Rational conversion of noncontinuous active region in proteins into a small orally bioavailable macrocyclic drug-like molecule: The HIV-1 CD4:gp120 paradigm
Titel:
Rational conversion of noncontinuous active region in proteins into a small orally bioavailable macrocyclic drug-like molecule: The HIV-1 CD4:gp120 paradigm
Auteur:
Hurevich, Mattan Swed, Avi Joubran, Salim Cohen, Shira Freeman, Noam S. Britan-Rosich, Elena Briant-Longuet, Laurence Bardy, Martine Devaux, Christian Kotler, Moshe Hoffman, Amnon Gilon, Chaim