nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
1 |
Affinity of aporphines for the human 5-HT2A receptor: Insights from homology modeling and molecular docking studies
|
Pecic, Stevan |
|
2010 |
18 |
15 |
p. 5562-5575 14 p. |
artikel |
2 |
1-Azaaurones derived from the naturally occurring aurones as potential antimalarial drugs
|
Souard, Florence |
|
2010 |
18 |
15 |
p. 5724-5731 8 p. |
artikel |
3 |
Baculiferins A–O, O-sulfated pyrrole alkaloids with anti-HIV-1 activity, from the Chinese marine sponge Iotrochota baculifera
|
Fan, Guotao |
|
2010 |
18 |
15 |
p. 5466-5474 9 p. |
artikel |
4 |
Benzo[b]thiophene-6-carboxamide 1,1-dioxides: Inhibitors of human cancer cell growth at nanomolar concentrations
|
Sagardoy, Aitziber A. |
|
2010 |
18 |
15 |
p. 5701-5707 7 p. |
artikel |
5 |
Comparison of demetalation properties between zinc chlorin and zinc porphyrin derivatives: Effect of macrocyclic structures
|
Saga, Yoshitaka |
|
2010 |
18 |
15 |
p. 5697-5700 4 p. |
artikel |
6 |
Conjugating folic acid to gold nanoparticles through glutathione for targeting and detecting cancer cells
|
Zhang, Zhaowu |
|
2010 |
18 |
15 |
p. 5528-5534 7 p. |
artikel |
7 |
Dual-target-directed 1,3-diphenylurea derivatives: BACE 1 inhibitor and metal chelator against Alzheimer’s disease
|
Huang, Wenhai |
|
2010 |
18 |
15 |
p. 5610-5615 6 p. |
artikel |
8 |
Editorial board
|
|
|
2010 |
18 |
15 |
p. IFC- 1 p. |
artikel |
9 |
Efficient synthesis of Hsp90 inhibitor dimers as potential antitumor agents
|
Sekiguchi, Hironori |
|
2010 |
18 |
15 |
p. 5732-5737 6 p. |
artikel |
10 |
Elucidation of the topography of the thapsigargin binding site in the sarco-endoplasmic calcium ATPase
|
Skytte, Dorthe Mondrup |
|
2010 |
18 |
15 |
p. 5634-5646 13 p. |
artikel |
11 |
Further delineation of hydrophobic binding sites in dopamine D2/D3 receptors for N-4 substituents on the piperazine ring of the hybrid template 5/7-{[2-(4-aryl-piperazin-1-yl)-ethyl]-propyl-amino}-5,6,7,8-tetrahydro-naphthalen-2-ol
|
Ghosh, Balaram |
|
2010 |
18 |
15 |
p. 5661-5674 14 p. |
artikel |
12 |
Genomic action of permanently charged tamoxifen derivatives via estrogen receptor-α
|
Rivera-Guevara, Claudia |
|
2010 |
18 |
15 |
p. 5593-5601 9 p. |
artikel |
13 |
Graphical contents list
|
|
|
2010 |
18 |
15 |
p. 5457-5465 9 p. |
artikel |
14 |
Identification of a potent and noncytotoxic inhibitor of melanin production
|
Hwang, Soonho |
|
2010 |
18 |
15 |
p. 5602-5609 8 p. |
artikel |
15 |
Investigations on the 2-thiazolylhydrazyne scaffold: Synthesis and molecular modeling of selective human monoamine oxidase inhibitors
|
Chimenti, Franco |
|
2010 |
18 |
15 |
p. 5715-5723 9 p. |
artikel |
16 |
Mutation of Phe91 to Asn in human carbonic anhydrase I unexpectedly enhanced both catalytic activity and affinity for sulfonamide inhibitors
|
Kockar, Feray |
|
2010 |
18 |
15 |
p. 5498-5503 6 p. |
artikel |
17 |
New chloro,fluorobenzylindole derivatives as integrase strand-transfer inhibitors (INSTIs) and their mode of action
|
Ferro, Stefania |
|
2010 |
18 |
15 |
p. 5510-5518 9 p. |
artikel |
18 |
Nε -Modified lysine containing inhibitors for SIRT1 and SIRT2
|
Huhtiniemi, Tero |
|
2010 |
18 |
15 |
p. 5616-5625 10 p. |
artikel |
19 |
Pharmacophore identification, synthesis, and biological evaluation of carboxylated chalcone derivatives as CysLT1 antagonists
|
Dong, Xiaowu |
|
2010 |
18 |
15 |
p. 5519-5527 9 p. |
artikel |
20 |
Photoaffinity labeling of Ras converting enzyme 1 (Rce1p) using a benzophenone-containing peptide substrate
|
Kyro, Kelly |
|
2010 |
18 |
15 |
p. 5675-5684 10 p. |
artikel |
21 |
Pyridazinopsoralens of wide chemotherapeutic interest
|
Dalla Via, Lisa |
|
2010 |
18 |
15 |
p. 5708-5714 7 p. |
artikel |
22 |
Rational conversion of noncontinuous active region in proteins into a small orally bioavailable macrocyclic drug-like molecule: The HIV-1 CD4:gp120 paradigm
|
Hurevich, Mattan |
|
2010 |
18 |
15 |
p. 5754-5761 8 p. |
artikel |
23 |
Substrate specificity and inhibitory study of human airway trypsin-like protease
|
Wysocka, M. |
|
2010 |
18 |
15 |
p. 5504-5509 6 p. |
artikel |
24 |
Synthesis and biological evaluation of arylidene analogues of Meldrum’s acid as a new class of antimalarial and antioxidant agents
|
Sandhu, Harmeet S. |
|
2010 |
18 |
15 |
p. 5626-5633 8 p. |
artikel |
25 |
Synthesis and biological evaluation of naphthoquinone analogs as a novel class of proteasome inhibitors
|
Lawrence, Harshani R. |
|
2010 |
18 |
15 |
p. 5576-5592 17 p. |
artikel |
26 |
Synthesis and biological evaluation of novel pyrazole compounds
|
Youssef, Amal M. |
|
2010 |
18 |
15 |
p. 5685-5696 12 p. |
artikel |
27 |
Synthesis and characterization of a triazine dendrimer that sequesters iron(III) using 12 desferrioxamine B groups
|
Lim, Jongdoo |
|
2010 |
18 |
15 |
p. 5749-5753 5 p. |
artikel |
28 |
Synthesis and in vivo evaluation of [11C]tariquidar, a positron emission tomography radiotracer based on a third-generation P-glycoprotein inhibitor
|
Bauer, Florian |
|
2010 |
18 |
15 |
p. 5489-5497 9 p. |
artikel |
29 |
Synthesis and pharmacology of 1-methoxy analogs of CP-47,497
|
Huffman, John W. |
|
2010 |
18 |
15 |
p. 5475-5482 8 p. |
artikel |
30 |
Synthesis, binding and bioactivity of γ-methylene γ-lactam ecdysone receptor ligands: Advantages of QSAR models for flexible receptors
|
Birru, Woldeamanuel |
|
2010 |
18 |
15 |
p. 5647-5660 14 p. |
artikel |
31 |
Targeting the ICB2 site of the topoisomerase IIα promoter with a formamido-pyrrole–imidazole–pyrrole H-pin polyamide
|
Franks, Andrew |
|
2010 |
18 |
15 |
p. 5553-5561 9 p. |
artikel |
32 |
The design, synthesis, and evaluation of 8 hybrid DFG-out allosteric kinase inhibitors: A structural analysis of the binding interactions of Gleevec®, Nexavar®, and BIRB-796
|
Dietrich, Justin |
|
2010 |
18 |
15 |
p. 5738-5748 11 p. |
artikel |
33 |
The peptide hormone ghrelin binds to membrane-mimetics via its octanoyl chain and an adjacent phenylalanine
|
Großauer, Jörg |
|
2010 |
18 |
15 |
p. 5483-5488 6 p. |
artikel |
34 |
The structure–activity relationships of A-ring-substituted aromathecin topoisomerase I inhibitors strongly support a camptothecin-like binding mode
|
Cinelli, Maris A. |
|
2010 |
18 |
15 |
p. 5535-5552 18 p. |
artikel |