Cellular pharmacokinetics and pharmacodynamics of the deoxycytidine analog 2′-C-cyano-2′-deoxy-1-β-d-arabino-pentofuranosylcytosine (CNDAC) 1 1 Abbreviations: ara-C, ara-CMP, and ara-CTP, 1-β-d-arabinofuranosylcytosine and its 5′-mono- and triphosphate, respectively; CNDAC, CNDACMP, CNDACDP, and CNDACTP, 2′-C-cyano-2′-deoxy-1-β-d-arabino-pentofuranosylcytosine and its 5′-mono-, di-, and triphosphate, respectively; dNTP, deoxynucleoside triphosphate; CEM, CCRF-CEM human lymphoblastoid cells; and pol, DNA polymerase.
Titel:
Cellular pharmacokinetics and pharmacodynamics of the deoxycytidine analog 2′-C-cyano-2′-deoxy-1-β-d-arabino-pentofuranosylcytosine (CNDAC) 1 1 Abbreviations: ara-C, ara-CMP, and ara-CTP, 1-β-d-arabinofuranosylcytosine and its 5′-mono- and triphosphate, respectively; CNDAC, CNDACMP, CNDACDP, and CNDACTP, 2′-C-cyano-2′-deoxy-1-β-d-arabino-pentofuranosylcytosine and its 5′-mono-, di-, and triphosphate, respectively; dNTP, deoxynucleoside triphosphate; CEM, CCRF-CEM human lymphoblastoid cells; and pol, DNA polymerase.