokinetics
Auteur:
Venkatraman, Srikanth Velazquez, Francisco Gavalas, Stephen Wu, Wanli Chen, Kevin X. Nair, Anilkumar G. Bennett, Frank Huang, Yuhua Pinto, Patrick Jiang, Yueheng Selyutin, Oleg Vibulbhan, Bancha Zeng, Qingbei Lesburg, Charles Duca, Jose Heimark, Larry Huang, Hsueh-Cheng Agrawal, Sony Jiang, Chuan-kui Ferrari, Eric Li, Cheng Kozlowski, Joseph Rosenblum, Stuart Shih, Neng-Yang Njoroge, F. George