| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
A concise synthesis of 1,4-dihydro-[1,4]diazepine-5,7-dione, a novel 7-TM receptor ligand core structure with melanocortin receptor agonist activity
|
Szewczyk, Jerzy R.
|
|
2010
|
18 |
5 |
p. 1822-1833
12 p.
|
artikel
|
| 2 |
Acylated phenylethanoid oligoglycosides with hepatoprotective activity from the desert plant Cistanche tubulosa 1
|
Morikawa, Toshio
|
|
2010
|
18 |
5 |
p. 1882-1890
9 p.
|
artikel
|
| 3 |
Antifungal 3,5-disubstituted furanones: From 5-acyloxymethyl to 5-alkylidene derivatives
|
Šenel, Petr
|
|
2010
|
18 |
5 |
p. 1988-2000
13 p.
|
artikel
|
| 4 |
Benzyl 1,2,3,5,11,11a-hexahydro-3,3-dimethyl-1-oxo-6H-imidazo[3′,4′:1,2]pyridin[3,4-b]indole-2-substituted acetates: One-pot-preparation, anti-tumor activity, docking toward DNA and 3D QSAR analysis
|
Liu, Jiawang
|
|
2010
|
18 |
5 |
p. 1910-1917
8 p.
|
artikel
|
| 5 |
Biomimetic synthesis and anti-HIV activity of dimeric phloroglucinols
|
Chauthe, Siddheshwar K.
|
|
2010
|
18 |
5 |
p. 2029-2036
8 p.
|
artikel
|
| 6 |
Characterization of anticancer properties of 2,6-diisopropylphenol–docosahexaenoate and analogues in breast cancer cells
|
Harvey, Kevin A.
|
|
2010
|
18 |
5 |
p. 1866-1874
9 p.
|
artikel
|
| 7 |
Colony stimulating factor-1 receptor as a target for small molecule inhibitors
|
Mashkani, Baratali
|
|
2010
|
18 |
5 |
p. 1789-1797
9 p.
|
artikel
|
| 8 |
Conservative secondary structure motif of streptavidin-binding aptamers generated by different laboratories
|
Bing, Tao
|
|
2010
|
18 |
5 |
p. 1798-1805
8 p.
|
artikel
|
| 9 |
Cytotoxic and anti-inflammatory cembranoids from the Dongsha Atoll soft coral Sarcophyton crassocaule
|
Lin, Wan-Yu
|
|
2010
|
18 |
5 |
p. 1936-1941
6 p.
|
artikel
|
| 10 |
Design, asymmetric synthesis, and evaluation of pseudosymmetric sulfoximine inhibitors against HIV-1 protease
|
Lu, Ding
|
|
2010
|
18 |
5 |
p. 2037-2048
12 p.
|
artikel
|
| 11 |
Design, synthesis and antimicrobial properties of non-hemolytic cationic α-cyclopeptoids
|
Comegna, Daniela
|
|
2010
|
18 |
5 |
p. 2010-2018
9 p.
|
artikel
|
| 12 |
Design, synthesis, and biological evaluation of novel water-soluble triptolide derivatives: Antineoplastic activity against imatinib-resistant CML cells bearing T315I mutant Bcr-Abl
|
Xu, Fang
|
|
2010
|
18 |
5 |
p. 1806-1815
10 p.
|
artikel
|
| 13 |
Design, synthesis and preliminary activity assay of 1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid derivatives as novel Histone deacetylases (HDACs) inhibitors
|
Zhang, Yingjie
|
|
2010
|
18 |
5 |
p. 1761-1772
12 p.
|
artikel
|
| 14 |
Design, synthesis, and preliminary pharmacological evaluation of new imidazolinones as l-DOPA prodrugs
|
Giorgioni, Gianfabio
|
|
2010
|
18 |
5 |
p. 1834-1843
10 p.
|
artikel
|
| 15 |
Development of selective and reversible pyrazoline based MAO-A inhibitors: Synthesis, biological evaluation and docking studies
|
Karuppasamy, Muthukumar
|
|
2010
|
18 |
5 |
p. 1875-1881
7 p.
|
artikel
|
| 16 |
Discovery of potent sulfonamide P4-capped ketoamide second generation inhibitors of hepatitis C virus NS3 serine protease with favorable pharmacokinetic profiles in preclinical species
|
Bogen, Stéphane L.
|
|
2010
|
18 |
5 |
p. 1854-1865
12 p.
|
artikel
|
| 17 |
Editorial board
|
|
|
2010
|
18 |
5 |
p. IFC-
1 p.
|
artikel
|
| 18 |
Exploring a synthetic organoselenium compound for antioxidant pharmacotherapy—toxicity and effects on ROS-production
|
Johansson, Henrik
|
|
2010
|
18 |
5 |
p. 1783-1788
6 p.
|
artikel
|
| 19 |
Graphical contents list
|
|
|
2010
|
18 |
5 |
p. 1739-1748
10 p.
|
artikel
|
| 20 |
Insight into the strong inhibitory action of salt on activity of neocarzinostatin
|
Chin, Der-Hang
|
|
2010
|
18 |
5 |
p. 1980-1987
8 p.
|
artikel
|
| 21 |
Interaction of (benzylidene-hydrazono)-1,4-dihydropyridines with β-amyloid, acetylcholine, and butyrylcholine esterases
|
Alptüzün, Vildan
|
|
2010
|
18 |
5 |
p. 2049-2059
11 p.
|
artikel
|
| 22 |
Novel thiophene derivatives as PTP1B inhibitors with selectivity and cellular activity
|
Ye, Deju
|
|
2010
|
18 |
5 |
p. 1773-1782
10 p.
|
artikel
|
| 23 |
Optimization of 6,6-dimethyl pyrrolo[3,4-c]pyrazoles: Identification of PHA-793887, a potent CDK inhibitor suitable for intravenous dosing
|
Brasca, Maria Gabriella
|
|
2010
|
18 |
5 |
p. 1844-1853
10 p.
|
artikel
|
| 24 |
S-Arachidonoyl-2-thioglycerol synthesis and use for fluorimetric and colorimetric assays of monoacylglycerol lipase
|
Casida, John E.
|
|
2010
|
18 |
5 |
p. 1942-1947
6 p.
|
artikel
|
| 25 |
SAR studies on new bis-aryls 5-HT7 ligands: Synthesis and molecular modeling
|
Badarau, Eduard
|
|
2010
|
18 |
5 |
p. 1958-1967
10 p.
|
artikel
|
| 26 |
Searching for multi-target antipsychotics: Discovery of orally active heterocyclic N-phenylpiperazine ligands of D2-like and 5-HT1A receptors
|
Neves, Gilda
|
|
2010
|
18 |
5 |
p. 1925-1935
11 p.
|
artikel
|
| 27 |
Selective benzimidazole inhibitors of the antigen receptor-mediated NF-κB activation pathway
|
Okolotowicz, Karl J.
|
|
2010
|
18 |
5 |
p. 1918-1924
7 p.
|
artikel
|
| 28 |
Synthesis and antiproliferative evaluation of certain indolo[3,2-c]quinoline derivatives
|
Lu, Chih-Ming
|
|
2010
|
18 |
5 |
p. 1948-1957
10 p.
|
artikel
|
| 29 |
Synthesis and biological evaluation of novel pyrazolyl-2,4-thiazolidinediones as anti-inflammatory and neuroprotective agents
|
Youssef, Amal M.
|
|
2010
|
18 |
5 |
p. 2019-2028
10 p.
|
artikel
|
| 30 |
Synthesis and biological screening of a combinatorial library of β-chlorovinyl chalcones as anticancer, anti-inflammatory and antimicrobial agents
|
Bandgar, Babasaheb P.
|
|
2010
|
18 |
5 |
p. 2060-2065
6 p.
|
artikel
|
| 31 |
Synthesis and characterization of novel 1,2,4-triazine derivatives with antiproliferative activity
|
Krauth, Fabian
|
|
2010
|
18 |
5 |
p. 1816-1821
6 p.
|
artikel
|
| 32 |
Synthesis and evaluation of 1,4-diphenylbutadiene derivatives as inhibitors of plasminogen activator inhibitor-1 (PAI-1) production
|
Miyazaki, Hiroshi
|
|
2010
|
18 |
5 |
p. 1968-1979
12 p.
|
artikel
|
| 33 |
Synthesis and pharmacological evaluation of novel 1,3,8- and 1,3,7,8-substituted xanthines as adenosine receptor antagonists
|
Rodríguez-Borges, José Enrique
|
|
2010
|
18 |
5 |
p. 2001-2009
9 p.
|
artikel
|
| 34 |
Synthesis, in vitro progesterone receptors affinity of gadolinium containing mifepristone conjugates and estimation of binding sites in human breast cancer cells
|
Saha, Pijus
|
|
2010
|
18 |
5 |
p. 1891-1898
8 p.
|
artikel
|
| 35 |
Synthesis, metabolism and in vitro cytotoxicity studies on novel lavendamycin antitumor agents
|
Cai, Wen
|
|
2010
|
18 |
5 |
p. 1899-1909
11 p.
|
artikel
|
| 36 |
Targeting Alzheimer’s disease: Novel indanone hybrids bearing a pharmacophoric fragment of AP2238
|
Rizzo, Stefano
|
|
2010
|
18 |
5 |
p. 1749-1760
12 p.
|
artikel
|
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