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64 results found

no	title	author	magazine	year	volume	issue	page(s)	type
1	A dual-acting 5-HT6 receptor inverse agonist/MAO-B inhibitor displays glioprotective and pro-cognitive properties	Canale, Vittorio			208	C	p.	article
2	Advances of CCR5 antagonists: From small molecules to macromolecules	Qi, Baowen			208	C	p.	article
3	4-Amino-1,2,4-triazole-3-thione-derived Schiff bases as metallo-β-lactamase inhibitors	Gavara, Laurent			208	C	p.	article
4	2-Anilinoquinoline based arylamides as broad spectrum anticancer agents with B-RAFV600E/C-RAF kinase inhibitory effects: Design, synthesis, in vitro cell-based and oncogenic kinase assessments	El-Damasy, Ashraf K.			208	C	p.	article
5	Anti-glioma effects of 2-aminothiophene-3-carboxamide derivatives, ANO1 channel blockers	Choi, Seung-Hye			208	C	p.	article
6	Benzyl and benzoyl benzoic acid inhibitors of bacterial RNA polymerase-sigma factor interaction	Ye, Jiqing			208	C	p.	article
7	Bioactive pyrrole-based compounds with target selectivity	Li Petri, Giovanna			208	C	p.	article
8	Combined MD/QTAIM techniques to evaluate ligand-receptor interactions. Scope and limitations	Rojas, Sebastián			208	C	p.	article
9	Contents continued				208	C	p.	article
10	Corrigendum to “New desulfured troglitazone derivatives: Improved synthesis and biological evaluation” [Eur. J. Med. Chem. 187 (2020) 111939]	Dupommier, Dorian			208	C	p.	article
11	Cyclic tailor-made amino acids in the design of modern pharmaceuticals	Liu, Jiang			208	C	p.	article
12	Design and characterization of cereblon-mediated androgen receptor proteolysis-targeting chimeras	Takwale, Akshay D.			208	C	p.	article
13	Design, synthesis and biological evaluation of indole-2-one derivatives as potent BRD4 inhibitors	Xu, Yu			208	C	p.	article
14	Design, synthesis and evaluation of covalent inhibitors of DprE1 as antitubercular agents	Liu, Lingfeng			208	C	p.	article
15	Design, synthesis and molecular docking study of α-triazolylsialosides as non-hydrolyzable and potent CD22 ligands	Abdu-Allah, Hajjaj H.M.			208	C	p.	article
16	Development of triazolothiadiazine derivatives as highly potent tubulin polymerization inhibitors: Structure-activity relationship, in vitro and in vivo study	Ma, Weifeng			208	C	p.	article
17	Discovery of 5-bromo-4-phenoxy-N-phenylpyrimidin-2-amine derivatives as novel ULK1 inhibitors that block autophagy and induce apoptosis in non-small cell lung cancer	Sun, Dejuan			208	C	p.	article
18	Discovery of novel quinazoline derivatives as potent PI3Kδ inhibitors with high selectivity	Teng, Yu			208	C	p.	article
19	Discovery of novel VX-809 hybrid derivatives as F508del-CFTR correctors by molecular modeling, chemical synthesis and biological assays	Parodi, Alice			208	C	p.	article
20	Discovery of potent small molecule PROTACs targeting mutant EGFR	Zhao, Hong-Yi			208	C	p.	article
21	Discovery of the first potent and selective αvβ5 integrin inhibitor based on an amide-containing core	Lippa, Rhys A.			208	C	p.	article
22	Editorial Board				208	C	p.	article
23	Effective anti-aromatase therapy to battle against estrogen-mediated breast cancer: Comparative SAR/QSAR assessment on steroidal aromatase inhibitors	Adhikari, Nilanjan			208	C	p.	article
24	Efficient chemoenzymatic synthesis of fluorinated sialyl Thomsen–Friedenreich antigens and investigation of their characteristics	Li, Tingshen			208	C	p.	article
25	FabI (enoyl acyl carrier protein reductase) - A potential broad spectrum therapeutic target and its inhibitors	Rana, Preeti			208	C	p.	article
26	Factor XII/XIIa inhibitors: Their discovery, development, and potential indications	Davoine, Clara			208	C	p.	article
27	Graphical abstract TOC				208	C	p.	article
28	Graphical abstract TOC				208	C	p.	article
29	Hydroxamate siderophores: Natural occurrence, chemical synthesis, iron binding affinity and use as Trojan horses against pathogens	Al Shaer, Danah			208	C	p.	article
30	Hydroxy-corrole and its gallium(III) complex as new photosensitizer for photodynamic therapy against breast carcinoma	Sun, Yan-Mei			208	C	p.	article
31	Induced protein degradation of histone deacetylases 3 (HDAC3) by proteolysis targeting chimera (PROTAC)	Cao, Fangyuan			208	C	p.	article
32	β-lactam antibiotics: An overview from a medicinal chemistry perspective	Lima, Lidia Moreira			208	C	p.	article
33	Modern trends in diuretics development	Titko, Tetiana			208	C	p.	article
34	Multiple biological active 4-aminopyrazoles containing trifluoromethyl and their 4-nitroso-precursors: Synthesis and evaluation	Burgart, Yanina V.			208	C	p.	article
35	New indolylarylsulfone non-nucleoside reverse transcriptase inhibitors show low nanomolar inhibition of single and double HIV-1 mutant strains	Nalli, Marianna			208	C	p.	article
36	New one-pot synthesis of anti-tuberculosis compounds inspired on isoniazid	Ghiano, Diego G.			208	C	p.	article
37	Novel 2-indolinone thiazole hybrids as sunitinib analogues: Design, synthesis, and potent VEGFR-2 inhibition with potential anti-renal cancer activity	Mahmoud, Huda K.			208	C	p.	article
38	Novel monomolecular derivatives of the anti-HIV-1 G-quadruplex-forming Hotoda’s aptamer containing inversion of polarity sites	Virgilio, Antonella			208	C	p.	article
39	Novel quinazolinone inhibitors of the Pseudomonas aeruginosa quorum sensing transcriptional regulator PqsR	Grossman, Scott			208	C	p.	article
40	One molecule two goals: A selective P-glycoprotein modulator increases drug transport across gastro-intestinal barrier and recovers doxorubicin toxicity in multidrug resistant cancer cells	Contino, Marialessandra			208	C	p.	article
41	Optimization of pyrazolo[1,5-a]pyrimidines lead to the identification of a highly selective casein kinase 2 inhibitor	Krämer, Andreas			208	C	p.	article
42	1,3-Oxazine-2-one derived dual-targeted molecules against replicating and non-replicating forms of Mycobacterium tuberculosis	Velappan, Anand Babu			208	C	p.	article
43	Phosphorus dendrimers as powerful nanoplatforms for drug delivery, as fluorescent probes and for liposome interaction studies: A concise overview	Shcharbin, Dzmitry			208	C	p.	article
44	Recent advances of podophyllotoxin/epipodophyllotoxin hybrids in anticancer activity, mode of action, and structure-activity relationship: An update (2010–2020)	Xiao, Jiaqi			208	C	p.	article
45	Recent progress on HDAC inhibitors with dual targeting capabilities for cancer treatment	Peng, Xiaopeng			208	C	p.	article
46	Research progress of mTOR inhibitors	Chen, Yifan			208	C	p.	article
47	Selective targeting of the αC and DFG-out pocket in p38 MAPK	Röhm, Sandra			208	C	p.	article
48	Some thermodynamic effects of varying nonpolar surfaces in protein-ligand interactions	Cramer, David L.			208	C	p.	article
49	Structural optimization of pyrazolo[1,5-a]pyrimidine derivatives as potent and highly selective DPP-4 inhibitors	Shen, Jian			208	C	p.	article
50	Structure-activity relationships for a series of (Bis(4-fluorophenyl)methyl)sulfinylethyl-aminopiperidines and -piperidine amines at the dopamine transporter: Bioisosteric replacement of the piperazine improves metabolic stability	Giancola, JoLynn B.			208	C	p.	article
51	Structure–activity relationship study of novel quinazoline-based 1,6-naphthyridinones as MET inhibitors with potent antitumor efficacy	Zhuo, Lin-Sheng			208	C	p.	article
52	Structure-activity relationship study of tryptophan-based butyrylcholinesterase inhibitors	Meden, Anže			208	C	p.	article
53	Synthesis and biological evaluation of organoselenium (NSAIDs-SeCN and SeCF3) derivatives as potential anticancer agents	He, Xianran			208	C	p.	article
54	Synthesis and evaluation of thiophene based small molecules as potent inhibitors of Mycobacterium tuberculosis	Meena, Chhuttan L.			208	C	p.	article
55	Synthesis and in vitro and in vivo biological evaluation of novel derivatives of flexicaulin A as antiproliferative agents	Huo, Jun-Feng			208	C	p.	article
56	Synthesis, bioevaluation and docking studies of some 2-phenyl-1H-benzimidazole derivatives as anthelminthic agents against the nematode Teladorsagia circumcincta	Escala, Nerea			208	C	p.	article
57	Synthesis, molecular modeling, in vivo study and anticancer activity against prostate cancer of (+) (S)-naproxen derivatives	Birgül, Kaan			208	C	p.	article
58	Synthesis of biphenyl oxazole derivatives via Suzuki coupling and biological evaluations as nucleotide pyrophosphatase/phosphodiesterase-1 and -3 inhibitors	Ahmad, Haseen			208	C	p.	article
59	Synthesis of ticagrelor analogues belonging to 1,2,3-triazolo[4,5-d]pyrimidines and study of their antiplatelet and antibacterial activity	Goffin, Eric			208	C	p.	article
60	Systematic ‘foldamerization’ of peptide inhibiting p53-MDM2/X interactions by the incorporation of trans- or cis-2-aminocyclopentanecarboxylic acid residues	Fortuna, Paulina			208	C	p.	article
61	Targeting histone demethylase KDM5B for cancer treatment	Fu, Yun-Dong			208	C	p.	article
62	The endocannabinoid system dual-target ligand N-cycloheptyl-1,2-dihydro-5-bromo-1-(4-fluorobenzyl)-6-methyl-2-oxo-pyridine-3-carboxamide improves disease severity in a mouse model of multiple sclerosis	Arena, Chiara			208	C	p.	article
63	Triphenylethylene analogues: Design, synthesis and evaluation of antitumor activity and topoisomerase inhibitors	Rani, Sudesh			208	C	p.	article
64	Unraveling the anti-influenza effect of flavonoids: Experimental validation of luteolin and its congeners as potent influenza endonuclease inhibitors	Zima, Václav			208	C	p.	article

64 results found

Koninklijke Bibliotheek - National Library of the Netherlands