nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
1 |
An evaluation of Minor Groove Binders as anti-fungal and anti-mycobacterial therapeutics
|
Scott, Fraser J. |
|
2017 |
136 |
C |
p. 561-572 12 p. |
artikel |
2 |
Antibacterial activity and mechanism of action of the benzazole acrylonitrile-based compounds: In vitro, spectroscopic, and docking studies
|
AlNeyadi, Shaikha S. |
|
2017 |
136 |
C |
p. 270-282 13 p. |
artikel |
3 |
Bioactivity-guided mixed synthesis accelerate the serendipity in lead optimization: Discovery of fungicidal homodrimanyl amides
|
Li, Dangdang |
|
2017 |
136 |
C |
p. 114-121 8 p. |
artikel |
4 |
Concise synthesis and antiproliferative activity evaluation of ellipticine quinone and its analogs
|
Nishiyama, Takashi |
|
2017 |
136 |
C |
p. 1-13 13 p. |
artikel |
5 |
Design and synthesis of bis(indolyl)ketohydrazide-hydrazones: Identification of potent and selective novel tubulin inhibitors
|
Tantak, Mukund P. |
|
2017 |
136 |
C |
p. 184-194 11 p. |
artikel |
6 |
Designing multi-targeted agents: An emerging anticancer drug discovery paradigm
|
Fu, Rong-geng |
|
2017 |
136 |
C |
p. 195-211 17 p. |
artikel |
7 |
Design, synthesis and antimicrobial evaluation of novel benzimidazole-incorporated sulfonamide analogues
|
Zhang, Hui-Zhen |
|
2017 |
136 |
C |
p. 165-183 19 p. |
artikel |
8 |
Design, synthesis and biological evaluation of nitrogen-containing macrocyclic bisbibenzyl derivatives as potent anticancer agents by targeting the lysosome
|
Sun, Bin |
|
2017 |
136 |
C |
p. 603-618 16 p. |
artikel |
9 |
Design, synthesis and biological evaluation of uncharged catechol derivatives as selective inhibitors of PTP1B
|
Li, Xiang-Qian |
|
2017 |
136 |
C |
p. 348-359 12 p. |
artikel |
10 |
Design, synthesis and evaluation of azaacridine derivatives as dual-target EGFR and Src kinase inhibitors for antitumor treatment
|
Cui, Zhishan |
|
2017 |
136 |
C |
p. 372-381 10 p. |
artikel |
11 |
Design, synthesis and primary biological evaluation of the novel 2-pyridone derivatives as potent non-nucleoside HBV inhibitors
|
Jia, Haiyong |
|
2017 |
136 |
C |
p. 144-153 10 p. |
artikel |
12 |
Design, synthesis, molecular docking and cytotoxic evaluation of novel 2-furybenzimidazoles as VEGFR-2 inhibitors
|
Abdullaziz, Mona A. |
|
2017 |
136 |
C |
p. 315-329 15 p. |
artikel |
13 |
Discorhabdin alkaloids from Antarctic Latrunculia spp. sponges as a new class of cholinesterase inhibitors
|
Botić, Tanja |
|
2017 |
136 |
C |
p. 294-304 11 p. |
artikel |
14 |
Discovery and characterization of selective human sphingomyelin synthase 2 inhibitors
|
Adachi, Ryutaro |
|
2017 |
136 |
C |
p. 283-293 11 p. |
artikel |
15 |
Discovery of a potent dual ALK and EGFR T790M inhibitor
|
Jang, Jaebong |
|
2017 |
136 |
C |
p. 497-510 14 p. |
artikel |
16 |
Discovery of efficient stimulators for adult hippocampal neurogenesis based on scaffolds in dragon's blood
|
Liang, Jian-Hua |
|
2017 |
136 |
C |
p. 382-392 11 p. |
artikel |
17 |
Editorial board
|
|
|
2017 |
136 |
C |
p. IFC- 1 p. |
artikel |
18 |
Efficient click chemistry towards fatty acids containing 1,2,3-triazole: Design and synthesis as potential antifungal drugs for Candida albicans
|
Fu, Nina |
|
2017 |
136 |
C |
p. 596-602 7 p. |
artikel |
19 |
Formation of platinum (II) as a six member ring for sustained polymeric delivery
|
Senadheera, Sanjeewa N. |
|
2017 |
136 |
C |
p. 452-456 5 p. |
artikel |
20 |
Graphical contents list
|
|
|
2017 |
136 |
C |
p. iii-xvi nvt p. |
artikel |
21 |
Improved synthesis and comparative analysis of the tool properties of new and existing D-ring modified (S)-blebbistatin analogs
|
Verhasselt, Sigrid |
|
2017 |
136 |
C |
p. 85-103 19 p. |
artikel |
22 |
Indole carboxylic acid esters of melampomagnolide B are potent anticancer agents against both hematological and solid tumor cells
|
Bommagani, Shobanbabu |
|
2017 |
136 |
C |
p. 393-405 13 p. |
artikel |
23 |
Indole-coumarin-thiadiazole hybrids: An appraisal of their MCF-7 cell growth inhibition, apoptotic, antimetastatic and computational Bcl-2 binding potential
|
Kamath, Pooja R. |
|
2017 |
136 |
C |
p. 442-451 10 p. |
artikel |
24 |
Investigation of pyrazolo-sulfonamides as putative small molecule oxytocin receptor agonists
|
Katte, Timothy A. |
|
2017 |
136 |
C |
p. 330-333 4 p. |
artikel |
25 |
LL-37-derived short antimicrobial peptide KR-12-a5 and its d-amino acid substituted analogs with cell selectivity, anti-biofilm activity, synergistic effect with conventional antibiotics, and anti-inflammatory activity
|
Kim, Eun Young |
|
2017 |
136 |
C |
p. 428-441 14 p. |
artikel |
26 |
Methyllysine binding domains: Structural insight and small molecule probe development
|
Teske, Kelly A. |
|
2017 |
136 |
C |
p. 14-35 22 p. |
artikel |
27 |
Molecular insight into specific 14-3-3 modulators: Inhibitors and stabilisers of protein–protein interactions of 14-3-3
|
Hartman, Alwin M. |
|
2017 |
136 |
C |
p. 573-584 12 p. |
artikel |
28 |
Nanomolar anti-sickling compounds identified by ligand-based pharmacophore approach
|
Paz, Odailson Santos |
|
2017 |
136 |
C |
p. 487-496 10 p. |
artikel |
29 |
New cycloartane type-triterpenoids from the areal parts of Caragana sukiensis and their biological activities
|
Reddy, S. Divya |
|
2017 |
136 |
C |
p. 74-84 11 p. |
artikel |
30 |
Nitric oxide-releasing derivatives of brefeldin A as potent and highly selective anticancer agents
|
Tian, Kangtao |
|
2017 |
136 |
C |
p. 131-143 13 p. |
artikel |
31 |
Novel amidino substituted benzimidazole and benzothiazole benzo[b]thieno-2-carboxamides exert strong antiproliferative and DNA binding properties
|
Cindrić, Maja |
|
2017 |
136 |
C |
p. 468-479 12 p. |
artikel |
32 |
Novel anti-inflammatory agents targeting CXCR4: Design, synthesis, biological evaluation and preliminary pharmacokinetic study
|
Bai, Renren |
|
2017 |
136 |
C |
p. 360-371 12 p. |
artikel |
33 |
Novel 1-(7-ethoxy-1-benzofuran-2-yl) substituted chalcone derivatives: Synthesis, characterization and anticancer activity
|
Coskun, Demet |
|
2017 |
136 |
C |
p. 212-222 11 p. |
artikel |
34 |
Novel Imidazo[4,5-c][1,2,6]thiadiazine 2,2-dioxides as antiproliferative trypanosoma cruzi drugs: Computational screening from neural network, synthesis and in vivo biological properties
|
Guerra, Angela |
|
2017 |
136 |
C |
p. 223-234 12 p. |
artikel |
35 |
Novel propanamides as fatty acid amide hydrolase inhibitors
|
Deplano, Alessandro |
|
2017 |
136 |
C |
p. 523-542 20 p. |
artikel |
36 |
Pharmacophore guided discovery of small-molecule interleukin 15 inhibitors
|
Żyżyńska-Granica, Barbara |
|
2017 |
136 |
C |
p. 543-547 5 p. |
artikel |
37 |
4-Phenyl quinoline derivatives as potential serotonin receptor ligands with antiproliferative activity
|
Joshi, Pranaya V. |
|
2017 |
136 |
C |
p. 246-258 13 p. |
artikel |
38 |
Quinazoline based α1-adrenoreceptor antagonists with potent antiproliferative activity in human prostate cancer cell lines
|
Maestri, Valentina |
|
2017 |
136 |
C |
p. 259-269 11 p. |
artikel |
39 |
Rational design, synthesis and biological screening of triazine-triazolopyrimidine hybrids as multitarget anti-Alzheimer agents
|
Jameel, Ehtesham |
|
2017 |
136 |
C |
p. 36-51 16 p. |
artikel |
40 |
Recent developments of coumarin-containing derivatives and their anti-tubercular activity
|
Hu, Yuan-Qiang |
|
2017 |
136 |
C |
p. 122-130 9 p. |
artikel |
41 |
Rhodium-catalyzed C-H bond activation for the synthesis of quinonoid compounds: Significant Anti-Trypanosoma cruzi activities and electrochemical studies of functionalized quinones
|
Jardim, Guilherme A.M. |
|
2017 |
136 |
C |
p. 406-419 14 p. |
artikel |
42 |
Rigid aromatic linking moiety in cationic lipids for enhanced gene transfection efficiency
|
Wang, Bing |
|
2017 |
136 |
C |
p. 585-595 11 p. |
artikel |
43 |
Ruthenium(II) complexes of saccharin with dipyridoquinoxaline and dipyridophenazine: Structures, biological interactions and photoinduced DNA damage activity
|
Kumar, Priyaranjan |
|
2017 |
136 |
C |
p. 52-62 11 p. |
artikel |
44 |
Structure-activity relationship study of the tumour-targeting peptide A20FMDV2 via modification of Lys16, Leu13, and N- and/or C-terminal functionality
|
Hung, Kuo-yuan |
|
2017 |
136 |
C |
p. 154-164 11 p. |
artikel |
45 |
Structure-based virtual screening and optimization of modulators targeting Hsp90-Cdc37 interaction
|
Wang, Lei |
|
2017 |
136 |
C |
p. 63-73 11 p. |
artikel |
46 |
Synthesis and in vitro evaluation of new fluorinated quinoline derivatives with high affinity for PDE5: Towards the development of new PET neuroimaging probes
|
Liu, Jianrong |
|
2017 |
136 |
C |
p. 548-560 13 p. |
artikel |
47 |
Synthesis and pharmacological evaluation of neurosteroid photoaffinity ligands
|
Savechenkov, Pavel Y. |
|
2017 |
136 |
C |
p. 334-347 14 p. |
artikel |
48 |
Synthesis and preclinical evaluation of [11C]MA-PB-1 for in vivo imaging of brain monoacylglycerol lipase (MAGL)
|
Ahamed, Muneer |
|
2017 |
136 |
C |
p. 104-113 10 p. |
artikel |
49 |
Synthesis and structure-activity relationships of novel fused ring analogues of Q203 as antitubercular agents
|
Kang, Sunhee |
|
2017 |
136 |
C |
p. 420-427 8 p. |
artikel |
50 |
Synthesis of novel indole derivatives as promising DNA-binding agents and evaluation of antitumor and antitopoisomerase I activities
|
Lafayette, Elizabeth Almeida |
|
2017 |
136 |
C |
p. 511-522 12 p. |
artikel |
51 |
The discovery of novel, potent ERR-alpha inverse agonists for the treatment of triple negative breast cancer
|
Du, Yongli |
|
2017 |
136 |
C |
p. 457-467 11 p. |
artikel |
52 |
The relevance of Ki calculation for bi-substrate enzymes illustrated by kinetic evaluation of a novel lysine (K) acetyltransferase 8 inhibitor
|
Wapenaar, Hannah |
|
2017 |
136 |
C |
p. 480-486 7 p. |
artikel |
53 |
Thiosemicarbazones and 4-thiazolidinones indole-based derivatives: Synthesis, evaluation of antiproliferative activity, cell death mechanisms and topoisomerase inhibition assay
|
de Oliveira, Jamerson Ferreira |
|
2017 |
136 |
C |
p. 305-314 10 p. |
artikel |
54 |
Two novel dinuclear ellipsoid Ni(II) and Co(II) complexes bridged by 4,5-bis(pyrazol-1-yl)phthalic acid: Synthesis, structural characterization and biological evaluation
|
Gao, Enjun |
|
2017 |
136 |
C |
p. 235-245 11 p. |
artikel |