nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
1 |
Activity profile relationships between structurally similar promiscuous compounds
|
Hu, Ye |
|
2013 |
69 |
C |
p. 393-398 6 p. |
artikel |
2 |
Aggrecanase-2 inhibitors based on the acylthiosemicarbazide zinc-binding group
|
Maingot, Lucie |
|
2013 |
69 |
C |
p. 244-261 18 p. |
artikel |
3 |
A novel [1,2,4] triazolo [1,5-a] pyrimidine-based phenyl-linked steroid dimer: Synthesis and its cytotoxic activity
|
Yu, Bin |
|
2013 |
69 |
C |
p. 323-330 8 p. |
artikel |
4 |
Anticancer evaluation of some newly synthesized N-nicotinonitrile derivative
|
Shamroukh, Ahmed H. |
|
2013 |
69 |
C |
p. 521-526 6 p. |
artikel |
5 |
Biological activity of neutral and cationic iridium(III) complexes with κP and κP,κS coordinated Ph2PCH2S(O) x Ph (x = 0–2) ligands
|
Ludwig, Gerd |
|
2013 |
69 |
C |
p. 216-222 7 p. |
artikel |
6 |
3-(3-Butylamino-2-hydroxy-propoxy)-1-hydroxy-xanthen-9-one acts as a topoisomerase IIα catalytic inhibitor with low DNA damage
|
Park, So-Eun |
|
2013 |
69 |
C |
p. 139-145 7 p. |
artikel |
7 |
Carbonic anhydrase inhibitors. Synthesis of heterocyclic 4-substituted pyridine-3-sulfonamide derivatives and their inhibition of the human cytosolic isozymes I and II and transmembrane tumor-associated isozymes IX and XII
|
Sławiński, Jarosław |
|
2013 |
69 |
C |
p. 701-710 10 p. |
artikel |
8 |
cis-Dichloroplatinum(II) complexes tethered to dibenzo[c,h][1,6]naphthyridin-6-ones: Synthesis and cytotoxicity in human cancer cell lines in vitro
|
Desbois, Nicolas |
|
2013 |
69 |
C |
p. 719-727 9 p. |
artikel |
9 |
Design and application of a rigid quinazolone scaffold based on two-face Bim α-helix mimicking
|
Zhang, Zhichao |
|
2013 |
69 |
C |
p. 711-718 8 p. |
artikel |
10 |
Design, syntheses, and characterization of pharmacophore based chemokine receptor CCR5 antagonists as anti prostate cancer agents
|
Arnatt, Christopher K. |
|
2013 |
69 |
C |
p. 647-658 12 p. |
artikel |
11 |
Design, synthesis and biological activities of some 7-aminocephalosporanic acid derivatives
|
Basoglu, Serap |
|
2013 |
69 |
C |
p. 622-631 10 p. |
artikel |
12 |
Design, synthesis and biological evaluation of a novel class of potent TGR5 agonists based on a 4-phenyl pyridine scaffold
|
Zhu, Junjie |
|
2013 |
69 |
C |
p. 55-68 14 p. |
artikel |
13 |
Design, synthesis, and biological evaluation of novel 2-ethyl-5-phenylthiazole-4-carboxamide derivatives as protein tyrosine phosphatase 1B inhibitors with improved cellular efficacy
|
Chen, Yue-Ting |
|
2013 |
69 |
C |
p. 399-412 14 p. |
artikel |
14 |
Design, synthesis and biological evaluation of 2-substituted quinolines as potential antileishmanial agents
|
Gopinath, Vadiraj S. |
|
2013 |
69 |
C |
p. 527-536 10 p. |
artikel |
15 |
Design, synthesis and biological evaluation of WC-9 analogs as antiparasitic agents
|
Elicio, Pablo D. |
|
2013 |
69 |
C |
p. 480-489 10 p. |
artikel |
16 |
Design, synthesis and efficacy of novel G protein-coupled receptor kinase 2 inhibitors
|
Carotenuto, Alfonso |
|
2013 |
69 |
C |
p. 384-392 9 p. |
artikel |
17 |
Design, synthesis, and in vitro cancer cell growth inhibition evaluation and antimalarial testing of trioxanes installed in cyclic 2-enoate substructures
|
Hossain, Md. Imran |
|
2013 |
69 |
C |
p. 294-309 16 p. |
artikel |
18 |
Design, synthesis and structure–activity relationship of novel quinoxaline derivatives as cancer chemopreventive agent by inhibition of tyrosine kinase receptor
|
Galal, Shadia A. |
|
2013 |
69 |
C |
p. 115-124 10 p. |
artikel |
19 |
Design, synthesis, and structure–activity relationships of novel 6,7-disubstituted-4-phenoxyquinoline derivatives as potential antitumor agents
|
Tang, Qidong |
|
2013 |
69 |
C |
p. 77-89 13 p. |
artikel |
20 |
Development of 3,4-dihydroisoquinolin-1(2H)-one derivatives for the Positron Emission Tomography (PET) imaging of σ2 receptors
|
Abate, Carmen |
|
2013 |
69 |
C |
p. 920-930 11 p. |
artikel |
21 |
Development of 3-phenyl-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridine derivatives as novel Mycobacterium tuberculosis pantothenate synthetase inhibitors
|
Samala, Ganesh |
|
2013 |
69 |
C |
p. 356-364 9 p. |
artikel |
22 |
Discovery of 4-amino-2-(thio)phenol derivatives as novel protein kinase and angiogenesis inhibitors for the treatment of cancer: Synthesis and biological evaluation. Part II
|
Xu, Fuming |
|
2013 |
69 |
C |
p. 191-200 10 p. |
artikel |
23 |
Discovery of a potent dual EGFR/HER-2 inhibitor L-2 (selatinib) for the treatment of cancer
|
Zhang, Long |
|
2013 |
69 |
C |
p. 833-841 9 p. |
artikel |
24 |
Editorial board
|
|
|
2013 |
69 |
C |
p. IFC- 1 p. |
artikel |
25 |
Experimental and molecular modeling studies on the interaction of the Ru(II)-piroxicam with DNA and BSA
|
Jannesari, Zahra |
|
2013 |
69 |
C |
p. 577-590 14 p. |
artikel |
26 |
Flavones as isosteres of 4(1H)-quinolones: Discovery of ligand efficient and dual stage antimalarial lead compounds
|
Rodrigues, Tiago |
|
2013 |
69 |
C |
p. 872-880 9 p. |
artikel |
27 |
Graphical contents list
|
|
|
2013 |
69 |
C |
p. iii-xxv nvt p. |
artikel |
28 |
2-Heteroarylimino-5-arylidene-4-thiazolidinones as a new class of non-nucleoside inhibitors of HCV NS5B polymerase
|
Küçükgüzel, İlkay |
|
2013 |
69 |
C |
p. 931-941 11 p. |
artikel |
29 |
2-(2-Hydrazinyl)thiazole derivatives: Design, synthesis and in vitro antimycobacterial studies
|
Makam, Parameshwar |
|
2013 |
69 |
C |
p. 564-576 13 p. |
artikel |
30 |
Identification and characterization of novel indole based small molecules as anticancer agents through SIRT1 inhibition
|
Panathur, Naveen |
|
2013 |
69 |
C |
p. 125-138 14 p. |
artikel |
31 |
Indenoindoles and cyclopentacarbazoles as bioactive compounds: Synthesis and biological applications
|
Rongved, Pal |
|
2013 |
69 |
C |
p. 465-479 15 p. |
artikel |
32 |
In vitro antimalarial activity, β-haematin inhibition and structure–activity relationships in a series of quinoline triazoles
|
Joshi, Mukesh C. |
|
2013 |
69 |
C |
p. 338-347 10 p. |
artikel |
33 |
β-Ionone derived chalcones as potent antiproliferative agents
|
Sharma, Vishal |
|
2013 |
69 |
C |
p. 310-315 6 p. |
artikel |
34 |
Isoxazole derivatives as potent transient receptor potential melastatin type 8 (TRPM8) agonists
|
Ostacolo, Carmine |
|
2013 |
69 |
C |
p. 659-669 11 p. |
artikel |
35 |
Mastering tricyclic ring systems for desirable functional cannabinoid activity
|
Petrov, Ravil R. |
|
2013 |
69 |
C |
p. 881-907 27 p. |
artikel |
36 |
Microwave assisted synthesis of dihydrobenzo[4,5]imidazo[1,2-a]pyrimidin-4-ones; synthesis, in vitro antimicrobial and anticancer activities of novel coumarin substituted dihydrobenzo[4,5]imidazo[1,2-a]pyrimidin-4-ones
|
Puttaraju, Kallimeledoddi B. |
|
2013 |
69 |
C |
p. 316-322 7 p. |
artikel |
37 |
Modulation of A2B adenosine receptor by 1-Benzyl-3-ketoindole derivatives
|
Taliani, Sabrina |
|
2013 |
69 |
C |
p. 331-337 7 p. |
artikel |
38 |
Monoamine oxidase inhibitory activity of 3,5-biaryl-4,5-dihydro-1H-pyrazole-1-carboxylate derivatives
|
Vishnu Nayak, B. |
|
2013 |
69 |
C |
p. 762-767 6 p. |
artikel |
39 |
Multifunctional tacrine–flavonoid hybrids with cholinergic, β-amyloid-reducing, and metal chelating properties for the treatment of Alzheimer's disease
|
Li, Su-Yi |
|
2013 |
69 |
C |
p. 632-646 15 p. |
artikel |
40 |
New combination of pharmacophoric elements of potent σ 1 ligands: Design, synthesis and σ receptor affinity of aminoethyl substituted tetrahydrobenzothiophenes
|
Harel, Dipak |
|
2013 |
69 |
C |
p. 490-497 8 p. |
artikel |
41 |
New di(hetero)arylethers and di(hetero)arylamines in the thieno[3,2-b]pyridine series: Synthesis, growth inhibitory activity on human tumor cell lines and non-tumor cells, effects on cell cycle and on programmed cell death
|
Queiroz, Maria-João R.P. |
|
2013 |
69 |
C |
p. 855-862 8 p. |
artikel |
42 |
New orally effective 3-(2-nitro)phenylpropanamide analgesic derivatives: Synthesis and antinociceptive evaluation
|
Since, Marc |
|
2013 |
69 |
C |
p. 728-734 7 p. |
artikel |
43 |
New synthetic aliphatic sulfonamido-quaternary ammonium salts as anticancer chemotherapeutic agents
|
Song, Doona |
|
2013 |
69 |
C |
p. 670-677 8 p. |
artikel |
44 |
Nonpeptidic angiotensin II AT1 receptor antagonists derived from 6-substituted aminocarbonyl and acylamino benzimidazoles
|
Zhang, Jun |
|
2013 |
69 |
C |
p. 44-54 11 p. |
artikel |
45 |
Novel acetamidothiazole derivatives: Synthesis and in vitro anticancer evaluation
|
Ali, Ahmed R. |
|
2013 |
69 |
C |
p. 908-919 12 p. |
artikel |
46 |
Novel 6β-acylaminomorphinans with analgesic activity
|
Váradi, András |
|
2013 |
69 |
C |
p. 786-789 4 p. |
artikel |
47 |
Novel heterocyclic-fused pyrimidine derivatives: Synthesis, molecular modeling and pharmacological screening
|
Arafa, Reem K. |
|
2013 |
69 |
C |
p. 498-507 10 p. |
artikel |
48 |
Novel N-methylsulfonamide and retro-N-methylsulfonamide derivatives as 17β-hydroxysteroid dehydrogenase type 2 (17β-HSD2) inhibitors with good ADME-related physicochemical parameters
|
Perspicace, Enrico |
|
2013 |
69 |
C |
p. 201-215 15 p. |
artikel |
49 |
Novel nonsecosteroidal VDR agonists with phenyl-pyrrolyl pentane skeleton
|
Shen, Wei |
|
2013 |
69 |
C |
p. 768-778 11 p. |
artikel |
50 |
Novel N-4-piperazinyl-ciprofloxacin-chalcone hybrids: Synthesis, physicochemical properties, anticancer and topoisomerase I and II inhibitory activity
|
Abdel-Aziz, Mohamed |
|
2013 |
69 |
C |
p. 427-438 12 p. |
artikel |
51 |
Novel promising linezolid analogues: Rational design, synthesis and biological evaluation
|
De Rosa, Margherita |
|
2013 |
69 |
C |
p. 779-785 7 p. |
artikel |
52 |
PAMAM dendrimer derivatives as a potential drug for antithrombotic therapy
|
Durán-Lara, Esteban |
|
2013 |
69 |
C |
p. 601-608 8 p. |
artikel |
53 |
Platinum(II) complexes with N-monoalkyl 1R,2R-diaminocyclohexane derivatives as carrier ligands and 3-hydroxycyclobutane-1,1-dicarboxylate as a leaving group: Potent cytotoxicity and DNA binding ability
|
Fang, Lei |
|
2013 |
69 |
C |
p. 842-847 6 p. |
artikel |
54 |
Preparation and biological evaluation of 99mTc-N4IPA for single photon emission computerized tomography imaging of hypoxia in mouse tumor
|
Li, Nan |
|
2013 |
69 |
C |
p. 223-231 9 p. |
artikel |
55 |
Pyranoxanthones: Synthesis, growth inhibitory activity on human tumor cell lines and determination of their lipophilicity in two membrane models
|
Azevedo, Carlos M.G. |
|
2013 |
69 |
C |
p. 798-816 19 p. |
artikel |
56 |
Pyrazole containing natural products: Synthetic preview and biological significance
|
Kumar, Vinod |
|
2013 |
69 |
C |
p. 735-753 19 p. |
artikel |
57 |
QSAR modeling of aromatase inhibitory activity of 1-substituted 1,2,3-triazole analogs of letrozole
|
Nantasenamat, Chanin |
|
2013 |
69 |
C |
p. 99-114 16 p. |
artikel |
58 |
Squaric acid/4-aminoquinoline conjugates: Novel potent antiplasmodial agents
|
Ribeiro, Carlos J.A. |
|
2013 |
69 |
C |
p. 365-372 8 p. |
artikel |
59 |
Structure-based design, synthesis and biological evaluation of novel anthra[1,2-d]imidazole-6,11-dione homologues as potential antitumor agents
|
Chen, Tsung-Chih |
|
2013 |
69 |
C |
p. 278-293 16 p. |
artikel |
60 |
Synthesis and allosteric modulation of the dopamine receptor by peptide analogs of l-prolyl-l-leucyl-glycinamide (PLG) modified in the l-proline or l-proline and l-leucine scaffolds
|
Ferreira da Costa, Joana |
|
2013 |
69 |
C |
p. 146-158 13 p. |
artikel |
61 |
Synthesis and antibacterial activity of novel modified 5-O-mycaminose 14-membered ketolides
|
Xu, Yanpeng |
|
2013 |
69 |
C |
p. 174-181 8 p. |
artikel |
62 |
Synthesis and anticancer activity of some novel 2-phenazinamine derivatives
|
Gao, Xiaochun |
|
2013 |
69 |
C |
p. 1-9 9 p. |
artikel |
63 |
Synthesis and anticancer activity of some novel trifluoromethylquinolines carrying a biologically active benzenesulfonamide moiety
|
Al-Dosari, Mohammed S. |
|
2013 |
69 |
C |
p. 373-383 11 p. |
artikel |
64 |
Synthesis and antiproliferative activity of benzofuran-based analogs of cercosporamide against non-small cell lung cancer cell lines
|
Bazin, Marc-Antoine |
|
2013 |
69 |
C |
p. 823-832 10 p. |
artikel |
65 |
Synthesis and antitumor activities of novel thiourea α-aminophosphonates from dehydroabietic acid
|
Huang, Xiao-Chao |
|
2013 |
69 |
C |
p. 508-520 13 p. |
artikel |
66 |
Synthesis and antiviral activity of a novel class of (5-oxazolyl)phenyl amines
|
Zhong, Zhao-Jin |
|
2013 |
69 |
C |
p. 32-43 12 p. |
artikel |
67 |
Synthesis and biological activity of mycophenolic acid-amino acid derivatives
|
Iwaszkiewicz-Grzes, Dorota |
|
2013 |
69 |
C |
p. 863-871 9 p. |
artikel |
68 |
Synthesis and biological evaluation of novel delta (δ) opioid receptor ligands with diazatricyclodecane skeletons
|
Loriga, Giovanni |
|
2013 |
69 |
C |
p. 413-426 14 p. |
artikel |
69 |
Synthesis and biological evaluation of phenyl substituted polyoxygenated xanthone derivatives as anti-hepatoma agents
|
Dai, Ming |
|
2013 |
69 |
C |
p. 159-166 8 p. |
artikel |
70 |
Synthesis and cytotoxic activity of some novel steroidal C-17 pyrazolinyl derivatives
|
Fan, Ning-Juan |
|
2013 |
69 |
C |
p. 182-190 9 p. |
artikel |
71 |
Synthesis and evaluation of α-ketotriazoles and α,β-diketotriazoles as inhibitors of Mycobacterium tuberculosis
|
Menendez, Christophe |
|
2013 |
69 |
C |
p. 167-173 7 p. |
artikel |
72 |
Synthesis and evaluation of (Z)-2,3-diphenylacrylonitrile analogs as anti-cancer and anti-microbial agents
|
Alam, Mohammad Sayed |
|
2013 |
69 |
C |
p. 790-797 8 p. |
artikel |
73 |
Synthesis and in vitro and in vivo evaluation of antimalarial polyamines
|
Liew, Lydia P.P. |
|
2013 |
69 |
C |
p. 22-31 10 p. |
artikel |
74 |
Synthesis and in vitro/in vivo antibacterial activity of oxazolidinones having thiocarbamate at C-5 on the A-ring and an amide- or urea-substituted [1,2,5]triazepane or [1,2,5]oxadiazepane as the C-ring
|
Suzuki, Hideyuki |
|
2013 |
69 |
C |
p. 262-277 16 p. |
artikel |
75 |
Synthesis and SAR study of novel 3,3-diphenyl-1,3-dihydroindol-2-one derivatives as potent eIF2·GTP·Met-tRNAi Met ternary complex inhibitors
|
Denoyelle, Séverine |
|
2013 |
69 |
C |
p. 537-553 17 p. |
artikel |
76 |
Synthesis, antibacterial and antioxidant activities of new 1-alkyl-4-(1-alkyl-4-oxo-1,4-dihydroquinolin-2-yl)pyridinium bromides
|
Kahriman, Nuran |
|
2013 |
69 |
C |
p. 348-355 8 p. |
artikel |
77 |
Synthesis, antimicrobial, antioxidant activities of novel 6-aryl-5-cyano thiouracil derivatives
|
Mohamed, M.S. |
|
2013 |
69 |
C |
p. 591-600 10 p. |
artikel |
78 |
Synthesis, characterization, antiparasitic and cytotoxic evaluation of thioureas conjugated to polyamine scaffolds
|
Stringer, Tameryn |
|
2013 |
69 |
C |
p. 90-98 9 p. |
artikel |
79 |
Synthesis, cytotoxicity and DNA binding of oxoazabenzo[de]anthracenes derivatives in colon cancer Caco-2 cells
|
Di Salvo, Alberto |
|
2013 |
69 |
C |
p. 754-761 8 p. |
artikel |
80 |
Synthesis, hypoglycemic activity and molecular modeling studies of pyrazole-3-carbohydrazides designed by a CoMFA model
|
Hernández-Vázquez, Eduardo |
|
2013 |
69 |
C |
p. 10-21 12 p. |
artikel |
81 |
Synthesis of conformationally constrained γ-d-glutamyl-meso-diaminopimelic acid derivatives as ligands of nucleotide-binding oligomerization domain protein 1 (Nod1)
|
Jakopin, Žiga |
|
2013 |
69 |
C |
p. 232-243 12 p. |
artikel |
82 |
Synthesis of lipoic acid–peptide conjugates and their effect on collagen and melanogenesis
|
Lu, Chichong |
|
2013 |
69 |
C |
p. 449-454 6 p. |
artikel |
83 |
Synthesis of new andrographolide derivatives and evaluation of their antidyslipidemic, LDL-oxidation and antioxidant activity
|
Pandeti, Sukanya |
|
2013 |
69 |
C |
p. 439-448 10 p. |
artikel |
84 |
Synthesis of novel benzo[4,5]thiazolo[1,2-a]pyrimidine-3-carboxylate derivatives and biological evaluation as potential anticancer agents
|
Nagarapu, Lingaiah |
|
2013 |
69 |
C |
p. 817-822 6 p. |
artikel |
85 |
Synthesis of pyrido[2,1-a]isoquinolin-4-ones and oxazino[2,3-a]isoquinolin-4-ones: New inhibitors of mitochondrial respiratory chain
|
Moreno, Laura |
|
2013 |
69 |
C |
p. 69-76 8 p. |
artikel |
86 |
Synthesis of quinoidal molecules: Strategies towards bioactive compounds with an emphasis on lapachones
|
de Castro, Solange L. |
|
2013 |
69 |
C |
p. 678-700 23 p. |
artikel |
87 |
Synthesis, physicochemical properties of allopurinol derivatives and their biological activity against Trypanosoma cruzi
|
Raviolo, M.A. |
|
2013 |
69 |
C |
p. 455-464 10 p. |
artikel |
88 |
The antitumor activity of zinc(II) and copper(II) complexes with 5,7-dihalo-substituted-8-quinolinoline
|
Liu, Yan-Cheng |
|
2013 |
69 |
C |
p. 554-563 10 p. |
artikel |
89 |
The development of bis(hydroxymethyl)pyrrole analogs as bifunctional DNA cross-linking agents and their chemotherapeutic potential
|
Su, Tsann-Long |
|
2013 |
69 |
C |
p. 609-621 13 p. |
artikel |
90 |
Thermoresponsive dendrimers based on oligoethylene glycols: Design, synthesis and cytotoxic activity against MCF-7 breast cancer cells
|
Abdel-Rahman, Mona A. |
|
2013 |
69 |
C |
p. 848-854 7 p. |
artikel |