nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
1 |
4-Amino-2-arylamino-5-indoloyl/cinnamoythiazoles, analogs of topsentin-class of marine alkaloids, induce apoptosis in HeLa cells
|
Juneja, Manisha |
|
2013 |
63 |
C |
p. 474-483 10 p. |
artikel |
2 |
Aminopropylindenes derived from Grundmann's ketone as a novel chemotype of oxidosqualene cyclase inhibitors
|
Lange, Stefanie |
|
2013 |
63 |
C |
p. 758-764 7 p. |
artikel |
3 |
Analysis of the antioxidant properties of differently substituted 2- and 3-indolyl carbohydrazides and related derivatives
|
Hadjipavlou-Litina, Dimitra |
|
2013 |
63 |
C |
p. 670-674 5 p. |
artikel |
4 |
A novel insulin mimetic vanadium–flavonol complex: Synthesis, characterization and in vivo evaluation in STZ-induced rats
|
Pillai, Subramanian Iyyam |
|
2013 |
63 |
C |
p. 109-117 9 p. |
artikel |
5 |
Antibacterial oxazolidinone analogues having a N-hydroxyacetyl-substituted seven-membered [1,2,5]triazepane or [1,2,5]oxadiazepane C-ring unit
|
Suzuki, Hideyuki |
|
2013 |
63 |
C |
p. 811-825 15 p. |
artikel |
6 |
Anticancer activity of novel hybrid molecules containing 5-benzylidene thiazolidine-2,4-dione
|
Romagnoli, Romeo |
|
2013 |
63 |
C |
p. 544-557 14 p. |
artikel |
7 |
Anti-neuroinflammatory properties of synthetic cryptolepine in human neuroblastoma cells: Possible involvement of NF-κB and p38 MAPK inhibition
|
Olajide, Olumayokun A. |
|
2013 |
63 |
C |
p. 333-339 7 p. |
artikel |
8 |
Biaryl tetrazolyl ureas as inhibitors of endocannabinoid metabolism: Modulation at the N-portion and distal phenyl ring
|
Ortar, Giorgio |
|
2013 |
63 |
C |
p. 118-132 15 p. |
artikel |
9 |
Biological evaluation of bisbenzaldehydes against four Mycobacterium species
|
Cappoen, Davie |
|
2013 |
63 |
C |
p. 731-738 8 p. |
artikel |
10 |
Bivalent angiotensin II suppresses oxidative stress-induced hyper-responsiveness of angiotensin II receptor type I
|
Sungkaworn, Titiwat |
|
2013 |
63 |
C |
p. 629-634 6 p. |
artikel |
11 |
4-Bromo-2-(piperidin-1-yl)thiazol-5-yl-phenyl methanone (12b) inhibits Na+/K+-ATPase and Ras oncogene activity in cancer cells
|
Lefranc, Florence |
|
2013 |
63 |
C |
p. 213-223 11 p. |
artikel |
12 |
Coumarins hinged directly on benzimidazoles and their ribofuranosides to inhibit hepatitis C virus
|
Tsay, Shwu-Chen |
|
2013 |
63 |
C |
p. 290-298 9 p. |
artikel |
13 |
Cycloadditions and condensations as essential tools in spiropyrazoline synthesis
|
Dadiboyena, Sureshbabu |
|
2013 |
63 |
C |
p. 347-377 31 p. |
artikel |
14 |
Cytotoxic 3,4,5-trimethoxychalcones as mitotic arresters and cell migration inhibitors
|
Salum, Lívia B. |
|
2013 |
63 |
C |
p. 501-510 10 p. |
artikel |
15 |
Design and synthesis of novel 4-benzothiazole amino quinazolines Dasatinib derivatives as potential anti-tumor agents
|
Cai, Jin |
|
2013 |
63 |
C |
p. 702-712 11 p. |
artikel |
16 |
Design, modeling, synthesis and biological activity evaluation of camptothecin-linked platinum anticancer agents
|
Cincinelli, Raffaella |
|
2013 |
63 |
C |
p. 387-400 14 p. |
artikel |
17 |
Design, synthesis and antimicrobial activity of novel benzothiazole analogs
|
Singh, Manavendra K. |
|
2013 |
63 |
C |
p. 635-644 10 p. |
artikel |
18 |
Design, synthesis and antiproliferative properties of some new 5-substituted-2-iminobenzimidazole derivatives
|
Mavrova, Anelia Ts. |
|
2013 |
63 |
C |
p. 696-701 6 p. |
artikel |
19 |
Design, synthesis and biological evaluation of new classes of thieno[3,2-d]pyrimidinone and thieno[1,2,3]triazine as inhibitor of vascular endothelial growth factor receptor-2 (VEGFR-2)
|
Perspicace, Enrico |
|
2013 |
63 |
C |
p. 765-781 17 p. |
artikel |
20 |
Design, synthesis, and biological evaluation of new 2′-deoxy-2′-fluoro-4′-triazole cytidine nucleosides as potent antiviral agents
|
Wu, Jie |
|
2013 |
63 |
C |
p. 739-745 7 p. |
artikel |
21 |
Discovery of 3,3′-diindolylmethanes as potent antileishmanial agents
|
Bharate, Sandip B. |
|
2013 |
63 |
C |
p. 435-443 9 p. |
artikel |
22 |
Discovery of novel 2,6-disubstituted pyridazinone derivatives as acetylcholinesterase inhibitors
|
Xing, Weiqiang |
|
2013 |
63 |
C |
p. 95-103 9 p. |
artikel |
23 |
DNA-binding, photocleavage, cytotoxicity in vitro, apoptosis and cell cycle arrest studies of symmetric ruthenium(II) complexes
|
Xie, Yang-Yin |
|
2013 |
63 |
C |
p. 603-610 8 p. |
artikel |
24 |
Editorial board
|
|
|
2013 |
63 |
C |
p. IFC- 1 p. |
artikel |
25 |
Efficient induction of apoptosis in HeLa cells by a novel cationic porphycene photosensitizer
|
Ruiz-González, Rubén |
|
2013 |
63 |
C |
p. 401-414 14 p. |
artikel |
26 |
Efficient synthesis of new (R)-2-amino-1-butanol derived ureas, thioureas and acylthioureas and in vitro evaluation of their antimycobacterial activity
|
Dobrikov, Georgi M. |
|
2013 |
63 |
C |
p. 468-473 6 p. |
artikel |
27 |
Ester prodrugs of acyclic nucleoside thiophosphonates compared to phosphonates: Synthesis, antiviral activity and decomposition study
|
Roux, Loïc |
|
2013 |
63 |
C |
p. 869-881 13 p. |
artikel |
28 |
Evolution in medicinal chemistry of E-ring-modified Camptothecin analogs as anticancer agents
|
Huang, Qingqing |
|
2013 |
63 |
C |
p. 746-757 12 p. |
artikel |
29 |
Functionalized indoleamines as potent, drug-like inhibitors of isoprenylcysteine carboxyl methyltransferase (Icmt)
|
Ramanujulu, Pondy M. |
|
2013 |
63 |
C |
p. 378-386 9 p. |
artikel |
30 |
Further studies on bis-charged tetraazacyclophanes as potent inhibitors of small conductance Ca2+-activated K+ channels
|
Yang, Donglai |
|
2013 |
63 |
C |
p. 907-923 17 p. |
artikel |
31 |
Graphical contents list
|
|
|
2013 |
63 |
C |
p. iii-xxvi nvt p. |
artikel |
32 |
Heterocyclic bismuth carboxylates based on a diphenyl sulfone scaffold: Synthesis and antifungal activity against Saccharomyces cerevisiae
|
Murafuji, Toshihiro |
|
2013 |
63 |
C |
p. 531-535 5 p. |
artikel |
33 |
Identification of novel FLT3 kinase inhibitors
|
Pauwels, Daphnie |
|
2013 |
63 |
C |
p. 713-721 9 p. |
artikel |
34 |
Microwave-assisted synthesis of arene ruthenium(II) complexes that induce S-phase arrest in cancer cells by DNA damage-mediated p53 phosphorylation
|
Wu, Qiong |
|
2013 |
63 |
C |
p. 57-63 7 p. |
artikel |
35 |
Molecular determinants for nuclear receptors selectivity: Chemometric analysis, dockings and site-directed mutagenesis of dual peroxisome proliferator-activated receptors α/γ agonists
|
Carrieri, Antonio |
|
2013 |
63 |
C |
p. 321-332 12 p. |
artikel |
36 |
Natural sesquiterpene lactones as inhibitors of Myb-dependent gene expression: Structure–activity relationships
|
Schomburg, Caroline |
|
2013 |
63 |
C |
p. 313-320 8 p. |
artikel |
37 |
New anticancer active and selective phenylene-bisbenzothiazoles: Synthesis, antiproliferative evaluation and DNA binding
|
Racané, Livio |
|
2013 |
63 |
C |
p. 882-891 10 p. |
artikel |
38 |
New insight into adenosine receptors selectivity derived from a novel series of [5-substituted-4-phenyl-1,3-thiazol-2-yl] benzamides and furamides
|
Inamdar, Gajanan S. |
|
2013 |
63 |
C |
p. 924-934 11 p. |
artikel |
39 |
New quinazoline derivatives for telomeric G-quadruplex DNA: Effects of an added phenyl group on quadruplex binding ability
|
He, Jin-Hui |
|
2013 |
63 |
C |
p. 1-13 13 p. |
artikel |
40 |
Nonclassical antifolates, part 3: Synthesis, biological evaluation and molecular modeling study of some new 2-heteroarylthio-quinazolin-4-ones
|
Al-Omary, Fatmah A.M. |
|
2013 |
63 |
C |
p. 33-45 13 p. |
artikel |
41 |
Novel chiral ferrocenylpyrazolo[1,5-a][1,4]diazepin-4-one derivatives – Synthesis, characterization and inhibition against lung cancer cells
|
Shen, Shi-Li |
|
2013 |
63 |
C |
p. 256-268 13 p. |
artikel |
42 |
Novel (coumarin-3-yl)carbamates as selective MAO-B inhibitors: Synthesis, in vitro and in vivo assays, theoretical evaluation of ADME properties and docking study
|
Matos, Maria J. |
|
2013 |
63 |
C |
p. 151-161 11 p. |
artikel |
43 |
Novel IKKβ inhibitors discovery based on the co-crystal structure by using binding-conformation-based and ligand-based method
|
Huang, Jing-Jie |
|
2013 |
63 |
C |
p. 269-278 10 p. |
artikel |
44 |
Novel oleanolic vinyl boronates: Synthesis and antitumor activity
|
Moreira, Vânia M. |
|
2013 |
63 |
C |
p. 46-56 11 p. |
artikel |
45 |
Novel pyrimidoazepine analogs as serotonin 5-HT2A and 5-HT2C receptor ligands for the treatment of obesity
|
Yang, Ha Yun |
|
2013 |
63 |
C |
p. 558-569 12 p. |
artikel |
46 |
Novel quinolone substituted thiazolidin-4-ones as anti-inflammatory, anticancer agents: Design, synthesis and biological screening
|
Suthar, Sharad Kumar |
|
2013 |
63 |
C |
p. 589-602 14 p. |
artikel |
47 |
Optimizing the control of apoptosis by amide/triazole isosteric substitution in a constrained peptoid
|
Corredor, Miriam |
|
2013 |
63 |
C |
p. 892-896 5 p. |
artikel |
48 |
(4-Phenoxyphenyl)tetrazolecarboxamides and related compounds as dual inhibitors of fatty acid amide hydrolase (FAAH) and monoacylglycerol lipase (MAGL)
|
Holtfrerich, Angela |
|
2013 |
63 |
C |
p. 64-75 12 p. |
artikel |
49 |
Phenylpropiophenone derivatives as potential anticancer agents: Synthesis, biological evaluation and quantitative structure–activity relationship study
|
Ivković, Branka M. |
|
2013 |
63 |
C |
p. 239-255 17 p. |
artikel |
50 |
Photocytotoxicity of copper(II) complexes of curcumin and N-ferrocenylmethyl-l-amino acids
|
Goswami, Tridib K. |
|
2013 |
63 |
C |
p. 800-810 11 p. |
artikel |
51 |
Platinum(II) complexes with mono-aminophosphonate ester targeting group that induce apoptosis through G1 cell-cycle arrest: Synthesis, crystal structure and antitumour activity
|
Huang, Ke-Bin |
|
2013 |
63 |
C |
p. 76-84 9 p. |
artikel |
52 |
Polysulfones of new structural types as perspective antioxidant agents
|
Gorbunova, Marina |
|
2013 |
63 |
C |
p. 655-661 7 p. |
artikel |
53 |
Potent naphthoquinones against antimony-sensitive and -resistant Leishmania parasites: Synthesis of novel α- and nor-α-lapachone-based 1,2,3-triazoles by copper-catalyzed azide–alkyne cycloaddition
|
Guimarães, Tiago T. |
|
2013 |
63 |
C |
p. 523-530 8 p. |
artikel |
54 |
Practical synthesis of a chromene analog for use as a retinoic acid receptor alpha antagonist lead compound
|
Jetson, Rachael |
|
2013 |
63 |
C |
p. 104-108 5 p. |
artikel |
55 |
Preparation and antimalarial activity of semisynthetic lycorenine derivatives
|
Cedrón, Juan C. |
|
2013 |
63 |
C |
p. 722-730 9 p. |
artikel |
56 |
Rational design, synthesis and QSAR study of vasorelaxant active 3-pyridinecarbonitriles incorporating 1H-benzimidazol-2-yl function
|
Nofal, Zeinab M. |
|
2013 |
63 |
C |
p. 14-21 8 p. |
artikel |
57 |
Recent advances in natural products from plants for treatment of liver diseases
|
Zhang, Aihua |
|
2013 |
63 |
C |
p. 570-577 8 p. |
artikel |
58 |
Static and dynamic interactions between GALK enzyme and known inhibitors: Guidelines to design new drugs for galactosemic patients
|
Chiappori, Federica |
|
2013 |
63 |
C |
p. 423-434 12 p. |
artikel |
59 |
Structure–activity relationship of 5-chloro-2-methyl-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole analogues as 5-HT6 receptor agonists
|
Mattsson, Cecilia |
|
2013 |
63 |
C |
p. 578-588 11 p. |
artikel |
60 |
Structure–activity relationships of hybrid annonaceous acetogenins: Powerful growth inhibitory effects of their connecting groups between heterocycle and hydrophobic carbon chain bearing THF ring on human cancer cell lines
|
Kojima, Naoto |
|
2013 |
63 |
C |
p. 833-839 7 p. |
artikel |
61 |
Synthesis and antibacterial evaluation of novel pleuromutilin derivatives
|
Shang, Ruofeng |
|
2013 |
63 |
C |
p. 231-238 8 p. |
artikel |
62 |
Synthesis and anticancer activity of novel 2-pyridyl hexahyrocyclooctathieno[2,3-d]pyrimidine derivatives
|
Kassab, Asmaa E. |
|
2013 |
63 |
C |
p. 224-230 7 p. |
artikel |
63 |
Synthesis and anticancer activity of novel spiro-isoxazoline and spiro-isoxazolidine derivatives of α-santonin
|
Khazir, Jabeena |
|
2013 |
63 |
C |
p. 279-289 11 p. |
artikel |
64 |
Synthesis and antifungal activity of 3-(1,3,4-oxadiazol-5-yl)-indoles and 3-(1,3,4-oxadiazol-5-yl)methyl-indoles
|
Zhang, Ming-Zhi |
|
2013 |
63 |
C |
p. 22-32 11 p. |
artikel |
65 |
Synthesis and antiviral bioactivity of novel (1E, 4E)-1-aryl-5-(2-(quinazolin-4-yloxy)phenyl)-1,4-pentadien-3-one derivatives
|
Luo, Hui |
|
2013 |
63 |
C |
p. 662-669 8 p. |
artikel |
66 |
Synthesis and biological activities of some novel aminomethyl derivatives of 4-substituted-5-(2-thienyl)-2,4-dihydro-3H-1,2,4-triazole-3-thiones
|
Koparir, Metin |
|
2013 |
63 |
C |
p. 340-346 7 p. |
artikel |
67 |
Synthesis and biological evaluation of novel aliphatic amido-quaternary ammonium salts for anticancer chemotherapy: Part II
|
Yang, Jee Sun |
|
2013 |
63 |
C |
p. 621-628 8 p. |
artikel |
68 |
Synthesis and biological evaluation of novel pyrrolidine-2,5-dione derivatives as potential antidepressant agents. Part 1
|
Wróbel, Martyna Z. |
|
2013 |
63 |
C |
p. 484-500 17 p. |
artikel |
69 |
Synthesis and biological evaluation of oleanolic acid derivatives as PTP1B inhibitors
|
Liu, Qing-Chao |
|
2013 |
63 |
C |
p. 511-522 12 p. |
artikel |
70 |
Synthesis and evaluation of 7,8-dehydrorutaecarpine derivatives as potential multifunctional agents for the treatment of Alzheimer's disease
|
He, Yan |
|
2013 |
63 |
C |
p. 299-312 14 p. |
artikel |
71 |
Synthesis and evaluation of 2,5-di(4-aryloylaryloxymethyl)-1,3,4-oxadiazoles as anti-cancer agents
|
Gurupadaswamy, H.D. |
|
2013 |
63 |
C |
p. 536-543 8 p. |
artikel |
72 |
Synthesis and evaluation of novel marine bromopyrrole alkaloid-based hybrids as anticancer agents
|
Rane, Rajesh A. |
|
2013 |
63 |
C |
p. 793-799 7 p. |
artikel |
73 |
Synthesis and identification of β-aryloxyquinoline based diversely fluorine substituted N-aryl quinolone derivatives as a new class of antimicrobial, antituberculosis and antioxidant agents
|
Kathrotiya, Harshad G. |
|
2013 |
63 |
C |
p. 675-684 10 p. |
artikel |
74 |
Synthesis and in vitro antiproliferative effect of novel quinoline-based potential anticancer agents
|
Arafa, Reem K. |
|
2013 |
63 |
C |
p. 826-832 7 p. |
artikel |
75 |
Synthesis and pharmacokinetic profile of highly deuterated brecanavir analogs
|
Velthuisen, Emile J. |
|
2013 |
63 |
C |
p. 202-212 11 p. |
artikel |
76 |
Synthesis and selected immunological properties of substituted quino[3,2-b]benzo[1,4]thiazines
|
Jeleń, Małgorzata |
|
2013 |
63 |
C |
p. 444-456 13 p. |
artikel |
77 |
Synthesis and structure–activity relationship studies in serotonin 5-HT1A receptor agonists based on fused pyrrolidone scaffolds
|
Cappelli, Andrea |
|
2013 |
63 |
C |
p. 85-94 10 p. |
artikel |
78 |
Synthesis, antimicrobial, antiquorum-sensing, antitumor and cytotoxic activities of new series of fused [1,3,4]thiadiazoles
|
El-Gohary, Nadia S. |
|
2013 |
63 |
C |
p. 185-195 11 p. |
artikel |
79 |
Synthesis, biological activity and resistance to proteolytic digestion of new cyclic dermorphin/deltorphin analogues
|
Bańkowski, Krzysztof |
|
2013 |
63 |
C |
p. 457-467 11 p. |
artikel |
80 |
Synthesis, in vitro antitumor evaluation and DNA-binding study of novel tetrahydroquinolines and some derived tricyclic and tetracyclic ring systems
|
Faidallah, Hassan M. |
|
2013 |
63 |
C |
p. 133-143 11 p. |
artikel |
81 |
Synthesis, local anaesthetic and antiarrhythmic activities of N-alkyl derivatives of proline anilides
|
Kalinin, Dmitrii V. |
|
2013 |
63 |
C |
p. 144-150 7 p. |
artikel |
82 |
Synthesis of C- and O-prenylated tetrahydroxystilbenes and O-prenylated cinnamates and their action towards cancer cells
|
Koolaji, Nooshin |
|
2013 |
63 |
C |
p. 415-422 8 p. |
artikel |
83 |
Synthesis of decacationic [60]fullerene decaiodides giving photoinduced production of superoxide radicals and effective PDT-mediation on antimicrobial photoinactivation
|
Wang, Min |
|
2013 |
63 |
C |
p. 170-184 15 p. |
artikel |
84 |
Synthesis of 1H-1,2,3-triazole linked β-lactam–isatin bi-functional hybrids and preliminary analysis of in vitro activity against the protozoal parasite Trichomonas vaginalis
|
Raj, Raghu |
|
2013 |
63 |
C |
p. 897-906 10 p. |
artikel |
85 |
Synthesis of novel 1,3,4-trisubstituted pyrazoles as anti-inflammatory and analgesic agents
|
Ragab, Fatma A. |
|
2013 |
63 |
C |
p. 645-654 10 p. |
artikel |
86 |
Synthesis of novel triterpene and N-allylated/N-alkylated niacin hybrids as α-glucosidase inhibitors
|
Narender, Tadigoppula |
|
2013 |
63 |
C |
p. 162-169 8 p. |
artikel |
87 |
Synthesis of 3-O-propargylated betulinic acid and its 1,2,3-triazoles as potential apoptotic agents
|
Majeed, Rabiya |
|
2013 |
63 |
C |
p. 782-792 11 p. |
artikel |
88 |
Synthesis, radioiodination and in vivo screening of novel potent iodinated and fluorinated radiotracers as melanoma imaging and therapeutic probes
|
Maisonial, Aurélie |
|
2013 |
63 |
C |
p. 840-853 14 p. |
artikel |
89 |
Synthesis, structure–activity relationship analysis and kinetics study of reductive derivatives of flavonoids as Helicobacter pylori urease inhibitors
|
Xiao, Zhu-Ping |
|
2013 |
63 |
C |
p. 685-695 11 p. |
artikel |
90 |
Synthesis using microwave irradiation and antibacterial evaluation of new N,O-acetals and N,S-acetals derived from 2-amino-1,4-naphthoquinones
|
Jordão, Alessandro K. |
|
2013 |
63 |
C |
p. 196-201 6 p. |
artikel |
91 |
Thiazolidin-4-one and thiazinan-4-one derivatives analogous to rosiglitazone as potential antihyperglycemic and antidyslipidemic agents
|
Raza, Saman |
|
2013 |
63 |
C |
p. 611-620 10 p. |
artikel |
92 |
Triazolothiadiazoles and triazolothiadiazines – Biologically attractive scaffolds
|
Khan, Imtiaz |
|
2013 |
63 |
C |
p. 854-868 15 p. |
artikel |