no |
title |
author |
magazine |
year |
volume |
issue |
page(s) |
type |
1 |
A combined experimental and computational study on peptide nucleic acid (PNA) analogues of tumor suppressive miRNA-34a
|
Piacenti, Valerio |
|
|
91 |
C |
p. |
article |
2 |
Amide-tethered quinoline-resorcinol conjugates as a new class of HSP90 inhibitors suppressing the growth of prostate cancer cells
|
Nepali, Kunal |
|
|
91 |
C |
p. |
article |
3 |
An efficient method for the synthesis of novel derivatives 4-{5-[4-(4-amino-5-mercapto-4H-[1,2,4]triazol-3-yl)-phenyl]-3-trifluoromethyl-pyrazol-1-yl}-benzenesulfonamide and their anti-inflammatory potential
|
Mustafa, Ghulam |
|
|
91 |
C |
p. |
article |
4 |
Antifungal activity and tautomeric cyclization equilibria of formylphenylboronic acids
|
Borys, Krzysztof M. |
|
|
91 |
C |
p. |
article |
5 |
Anti-inflammatory and antiproliferative prenylated carbazole alkaloids from Clausena vestita
|
Liu, Yan-Ping |
|
|
91 |
C |
p. |
article |
6 |
Anti-inflammatory spiroaxane and drimane sesquiterpenoids from Talaromyces minioluteus (Penicillium minioluteum)
|
Chen, Chunmei |
|
|
91 |
C |
p. |
article |
7 |
Arylboronate prodrugs of doxorubicin as promising chemotherapy for pancreatic cancer
|
Skarbek, Charles |
|
|
91 |
C |
p. |
article |
8 |
A solid-phase method for synthesis of dimeric and trimeric ligands: Identification of potent bivalent ligands of 14-3-3σ
|
Lee, Yeongju |
|
|
91 |
C |
p. |
article |
9 |
Bioactivatable reductive cleavage of azobenzene for controlling functional dumbbell oligodeoxynucleotides
|
Lei, Huajun |
|
|
91 |
C |
p. |
article |
10 |
Bis-coumarins; non-cytotoxic selective urease inhibitors and antiglycation agents
|
Salar, Uzma |
|
|
91 |
C |
p. |
article |
11 |
cAMPS derivatives. A minireview over synthetic medicinal chemistry
|
Undheim, Kjell |
|
|
91 |
C |
p. |
article |
12 |
Chalcone derivatives and their antibacterial activities: Current development
|
Xu, Man |
|
|
91 |
C |
p. |
article |
13 |
Chemical constituents of the root bark of Ulmus davidiana var. japonica and their potential biological activities
|
So, Hae Min |
|
|
91 |
C |
p. |
article |
14 |
Chemo-sensitizing activity of natural cadinanes from Heterotheca inuloides in human uterine sarcoma cells and their in silico interaction with ABC transporters
|
Rodríguez-Chávez, José Luis |
|
|
91 |
C |
p. |
article |
15 |
Designing of promising medicinal scaffolds for Alzheimer’s disease through enzyme inhibition, lead optimization, molecular docking and dynamic simulation approaches
|
Hassan, Mubashir |
|
|
91 |
C |
p. |
article |
16 |
Design, synthesis and antibacterial activity evaluation of moxifloxacin-amide-1,2,3-triazole-isatin hybrids
|
Gao, Feng |
|
|
91 |
C |
p. |
article |
17 |
Design, synthesis and biological evaluation of 4-aminoquinoline-guanylthiourea derivatives as antimalarial agents
|
Bhagat, Shweta |
|
|
91 |
C |
p. |
article |
18 |
Design, synthesis and biological evaluation of novel perimidine o-quinone derivatives as non-intercalative topoisomerase II catalytic inhibitors
|
Zhou, Du-Chao |
|
|
91 |
C |
p. |
article |
19 |
Design, synthesis and biological evaluation of trinary benzocoumarin-thiazoles-azomethines derivatives as effective and selective inhibitors of alkaline phosphatase
|
Channar, Pervaiz Ali |
|
|
91 |
C |
p. |
article |
20 |
Design, synthesis and evaluation of phthalazinone thiohydantoin-based derivative as potent PARP-1 inhibitors
|
Zhong, Yi |
|
|
91 |
C |
p. |
article |
21 |
Design, synthesis, anticancer evaluation and docking studies of new pyrimidine derivatives as potent thymidylate synthase inhibitors
|
Amin, Lamia H.T. |
|
|
91 |
C |
p. |
article |
22 |
Design, synthesis, biological and in silico evaluation of coumarin-hydrazone derivatives as tubulin targeted antiproliferative agents
|
Govindaiah, Pilli |
|
|
91 |
C |
p. |
article |
23 |
Design, synthesis, molecular modeling and anti-hyperglycemic evaluation of phthalimide-sulfonylurea hybrids as PPARγ and SUR agonists
|
El-Zahabi, Mohamed Ayman |
|
|
91 |
C |
p. |
article |
24 |
Discovery of Michael acceptor containing 1,4-dihydropyridines as first covalent inhibitors of L-/T-type calcium channels
|
Aygün Cevher, Hande |
|
|
91 |
C |
p. |
article |
25 |
Discovery of novel cage-like heterocyclic hybrids as anti-inflammatory agents through the inhibition of nitrite, PGE2 and TNF-α
|
Kumar, Raju Suresh |
|
|
91 |
C |
p. |
article |
26 |
Discovery, synthesis and molecular substantiation of N-(benzo[d]thiazol-2-yl)-2-hydroxyquinoline-4-carboxamides as anticancer agents
|
Bindu, B. |
|
|
91 |
C |
p. |
article |
27 |
2,5-Disubstituted thiadiazoles as potent β-glucuronidase inhibitors; Synthesis, in vitro and in silico studies
|
Taha, Muhammad |
|
|
91 |
C |
p. |
article |
28 |
Editorial Board
|
|
|
|
91 |
C |
p. |
article |
29 |
Flavonols and 4-thioflavonols as potential acetylcholinesterase and butyrylcholinesterase inhibitors: Synthesis, structure-activity relationship and molecular docking studies
|
Mughal, Ehsan Ullah |
|
|
91 |
C |
p. |
article |
30 |
FtsZ inhibitors as a new genera of antibacterial agents
|
Tripathy, Swayansiddha |
|
|
91 |
C |
p. |
article |
31 |
Genetic dereplication of Trichoderma hypoxylon reveals two novel polycyclic lactones
|
Chen, Lin |
|
|
91 |
C |
p. |
article |
32 |
Identification of novel peptidomimetics targeting the polo-box domain of polo-like kinase 1
|
Li, Zhiyan |
|
|
91 |
C |
p. |
article |
33 |
Iizukines C−E from a saline soil fungus Aspergillus iizukae
|
Kang, Hui-Hui |
|
|
91 |
C |
p. |
article |
34 |
Issue TOC
|
|
|
|
91 |
C |
p. |
article |
35 |
Labeling of VEGFR1D2 through oxime ligation
|
De Rosa, Lucia |
|
|
91 |
C |
p. |
article |
36 |
Lysosome imaging in cancer cells by pyrene-benzothiazolium dyes: An alternative imaging approach for LAMP-1 expression based visualization methods to avoid background interference
|
Abeywickrama, Chathura S. |
|
|
91 |
C |
p. |
article |
37 |
Mechanistic studies on Pyrobaculum calidifontis porphobilinogen synthase (5-aminolevulinic acid dehydratase)
|
Azim, Naseema |
|
|
91 |
C |
p. |
article |
38 |
Multi-target 1,4-dihydropyridines showing calcium channel blockade and antioxidant capacity for Alzheimer’s disease therapy
|
Malek, Rim |
|
|
91 |
C |
p. |
article |
39 |
Natural neuroprotective alkaloids from Stephania japonica (Thunb.) Miers
|
Xiao, Jiao |
|
|
91 |
C |
p. |
article |
40 |
New classes of carbazoles as potential multi-functional anti-Alzheimer’s agents
|
Choubdar, Niloufar |
|
|
91 |
C |
p. |
article |
41 |
New hexalactone derivatives and a pair of new oxaspiro-carbon epimeric glycosides from the fruits of Illicium lanceolatum
|
Liu, Yang-Lan |
|
|
91 |
C |
p. |
article |
42 |
New phenolic cinnamic acid derivatives as selective COX-2 inhibitors. Design, synthesis, biological activity and structure-activity relationships
|
Ribeiro, Daniela |
|
|
91 |
C |
p. |
article |
43 |
Novel 2-aminopyridine liganded Pd(II) N-heterocyclic carbene complexes: Synthesis, characterization, crystal structure and bioactivity properties
|
Erdemir, Fatoş |
|
|
91 |
C |
p. |
article |
44 |
Novel steroidal 1,3,4-thiadiazines: Synthesis and biological evaluation in androgen receptor-positive prostate cancer 22Rv1 cells
|
Komendantova, Anna S. |
|
|
91 |
C |
p. |
article |
45 |
N-substituted noscapine derivatives as new antiprotozoal agents: Synthesis, antiparasitic activity and molecular docking study
|
Babanezhad Harikandei, Kosar |
|
|
91 |
C |
p. |
article |
46 |
One-step immobilization and purification of genetic engineering CBD fusion EndoS on cellulose for antibodies Fc-glycan remodeling
|
Zhao, Kai |
|
|
91 |
C |
p. |
article |
47 |
Optimization of a single HPLC-PDA method for quantifying Metformin, Gliclazide, Pioglitazone, Dapagliflozin, Empagliflozin, Saxagliptin, Linagliptin and Teneligliptin using central composite design
|
Kant, Ravi |
|
|
91 |
C |
p. |
article |
48 |
Phytoscreening of Vochysiaceae species: Molecular identification by HPLC-ESI-MS/MS and evaluating of their antioxidant activity and inhibitory potential against human α-amylase and protein glycation
|
Franco, R.R. |
|
|
91 |
C |
p. |
article |
49 |
Revealing synergistic mechanism of multiple components in Stauntonia brachyanthera Hand.-Mazz. for gout by virtual screening and system pharmacological approach
|
Hua, Qiong-qiong |
|
|
91 |
C |
p. |
article |
50 |
Searching new structural scaffolds for BRAF inhibitors. An integrative study using theoretical and experimental techniques
|
Campos, Ludmila E. |
|
|
91 |
C |
p. |
article |
51 |
Small molecule HDAC inhibitors: Promising agents for breast cancer treatment
|
Huang, Meiling |
|
|
91 |
C |
p. |
article |
52 |
Strategy and validation of a structure-based method for the discovery of selective inhibitors of PAK isoforms and the evaluation of their anti-cancer activity
|
Song, Pei-Lu |
|
|
91 |
C |
p. |
article |
53 |
Structural modifications and in vitro pharmacological evaluation of 4-pyridyl-piperazine derivatives as an active and selective histamine H3 receptor ligands
|
Szczepańska, Katarzyna |
|
|
91 |
C |
p. |
article |
54 |
1,8-Substituted anthraquinones, anthrones and bianthrones as potential non-azole leads against fungal infections
|
Jalab, Murhaf |
|
|
91 |
C |
p. |
article |
55 |
Sulfonamides incorporating piperazine bioisosteres as potent human carbonic anhydrase I, II, IV and IX inhibitors
|
Chiaramonte, Niccolò |
|
|
91 |
C |
p. |
article |
56 |
Synthesis and application of a “turn on” fluorescent probe for glutathione based on a copper complex of coumarin hydrazide Schiff base derivative
|
He, Guangjie |
|
|
91 |
C |
p. |
article |
57 |
Synthesis and biological evaluation of bergenin-1,2,3-triazole hybrids as novel class of anti-mitotic agents
|
Pavan Kumar, P. |
|
|
91 |
C |
p. |
article |
58 |
Synthesis, biological evaluation and molecular docking studies of bis-chalcone derivatives as xanthine oxidase inhibitors and anticancer agents
|
Burmaoglu, Serdar |
|
|
91 |
C |
p. |
article |
59 |
Synthesis, in silico and in vitro studies of new 1,4-dihydropiridine derivatives for antitumor and P-glycoprotein inhibitory activity
|
Mollazadeh, Shirin |
|
|
91 |
C |
p. |
article |
60 |
Synthesis, in-vitro α-glucosidase inhibition, antioxidant, in-vivo antidiabetic and molecular docking studies of pyrrolidine-2,5-dione and thiazolidine-2,4-dione derivatives
|
Hussain, Fida |
|
|
91 |
C |
p. |
article |
61 |
Synthesis, molecular docking analysis and carbonic anhydrase I-II inhibitory evaluation of new sulfonamide derivatives
|
Sağlık, Begüm Nurpelin |
|
|
91 |
C |
p. |
article |
62 |
Synthesis, molecular docking, and biological evaluation of 3-oxo-2-tolylhydrazinylidene-4,4,4-trifluorobutanoates bearing higher and natural alcohol moieties as new selective carboxylesterase inhibitors
|
Makhaeva, Galina F. |
|
|
91 |
C |
p. |
article |
63 |
Synthesis of 3-indolylmethyl substituted (pyrazolo/benzo)triazinone derivatives under Pd/Cu-catalysis: Identification of potent inhibitors of chorismate mutase (CM)
|
Reddy, Gangireddy Sujeevan |
|
|
91 |
C |
p. |
article |
64 |
Synthesis of new arylhydrazide bearing Schiff bases/thiazolidinone: α-Amylase, urease activities and their molecular docking studies
|
Rahim, Fazal |
|
|
91 |
C |
p. |
article |
65 |
Synthesis of novel methyl jasmonate derivatives and evaluation of their biological activity in various cancer cell lines
|
Sucu, Bilgesu Onur |
|
|
91 |
C |
p. |
article |
66 |
Synthesis of novel (R)-4-fluorophenyl-1H-1,2,3-triazoles: A new class of α-glucosidase inhibitors
|
Avula, Satya Kumar |
|
|
91 |
C |
p. |
article |
67 |
Synthesis, physicochemical and biological evaluation of tacrine derivative labeled with technetium-99m and gallium-68 as a prospective diagnostic tool for early diagnosis of Alzheimer’s disease
|
Gniazdowska, Ewa |
|
|
91 |
C |
p. |
article |
68 |
The 5-hydrazino-3-methylisothiazole-4-carboxylic acid, its new 5-substituted derivatives and their antiproliferative activity
|
Jęśkowiak, Izabela |
|
|
91 |
C |
p. |
article |
69 |
The influence of cationic dendrimers on antibacterial activity of phage endolysin against P. aeruginosa cells
|
Ciepluch, Karol |
|
|
91 |
C |
p. |
article |
70 |
The novel economical synthesis and antimicrobial activity of a trithiocarbonate derivative
|
Mabkhot, Yahia N. |
|
|
91 |
C |
p. |
article |
71 |
Thiohydantoin derivatives incorporating a pyrazole core: Design, synthesis and biological evaluation as dual inhibitors of topoisomerase-I and cycloxygenase-2 with anti-cancer and anti-inflammatory activities
|
Abdellatif, Khaled R.A. |
|
|
91 |
C |
p. |
article |
72 |
Three new cyclopiane-type diterpenes from a deep-sea derived fungus Penicillium sp. YPGA11 and their effects against human esophageal carcinoma cells
|
Cheng, Zhongbin |
|
|
91 |
C |
p. |
article |
73 |
Tyrosine-based asymmetric urea ligand for prostate carcinoma: Tuning biological efficacy through in silico studies
|
Sengupta, Sagnik |
|
|
91 |
C |
p. |
article |
74 |
Tyrosol from marine Fungi, a novel Quorum sensing inhibitor against Chromobacterium violaceum and Pseudomonas aeruginosa
|
Chang, Aiping |
|
|
91 |
C |
p. |
article |
75 |
Ugi efficient synthesis, biological evaluation and molecular docking of coumarin-quinoline hybrids as apoptotic agents through mitochondria-related pathways
|
Taheri, Salman |
|
|
91 |
C |
p. |
article |
76 |
Ureidobenzenesulfonamides as efficient inhibitors of carbonic anhydrase II
|
Serbian, Immo |
|
|
91 |
C |
p. |
article |
77 |
Utilization of tetrahydrobenzo[4,5]thieno[2,3-d]pyrimidinone as a cap moiety in design of novel histone deacetylase inhibitors
|
Mohamed, Mamdouh F.A. |
|
|
91 |
C |
p. |
article |
78 |
Water soluble thioglycosylated BODIPYs for mitochondria targeted cytotoxicity
|
Kesavan, Praseetha E. |
|
|
91 |
C |
p. |
article |