Targeting conserved water molecules: Design of 4-aryl-5-cyanopyrrolo[2,3-d]pyrimidine Hsp90 inhibitors using fragment-based screening and structure-based optimization
Title:
Targeting conserved water molecules: Design of 4-aryl-5-cyanopyrrolo[2,3-d]pyrimidine Hsp90 inhibitors using fragment-based screening and structure-based optimization
Author:
Davies, Nicholas G.M. Browne, Helen Davis, Ben Drysdale, Martin J. Foloppe, Nicolas Geoffrey, Stephanie Gibbons, Ben Hart, Terance Hubbard, Roderick Jensen, Michael Rugaard Mansell, Howard Massey, Andrew Matassova, Natalia Moore, Jonathan D. Murray, James Pratt, Robert Ray, Stuart Robertson, Alan Roughley, Stephen D. Schoepfer, Joseph Scriven, Kirsten Simmonite, Heather Stokes, Stephen Surgenor, Allan Webb, Paul Wood, Mike Wright, Lisa Brough, Paul